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N-[(2-methoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)oxolane-3-carboxamide
(3S)-3-{[5-(6-aminopyridin-3-yl)-4-(4-methylphenyl)pyrimidin-2-yl]amino}azepan-2-one
N-[(2-fluorophenyl)methyl]-2-{[3-(morpholin-4-yl)propyl]amino}acetamide
methyl (2S,4R)-1-methyl-4-{2-methylimidazo[1,2-a]pyrimidine-3-amido}pyrrolidine-2-carboxylate
1-ethyl-N-({5-methyl-2-[2-(3-phenoxypropanamido)phenyl]-1,3-oxazol-4-yl}methyl)-1H-pyrazole-4-carboxamide
2-[2-(ethylsulfanyl)propanoyl]-N-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
2-{2-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethyl}pyridine
2-cyclopropyl-3-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]-6-methyl-1-(thiophen-2-ylmethyl)-1,4-dihydropyridin-4-one
1-(3-methylpyrazin-2-yl)-4-(oxolane-2-carbonyl)-1,4-diazepane
[(5-methoxy-3-methyl-1H-indol-2-yl)methyl](methyl)[3-(1H-pyrazol-1-yl)propyl]amine
2-methyl-6-{1-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidin-3-yl}pyrimidin-4-ol
1-(7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(thiophen-2-yl)ethan-1-one
2-{[1-(4-phenylpiperazine-1-carbonyl)-6-azaspiro[2.5]octan-6-yl]methyl}-1H-1,3-benzodiazole
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-2-ethoxy-N-methylpyridine-3-carboxamide
6-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]quinoxaline
4-[(4-fluoro-3-methylphenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
1-(3-{[3-(2-hydroxyethyl)-4-(3-methylbut-2-en-1-yl)piperazin-1-yl]methyl}phenyl)ethan-1-one
2-amino-4-[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]-6-(6-methoxypyridin-3-yl)pyridine-3-carbonitrile
6-methyl-2-[7-(oxan-4-yl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]pyridine-3-carbonitrile
1-(1H-imidazol-4-ylmethyl)-4-[(propan-2-yl)carbamoyl]-1,4-diazepane-6-carboxylic acid
2-{methyl[(4-methyl-5-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]amino}ethan-1-ol
(2S)-2-{[3-(3-hydroxy-3-methylbutyl)phenyl]formamido}-3-(1H-imidazol-4-yl)propanamide
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-2-oxo-2H-pyran-5-carboxamide
4,4,4-trifluoro-N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]butanamide
(3R,4S)-N-(cyclohexylmethyl)-4-hydroxy-3,4-dimethylpiperidine-1-carboxamide
4-({1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}methyl)-2-(prop-2-en-1-yl)phenol
ethyl 4-[(4-methoxyphenyl)methyl]-1-(2-phenoxypropanoyl)piperidine-4-carboxylate
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-[5-(propan-2-yl)pyrimidin-4-yl]piperidin-4-ol
(2S)-1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-methyl-2-phenylpiperazine
3-{2-[6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]-2-oxoethyl}-1λ6-thiolane-1,1-dione
3-methyl-N-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]pyridin-4-amine
6-(2-chlorophenyl)-2-(4-{[methyl(propyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N-[(3R,4S)-4-cyclopropyl-1-(oxan-4-yl)pyrrolidin-3-yl]-2-(2H-1,2,3-triazol-2-yl)acetamide
3-(2-benzyl-5-oxopyrrolidin-2-yl)-N-(2,2-diphenylethyl)propanamide
methyl 1-{3-[(2-chlorophenyl)methyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}piperidine-2-carboxylate
4-{[({4-[2-hydroxy-3-(4-methylpiperazin-1-yl)propoxy]phenyl}methyl)amino]methyl}hepta-1,6-dien-4-ol
2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]-N-(propan-2-yl)acetamide
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)but-2-ynamide
5-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-(1-{7-[(4-hydroxy-2-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylpropanamide
1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-4-(3-methoxybenzoyl)piperazine
N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
3-(2-chlorophenyl)-3-{2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-oxoethyl}-1-(2-methoxyethyl)pyrrolidine-2,5-dione
3-{[1-(but-3-enoyl)piperidin-4-yl]oxy}-N-[2-(dimethylamino)ethyl]-N-methylbenzamide
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-3,4-dimethoxybenzamide
2-(4-methoxyphenoxymethyl)-N-(propan-2-yl)-1,3-oxazole-4-carboxamide
1-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-2-(2-methoxyethyl)piperidine
2-({[(3R,4R)-1-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
2-[4-(2-amino-5-butyl-6-methylpyrimidin-4-yl)morpholin-2-yl]ethan-1-ol
N-ethyl-N-(2-hydroxyethyl)-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide