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1-{4-[(3-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-1,2-oxazol-5-yl)methoxy]phenyl}ethan-1-one
(2S,4R)-4-amino-1-(4-methyl-5-phenylthiophene-2-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
5-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one
7-(2-methoxyethyl)-2-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
1-[1-(cyclohex-1-en-1-yl)ethyl]-3-[3-methoxy-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
3-[2-methyl-5-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-1-[1-(3-methylpyridin-2-yl)propan-2-yl]urea
5-{[4-ethyl-5-oxo-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]methyl}-N-methylfuran-2-carboxamide
2-(4-fluorophenyl)-N-[2-(7-{[4-(methylsulfanyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]acetamide
1-{[5-(3-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-3-[1-(3-methylbutyl)-1H-pyrazol-5-yl]urea
N-tert-butyl-1-(3-methylbutyl)-4-oxo-5-[4-(pyridin-4-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
1-methanesulfonyl-N-[1-(thiophen-2-yl)propyl]piperidin-4-amine
1-{2-[(3-fluorophenyl)methyl]morpholin-4-yl}-3-(3-methoxyphenyl)propan-1-one
N3-(cyclohexylmethyl)-1-cyclopropyl-N5-[furan-2-yl(phenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-(pyrrolidine-1-carbonyl)-2-[1-(2,2,2-trifluoroethyl)-1H-pyrazol-4-yl]quinoline
N-[2-(azepan-1-yl)-2-phenylethyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(4-tert-butylphenyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-ethyl-4-[({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]piperidine-1-carboxamide
3-{1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]piperidin-3-yl}benzoic acid
methyl 5-(2-methyl-1H-1,3-benzodiazole-4-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-cyclopropanecarbonyl-N-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]piperidine-4-carboxamide
(3S,9aR)-8-(3-fluoro-4-methylbenzoyl)-3-(1H-indol-3-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[(1S)-1-phenylethyl]urea
2-{4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}pyridine-4-carbonitrile
5-[3-(methoxymethyl)phenyl]-3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
N-[2-(2,3-dichlorophenyl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-methyl-1,2,3-thiadiazole-5-carboxamide
(1R,5R)-3-benzoyl-6-(1-benzofuran-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-(methoxymethyl)-1-{[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}piperidine
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]pyridine-2-carboxamide
2-(1H-imidazol-2-yl)-8-methoxyquinoline
3-[2-oxo-2-(piperidin-1-yl)ethyl]-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidine-2,5-dione
2-{4-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]morpholin-3-yl}-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]acetamide
2-({3-[2-(3-methoxyphenyl)pyridin-4-yl]pyrrolidin-1-yl}methyl)benzoic acid
(2S,4S)-4-{[(3,4-difluorophenyl)methyl]amino}-N-ethyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[2-(1H-imidazol-1-yl)ethyl]methylamine
2-[(2S,3R)-2-amino-3-hydroxybutanoyl]-N-(5-methyl-1,2-oxazol-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-{1-[6-(2,3-dihydro-1H-isoindol-2-yl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
N-[3-(propan-2-yloxy)propyl]-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
methyl 2-[(1-methoxypropan-2-yl)sulfamoyl]-6-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-{4-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
1-cyclopentyl-4-[({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}(methyl)amino)methyl]pyrrolidin-2-one
3-(3-fluoro-4-methoxybenzoyl)-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidine
N,N-diethyl-1-[2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]pyrrolidin-3-amine
5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-2,1,3-benzoxadiazole
1-[(3,5-dimethoxyphenyl)methyl]-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,4S)-1-(4-methoxybenzoyl)-4-(4-methoxypiperidin-1-yl)pyrrolidin-3-ol
4-[5-({[(1-ethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-1,2,4-oxadiazol-3-yl]benzoic acid
3-[(1-acetylpiperidin-4-yl)oxy]-N-(6-hydroxy-6-methylheptan-2-yl)-4-methoxybenzamide
5-benzyl-4-[1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]-2-methylpyrimidine
methyl 6-(4-fluorobenzoyl)-2-[(3-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate