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1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-4-(2-methylphenyl)-1,4-diazepane
N,7-dimethyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-2-(pyrimidin-5-yl)quinoline-4-carboxamide
1-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
(1S,5R)-6-[(dimethylcarbamoyl)methyl]-N-(2,4-dimethylphenyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
methyl 2-{[3-(morpholin-4-yl)piperidine-1-carbonyl]amino}benzoate
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-2-(1H-pyrazol-1-yl)acetamide
N-({3-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)-2-(thiophen-3-yl)acetamide
(2S,4R)-N-[2-(3-fluorophenyl)ethyl]-4-[(4-fluorophenyl)sulfanyl]-1-[(4-hydroxyphenyl)methyl]pyrrolidine-2-carboxamide
2-(1-{1-[3-(morpholin-4-yl)benzoyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-ol
2,6-dimethyl-4-({methyl[1-(pyridin-4-yl)ethyl]amino}methyl)phenyl acetate
2-{4-[3-(benzenesulfonyl)propanoyl]morpholin-3-yl}-N-(2-fluoroethyl)acetamide
{[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(3-phenylpropyl)amine
1-{2-oxo-2-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-2-yl]ethyl}imidazolidine-2,4-dione
3-[(2R,6R)-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-2,1-benzoxazole
2-(dimethylamino)-2-(3-fluorophenyl)-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]acetamide
4-cyano-N,1-dimethyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-1H-pyrrole-2-carboxamide
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}[(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
4-[1-(2,5-dimethylphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazole-5-carbonyl]morpholine
4-{1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-2-(thiophen-2-yl)-1,3-thiazole
N-[2-(3-methoxyphenyl)phenyl]-1-(quinolin-8-ylmethyl)piperidine-4-carboxamide
{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}(methyl)(oxan-2-ylmethyl)amine
N-[2-(4-fluorophenyl)ethyl]-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-2-methyl-1,3-thiazole-4-carboxamide
2-[3-(3-phenyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]acetamide
N-methyl-5-(1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
{4-[4-(benzyloxy)piperidine-1-carbonyl]cyclohexyl}methanamine
3-[2-(3-methoxyphenyl)ethyl]-1-(1-methylcyclopropanecarbonyl)piperidine
2-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinoline
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-({7-[(5-methylfuran-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-phenoxyacetamide
4-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1λ6-thiomorpholine-1,1-dione
(1R,5R)-N,N-dimethyl-6-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-chloro-4-fluoro-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-benzothiophene-2-carboxamide
[5-(1H-pyrazol-3-yl)-1H-1,3-benzodiazol-2-yl]methanol
5-{[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]methyl}-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-[(3,5-difluorophenyl)methyl]-3-(methanesulfonylmethyl)piperidine
methyl 6-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]pyrimidine-4-carboxylate
6-methyl-2-[2-({5-propylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-3,4-dihydropyrimidin-4-one
N-[(3S,4R)-1-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
3-(1-methyl-4-phenyl-1H-pyrazol-5-yl)-1-[1-(morpholin-4-ylmethyl)cyclopentyl]urea
1-{4-[1-(2-fluoroethyl)-4-phenyl-1H-imidazol-5-yl]phenyl}-1H-1,2,4-triazole
[(4-ethynylphenyl)methyl][(2-methoxyphenyl)methyl](pyridin-3-ylmethyl)amine
2-(1-{5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carbonyl}pyrrolidin-2-yl)pyridine
3-(1H-1,3-benzodiazol-2-yl)-1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}propan-1-one
(1S,6R)-3-methyl-9-{2-[4-(3-methylphenyl)piperazin-1-yl]acetyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
2-methyl-5-(3-{[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)pyrazine
(2R)-2-[(3-methyl-1-propyl-1H-pyrazol-4-yl)formamido]-3-(3,4,5-trifluorophenyl)propanoic acid
2-cyclopropyl-9-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}-2,9-diazaspiro[5.5]undecan-3-one
methyl 3-(2-chlorobenzenesulfonamido)-5-{[2-(2-fluorophenyl)acetamido]methyl}benzoate
1-cyclohexyl-4-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
1-(but-2-ynoyl)-N-[3-(3-methylphenyl)phenyl]piperidine-3-carboxamide