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N-methyl-2-(2-oxoazepan-1-yl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)acetamide
[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)(oxolan-3-ylmethyl)amine
3-(but-2-yn-1-yl)-5-(1-{[3-(2-hydroxyethoxy)phenyl]methyl}piperidin-4-yl)-5-(2-phenylethyl)imidazolidine-2,4-dione
1-(2-phenylpropyl)-4-(pyridin-3-ylmethyl)-1,4-diazepane
2-(2-hydroxyethyl)-5-[methyl(2-phenylethyl)amino]-2,3-dihydropyridazin-3-one
2-[2-({[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]-6-phenyl-2,3-dihydropyridazin-3-one
2-oxo-N-(propan-2-yl)-2-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)acetamide
3-(benzenesulfonyl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}propanamide
4-(hydroxymethyl)-1-{[6-(4-methylphenyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}azepan-4-ol
ethyl 1-(2,4-difluorobenzoyl)-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
2-{1-benzyl-4-[(8-fluoroquinolin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
6-[7-(3-methoxypropyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]pyridine-2-carbonitrile
2-(2-acetylphenyl)pyridine-4-carbonitrile
N-[(2R,3R)-2-(benzyloxy)-1'-(3-chlorothiophene-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
4-(6-ethylpyrimidin-4-yl)-N-(1,2,3-thiadiazol-5-yl)piperazine-1-carboxamide
N-{1-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]piperidin-4-yl}acetamide
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]amine
(3aR,7aS)-2-(2-propyl-1,3-thiazole-4-carbonyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
2-{2-oxo-8-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetic acid
1-{2-[2-(3-methoxyphenyl)azetidin-1-yl]-2-oxoethyl}azepan-2-one
2-[3-(furan-2-yl)-5-oxo-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-[(5-methyl-1,2-oxazol-3-yl)methyl]acetamide
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(thiophen-3-yl)ethan-1-one
(3aS,6aS)-2-cyclohexyl-5-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
{6-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]pyridin-2-yl}methanol
N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)isoquinoline-5-carboxamide
N,N-diethyl-1-({1-[3-(2-methoxyphenyl)propanoyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxamide
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
5-(dimethylamino)-2-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-2,3-dihydropyridazin-3-one
6-[3-oxo-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-2-carboxylic acid
(2S,4S)-4-amino-1-(6-ethyl-2-methylquinoline-4-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-(1-{[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
ethyl 4-{[3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylate
N-[(1-cyclopentylpiperidin-4-yl)methyl]-2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-(2-butoxybenzoyl)-4-[(3-methylpyridin-2-yl)methyl]piperazine
6-[(5-fluoro-2-methylphenyl)methyl]-3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
N-[2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-2-(3,4,5-trimethoxyphenyl)acetamide
4-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}thiomorpholine
N-[(3R,4S)-4-cyclopropyl-1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]pyrrolidin-3-yl]cyclohexanecarboxamide
1-{3,9-diazaspiro[5.5]undecan-3-yl}-2-(prop-2-en-1-ylsulfanyl)ethan-1-one
5-(1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-4-yl)-5-methylimidazolidine-2,4-dione
2-(2,6-dimethoxypyridin-3-yl)-2-[4-(4-hydroxyphenyl)piperazin-1-yl]acetic acid
3-phenyl-1-[1-(pyrrolidine-1-sulfonyl)piperidin-3-yl]propan-1-one
4-[(2,5-dimethoxyphenyl)methyl]-2-[(4-fluorophenyl)methyl]morpholine
1-[2-(4-fluorophenyl)morpholin-4-yl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
2-(5-methyl-1H-pyrazol-1-yl)-1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
N-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-3-(2-hydroxypropan-2-yl)piperidine-1-carboxamide
1-benzyl-4-[(2E)-2-methylbut-2-en-1-yl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
N-[3-(pyridin-2-yl)propyl]-6-{[(2S)-pyrrolidin-2-ylmethyl]amino}pyridine-3-carboxamide
1-[3-(1,3-benzoxazol-2-yl)piperidin-1-yl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
8-(3-chloro-2-methylbenzoyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid