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2-(3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
3-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-3,9-diazaspiro[5.5]undecane
1-methyl-3-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}-1,2-dihydroquinolin-2-one
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[2-(dimethylsulfamoyl)ethyl]propanamide
(2S,4R)-N-ethyl-1-(1H-imidazol-2-ylmethyl)-4-[3-(pyridin-4-yl)propanamido]pyrrolidine-2-carboxamide
2-(4-fluorophenyl)-2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethan-1-ol
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-[2-(1H-imidazol-1-yl)ethyl]-2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
(1-benzothiophen-2-ylmethyl)({[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
[(5-{1-[(4-chloro-3-fluorophenyl)methyl]piperidin-4-yl}-4-ethyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
N-(3-benzamido-4-methoxyphenyl)oxane-4-carboxamide
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-1-{8-fluoro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}ethan-1-one
methyl 8-[(5-methylfuran-2-yl)methyl]-1-(naphthalen-2-ylmethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-4-(thiophen-2-yl)butan-1-one
N-[3-(cyclopentyloxy)propyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
N-[2-(2-chlorophenyl)ethyl]-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-(3,4-difluorophenyl)-1-(pyridin-4-ylmethyl)piperidin-3-amine
2-[3-({[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenoxy]ethan-1-ol
1-amino-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)cyclobutane-1-carboxamide
N4-methyl-N4-[(2-methylpyridin-4-yl)methyl]-N6-(propan-2-yl)pyrimidine-4,6-diamine
2-[1-benzyl-4-(quinolin-2-ylmethyl)piperazin-2-yl]ethan-1-ol
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
N-[4-({[2-(3,5-dimethylphenoxy)ethyl](methyl)carbamoyl}methyl)phenyl]cyclopropanecarboxamide
1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-amine
N,N-diethyl-2-[4-(4-phenylazepane-1-carbonyl)-1H-1,2,3-triazol-1-yl]acetamide
7-methanesulfonyl-4-methyl-2-[4-(3-phenylpiperidine-1-carbonyl)piperidin-1-yl]quinazoline
2-(4-methoxyphenoxymethyl)-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,3-oxazole-4-carboxamide
2-{[2-(2,6-difluorophenyl)-1H-imidazol-1-yl]methyl}-3-(furan-2-yl)propan-1-ol
1-(3-ethylphenyl)-3-[2-(1-methylpyrrolidin-2-yl)ethyl]urea
1-[2-(piperidin-1-yl)ethyl]-3-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]urea
3-(1-{[2-(ethylamino)pyrimidin-5-yl]methyl}piperidin-4-yl)-N-(3-methylphenyl)propanamide
1-(4-chlorophenyl)-N-{[1-(1,3-thiazol-5-ylmethyl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
5-phenyl-1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]pentan-1-one
1-[2-(benzenesulfonyl)ethyl]-4-[(dimethylamino)methyl]azepan-4-ol
(4aS,7aR)-1-(3-hydroxy-4-methylbenzoyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[1-(propan-2-yl)piperidin-4-yl]-1-[1-(pyridin-3-yl)-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl]ethan-1-one
4-cyclopentyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrimidin-2-amine
N-[(5-{[4-(propan-2-yl)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]cyclobutanecarboxamide
8-methoxy-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-(propan-2-yl)acetamide
{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
N-{5-[({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)carbamoyl)amino]-2-methoxyphenyl}acetamide
3-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[3-(pyridin-4-yl)propyl]propanamide
2-(3-methylbutyl)-8-[3-(4H-1,2,4-triazol-4-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-2,3,6-trimethylquinoline-4-carboxamide
(2R,6R)-4-[2-(1H-imidazol-1-yl)ethyl]-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
9-(1H-1,2,3-benzotriazole-5-carbonyl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(2,6-dimethylpyrimidine-4-carbonyl)piperidin-3-amine
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3-propanamidobenzamide