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3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(furan-2-ylmethyl)-N-(2-hydroxyethyl)benzamide
methyl 3-[4-(cyclohex-3-ene-1-carbonyl)-2-oxo-6-(pyridin-4-ylmethoxy)-1,4-diazepan-1-yl]propanoate
methyl 2-[methyl(2-methylpropyl)sulfamoyl]-6-{[4-(methylsulfanyl)phenyl]methyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-(2,5-dimethoxyphenyl)-2-[5-methyl-4-(pyrrolidine-1-carbonyl)-1H-pyrazol-1-yl]pyrimidine
N,3-dimethyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
4-ethyl-1-methyl-3-({1-[2-(pyridin-4-yl)acetyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl){[5-(oxolan-2-yl)thiophen-2-yl]methyl}amine
(2S,4R)-4-amino-N,N-diethyl-1-[3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanoyl]pyrrolidine-2-carboxamide
2-(3-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}phenoxy)acetamide
{2-[5-(1,2-dimethyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}bis(propan-2-yl)amine
1-ethyl-4-{1-[4-(3-fluorophenyl)phenyl]piperidin-4-yl}piperazine
2-(2-phenoxyphenyl)pyridine-4-carboxamide
2-{1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperidin-2-yl}pyridine
1-{3-[(4-methylpiperazin-1-yl)methyl]-1,2,4-oxadiazol-5-yl}cyclopentan-1-amine
1-ethyl-8-(1H-indol-3-ylmethyl)-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-(ethoxymethyl)-3-(1-phenylcyclopropyl)-1,2,4-oxadiazole
6-(cyclopropylmethoxy)-4-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
3-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-3-methyl-1-[2-(trifluoromethyl)phenyl]urea
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-1-methyl-1H-pyrazole-4-carboxamide
1-[2-(4-methoxyphenyl)ethyl]-N,N-dimethyl-5-[(2-methyl-1H-indol-3-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(azepane-1-carbonyl)-N-[2-(3-methoxyphenyl)ethyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3aR,6aR)-2-ethyl-5-{[(4-methoxyphenyl)methyl]carbamoyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(cyclopentylmethyl)-3-[4-(4-fluorophenyl)piperazine-1-carbonyl]-1-(2-methoxyethyl)-6-methyl-1,4-dihydropyridin-4-one
N-{1-[1-phenyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]propan-2-yl}acetamide
N-[3-(4-fluorophenyl)phenyl]-3-methoxypiperidine-1-carboxamide
(3S,4S)-4-cyclopropyl-1-[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl]pyrrolidine-3-carboxylic acid
N-({1-[2-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)-2-oxoethyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)acetamide
2-({[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(ethyl)amino)ethan-1-ol
N,1-dimethyl-2-(morpholin-4-yl)-N-[1-(1,2-oxazol-3-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
9-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-3-oxa-9-azaspiro[5.5]undecane
1-{3-azaspiro[5.5]undecan-9-yl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-[1-(1-ethylpiperidin-4-yl)piperidin-3-yl]-4-(2-methoxyphenyl)piperazine
4-(1H-imidazol-1-yl)-1-[1-(methoxymethyl)cyclobutanecarbonyl]piperidine-4-carboxylic acid
4-(2-oxoimidazolidine-4-carbonyl)-1-phenylpiperazin-2-one
N-(1-benzylpyrrolidin-3-yl)-1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-[(4,4-difluoropiperidin-1-yl)sulfonyl]-N-(pyrrolidin-3-yl)benzamide
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(4-fluoro-3-methylphenyl)methyl]piperidine
4-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-1-cyclopentylpiperazin-2-one
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-3,5-dimethylfuran-2-carboxamide
2-[5-(4-fluoro-2-methylbenzenesulfonamidomethyl)-1-(2-hydroxyethyl)-1H-1,2,4-triazol-3-yl]acetamide
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-1-{4-[(2-methylphenyl)methyl]piperazin-1-yl}ethan-1-one
(3R,4S)-4-[methyl({[2-(trifluoromethyl)phenyl]methyl})amino]oxolan-3-ol
5-methoxy-2-{[9-methoxy-7-(4-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenol
3-(5-amino-1H-1,2,4-triazol-3-yl)-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}propanamide
7-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
1-{5-[(cyclobutylamino)methyl]-2-methoxyphenoxy}-3-(diethylamino)propan-2-ol
1-[(3-chloro-2,4-difluorophenyl)methyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
N-{3-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-3-oxopropyl}methanesulfonamide
{5-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]-1H-1,3-benzodiazol-2-yl}methanol
(2S)-2-amino-3-(1H-imidazol-4-yl)-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one