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2-amino-4-(2-chloro-4-hydroxy-5-methoxyphenyl)-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
1-(5,6,7-trimethoxy-3-{[(2-methylpropyl)amino]methyl}quinolin-2-yl)piperidin-3-ol
N-[(trimethyl-1H-imidazol-2-yl)methyl]-9H-purin-6-amine
N,1-dimethyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrrole-2-carboxamide
2-{[3-(4-propyl-1,4-diazepane-1-carbonyl)-1,2-oxazol-5-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
3-({3-[4-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)pyridine
3-[1-(5-ethyl-1,2,4-oxadiazol-3-yl)piperidin-3-yl]-N-(4-methoxy-2-methylphenyl)propanamide
9-[(2-methoxyphenyl)methyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
[7-(3,6-dimethylpyrazin-2-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methanamine
N-[(3-ethoxyphenyl)methyl]-2-hydroxy-N-(prop-2-en-1-yl)pyridine-3-carboxamide
N-(3-chloro-4-fluorophenyl)-3-{1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidin-4-yl}propanamide
9-(cyclopropylmethyl)-1-methyl-4-[2-(morpholin-4-yl)-2-oxoethyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-methyl-N-[(3-methylpyridin-4-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
3-butyl-4-(4-methanesulfonylbenzoyl)-1-methylpiperazin-2-one
2-cyclobutyl-7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-3-(2-oxopyrrolidin-1-yl)propanamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(6-methylpyridine-3-carbonyl)piperidin-3-amine
(4aS,7aR)-1-[2-(furan-2-yl)-2-oxoacetyl]-4-[(5-methylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-chloro-2-{3-[(4-methylpiperazin-1-yl)methyl]piperidine-1-carbonyl}phenol
5,6-dimethyl-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}pyrimidin-4-amine
N-cyclohexyl-2-(ethylamino)-N-(pyridin-2-ylmethyl)pyrimidine-5-carboxamide
3-(difluoromethoxy)-N-methyl-N-[(1-methylpiperidin-2-yl)methyl]benzamide
3-(4-fluorophenyl)-3-{2-[1-(propan-2-yl)piperidin-4-yl]acetamido}propanoic acid
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N,3-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
7-methyl-2-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}-2,7-diazaspiro[4.5]decan-6-one
N-[(3,5-dimethoxyphenyl)methyl]-4-(piperidin-3-yl)benzamide
2-(2,4-dichlorophenoxy)-N-[2-(pyridin-3-yloxy)propyl]acetamide
(3aS,6aR)-5-(1-methyl-1H-pyrazole-5-carbonyl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-(4-phenoxybenzoyl)-1-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]piperidine
2-hydroxy-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-6-(trifluoromethyl)pyridine-3-carboxamide
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(5-methylfuran-2-yl)-5-(oxolan-3-yl)-1H-1,2,4-triazole
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N,1-dimethyl-3-propyl-1H-pyrazole-5-carboxamide
4-(4-ethoxy-3-methylphenyl)-1-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]butan-1-one
6-{1-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-3-ol
N,7-dimethyl-N-(2-methylpropyl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
2-(2-methoxyethyl)-9-[2-(4-methoxyphenoxy)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(3S,4S)-1-({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
5-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-2-amine
4-({4-methyl-5-[1-(pyridine-4-carbonyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
5-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-(hydroxymethyl)-1H-1,3-benzodiazole-5-carboxamide
N-methyl-4-(4-methylpiperazin-1-yl)-N-[2-(1,2,4-oxadiazol-3-yl)ethyl]benzamide
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxamide
2-[5-(5-cyclopropyl-3-methyl-1H-pyrazol-4-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]acetic acid
1-{[3-(5-methylfuran-2-yl)phenyl]methyl}azepan-4-amine
4-{2-[4-(2-propyl-1,3-thiazole-4-carbonyl)piperazin-1-yl]ethyl}morpholine
(1-methyl-1H-imidazol-2-yl)[1-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl]methanol
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
N-(1,4-dioxan-2-ylmethyl)-1-(6-methyl-2-propylpyrimidin-4-yl)piperidin-4-amine