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1-[(5-acetylthiophen-3-yl)methyl]-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[2-(3-fluorophenyl)ethyl]piperidine
4-{[4-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperazin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}spiro[azepane-4,2'-chromene]
4-(prop-2-en-1-yl)-3-[1-(propan-2-yloxy)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(4-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl]-4-(pyridin-3-yl)piperidin-4-ol
N-(2,3-dihydro-1H-inden-2-yl)-3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}propanamide
N-[(1R,2S)-2-(methoxymethyl)cyclopentyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
3-(4-{1-[(2-methoxypyridin-3-yl)methyl]pyrrolidin-3-yl}pyridin-2-yl)phenol
6-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
N-benzyl-N-(1,3-thiazol-2-ylmethyl)pyrrolidine-2-carboxamide
6-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-N,N-dimethylpyrazine-2-carboxamide
2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-[4-(morpholin-4-yl)piperidin-1-yl]ethan-1-one
N-ethyl-2-(7-methyl-3-oxo-3,4-dihydro-2H-1,4-benzothiazin-4-yl)-N-(oxan-4-ylmethyl)acetamide
(3R,5S)-N3-[(4,6-dimethylpyrimidin-2-yl)methyl]-N5-(4-methylphenyl)piperidine-3,5-dicarboxamide
N3-(cyclohexylmethyl)-1-cyclopropyl-N5-[(1-methylpiperidin-3-yl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-methyl-N-{[4-(2-methylpropyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-1,3-thiazole-4-carboxamide
4-methyl-2-(propan-2-yl)-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,3-thiazole-5-carboxamide
2-(2-chloro-4-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}phenoxy)acetamide
N-(oxan-4-ylmethyl)-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
1-[(2-fluorophenyl)methyl]-N-methyl-N-[(3-methylthiophen-2-yl)methyl]-6-oxopiperidine-3-carboxamide
(4aR,8aR)-2-cyclobutanecarbonyl-7-[(4-methylnaphthalen-1-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
N3-cyclooctyl-N5-(3-methoxypropyl)-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-[2-methoxy-4-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(2-hydroxyethyl)-5-methoxybenzamide
(4aR,7aS)-1-acetyl-4-(4-methyl-1,3-thiazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[(4-fluorophenyl)methyl]-N-[2-(pyrazin-2-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
N-[(3-chlorophenyl)methyl]-3-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-propylpropanamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]-N-(propan-2-yl)propanamide
2-(3-hydroxypiperidin-1-yl)-1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]ethan-1-one
(2R,3R)-3-(1,2,3,6-tetrahydropyridin-1-yl)-1'-(1H-1,2,4-triazole-5-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-[2-(pyrimidin-5-yl)pyrimidin-4-yl]piperidin-3-ol
N-methyl-N-[3-(oxolan-2-yl)propyl]-1-propylpiperidin-4-amine
(2,1,3-benzoxadiazol-4-ylmethyl)(methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
2-{1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-3-yl}-1H-1,3-benzodiazole
3-amino-N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)thiophene-2-carboxamide
N-[2-(4-ethyl-1,3-thiazol-2-yl)ethyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
(1S,6R)-9-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
1-[(4-{[1-(furan-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]-4-phenylpiperidine
1-ethyl-5-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1H-1,2,4-triazole
1-(propan-2-yl)-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}piperidine-4-carboxamide
2-{[5-(pyridin-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-(pyrimidin-4-yl)morpholine
N,N,4-trimethyl-3-{[(2-phenylpropan-2-yl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
7-(1-benzothiophen-3-yl)-4-(2-methyl-1,3-thiazole-4-carbonyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-cyclopropyl-2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-{6-[(propan-2-yl)amino]pyrimidin-4-yl}pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-(4-fluorophenyl)-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]cyclopropane-1-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(2-hydroxyethyl)pyrrolidin-3-yl]-4-methoxypiperidine-1-sulfonamide