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2-ethyl-4-{1-[2-(2-fluorophenoxy)ethyl]-1H-imidazol-2-yl}pyrimidine
5-chloro-4-({3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}methyl)-2-methoxyphenol
[(4-methyl-1H-imidazol-5-yl)methyl]({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(pyridin-3-ylmethyl)amine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-1,3-benzothiazole-6-carboxamide
2-methoxy-1-{1'-[(4-methylphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-3-phenylpyrrolidin-3-ol
N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-3-(piperidine-1-carbonyl)pyrazine-2-carboxamide
N4-[(4-chlorophenyl)methyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N,1,3,6-tetramethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(cyclohexylmethyl)-9-ethyl-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
methyl 4-{4-[3-(morpholine-4-carbonyl)phenoxy]piperidin-1-yl}-4-oxobutanoate
N-[(3S,4R)-1-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
N2-[(2,3-dimethyl-1H-indol-5-yl)methyl]-N4-ethylpyrimidine-2,4-diamine
3,7-dimethyl-11-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-3,7,11-triazaspiro[5.6]dodecane
1-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(3-methoxybenzoyl)piperazine
1-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-(4-methylphenyl)piperazine
5-(4-methanesulfonyl-1,4-diazepane-1-carbonyl)-1-methyl-1H-1,3-benzodiazole
4,6-dimethyl-1-(2-{[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]amino}ethyl)-1,2-dihydropyrimidin-2-one
N-[2-(3,5-dimethylphenoxy)ethyl]-N-methyl-4-(4-methylpiperazin-1-yl)pentanamide
3-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-1-[2-(oxolan-2-ylmethoxy)phenyl]urea
ethyl 4-{[({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}-1H-pyrazole-3-carboxylate
methyl[2-(pyridin-2-yl)ethyl]{[3-({1-[4-(trifluoromethyl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}amine
7-fluoro-3-[({1H-pyrrolo[2,3-b]pyridin-6-yl}amino)methyl]-1,2-dihydroquinolin-2-one
4-{[(2-methoxyethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]carbamoyl]amino}-N,3-dimethylbenzamide
4-{[3-(diethylamino)pyrrolidin-1-yl]methyl}-N-(1-methyl-1H-pyrazol-4-yl)benzamide
5-ethyl-2,3-dimethyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
ethyl 3-(2-phenylethyl)-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidine-3-carboxylate
6-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-1,2-dihydropyridin-2-one
4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-[2-oxo-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]piperazin-2-one
N-methyl-N-(quinolin-8-ylmethyl)-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
1-[4-(3-chloro-4-methoxyphenyl)phenyl]-2-(morpholin-4-yl)ethan-1-ol
[2-fluoro-5-(quinolin-2-yl)phenyl]methanol
N-{[5-(benzylsulfanyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-6-[3-(trifluoromethyl)benzoyl]-6-azaspiro[2.5]octane-1-carboxamide
4-[(4-methylphenyl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-amino-4-[5-(hydroxymethyl)furan-2-yl]-5H,6H,7H-pyrrolo[2,3-h]quinoline-3-carbonitrile
N-[2-(2-ethoxyphenyl)ethyl]-2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
2-[(4-hydroxyquinazolin-2-yl)sulfanyl]-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
N-methyl-6-(2-methylphenyl)-N-[2-(morpholin-4-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
1-[1-(4-methoxy-3-methylbenzoyl)piperidin-3-yl]-4-(2-methoxyphenyl)piperazine
1-[2-methoxy-4-({[3-(methylsulfanyl)propyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
2-(2-ethylpiperidin-1-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
N-methyl-2-{4-[3-(1H-pyrazol-1-yl)phenyl]-1H-pyrazol-1-yl}acetamide
3-(3-methylphenyl)-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-1H-pyrazole-4-carboxamide
2-{[4-(3-chlorophenyl)-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
4-[2-(4-methyl-1,4-diazepane-1-carbonyl)-1-benzofuran-5-yl]-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-4-ol
2-[1-(3-methylbut-2-en-1-yl)-4-(quinolin-8-ylmethyl)piperazin-2-yl]ethan-1-ol
2-(ethylamino)-N,4-dimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1,3-thiazole-5-carboxamide