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3-[(propan-2-yl)sulfamoyl]-5-(quinolin-6-yl)benzoic acid
1-ethyl-N-methyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-N-(thiophen-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{4-[2-(3,4-dimethoxyphenyl)-5-fluoro-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-methylpropan-1-one
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetamide
[(2-ethoxyphenyl)methyl][2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}-1-(3-propanoylpiperidin-1-yl)propan-1-one
1-methyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
2-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptane-2-carbonyl]-3,5,7-trimethyl-1H-indole
1-(4-fluorophenyl)-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}cyclopropane-1-carboxamide
N-(1-hydroxybutan-2-yl)-6-oxo-N-(pyridin-2-ylmethyl)-1,6-dihydropyridine-3-carboxamide
N-(3-ethyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-4-(4-methyl-1H-pyrazol-3-yl)piperidine-1-carboxamide
1-{2-[(3-fluorophenyl)methyl]morpholin-4-yl}-3-(methylsulfanyl)propan-1-one
2-cyclopropyl-9-[(4-oxo-4H-chromen-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(1H-indol-3-yl)-1-{5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}ethan-1-one
7-[(4-fluorophenyl)methyl]-N-(furan-2-ylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
8-fluoro-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}quinoline-2-carboxamide
(2S,4S)-1-methyl-4-(4-oxo-3,4-dihydrophthalazine-1-amido)pyrrolidine-2-carboxylic acid
5-(1-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)-1-methyl-1H-1,2,4-triazole
8-{[2-(furan-2-yl)phenyl]methyl}-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{4-[1-cyclohexyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]phenoxy}acetamide
2,7,8-trimethyl-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}quinoline-4-carboxamide
4-chloro-N-[1-(4-chlorophenyl)cyclobutyl]-1-methyl-1H-pyrazole-3-carboxamide
3-(1-cyclopentanecarbonylpiperidin-4-yl)-N-(3-methylphenyl)propanamide
N-[3-(4-fluorophenyl)phenyl]-1-(pyridine-3-carbonyl)piperidine-3-carboxamide
3-methyl-2-{4-[(2-propylpyrimidin-5-yl)methyl]piperazin-1-yl}quinoline
2-{3-oxo-9-[4-(trifluoromethyl)pyridin-2-yl]-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
3-(2-fluorophenyl)-5-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-[4-(4-cyclobutyl-6-methylpyrimidin-2-yl)morpholin-2-yl]ethan-1-amine
6-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}pyrimidin-4-amine
1-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-5-oxopyrrolidine-3-carboxylic acid
N-(2-hydroxyethyl)-N-methyl-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}acetamide
2-methyl-3-[3-(piperidin-1-yl)azetidine-1-carbonyl]-N-(pyridin-3-ylmethyl)aniline
1-ethyl-3-[4-(furan-2-yl)phenyl]-1-(oxan-4-yl)urea
2-oxo-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-1,2-dihydroquinoline-4-carboxamide
1-{1-[1-(3-chloro-4-fluorobenzoyl)piperidin-4-yl]ethyl}-4-methylpiperazine
2-methyl-1-{4-[4-(5-propylpyrimidin-4-yl)piperazin-1-yl]piperidin-1-yl}propan-1-one
3-(2-{4-[hydroxy(pyridin-2-yl)methyl]piperidin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
N-({7-[(2,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-2-carboxamide
N-[(2R,3R)-2-methoxy-1'-[(2-methoxyphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-3-carboxamide
6-cyclopentyl-2-methoxy-3-{[(4,4,4-trifluorobutan-2-yl)amino]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
[(2-cyclohexylpyrimidin-5-yl)methyl](methyl)[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amine
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(1,3-dihydroxy-2-methylpropan-2-yl)acetamide
2-[3-(methoxymethyl)pyrrolidin-1-yl]-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridine
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-(2,3-dihydro-1H-inden-1-yl)propanamide
8-[2-(2-hydroxyphenoxy)acetyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-methyl-3-[5-(2-methyloxolane-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]-1,2-oxazole
4-[3-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-6-methylpyrimidin-2-amine
3-methyl-N-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-4-yl)ethyl]-5-(phenoxymethyl)furan-2-carboxamide
N-[3-(furan-2-amido)-4-methoxyphenyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide