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N-(4-{[(dimethyl-1,3-thiazol-5-yl)methyl]carbamoyl}phenyl)-2-methylfuran-3-carboxamide
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)propanamide
1-[2-(cyclohexylsulfanyl)ethyl]-3-(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
N-[2-(dimethylamino)ethyl]-N-(2-hydroxyethyl)-2-methyl-1,3-thiazole-4-carboxamide
(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-7-({[4-(propan-2-yl)phenyl]methyl}amino)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(azocan-1-yl)-3-[4-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)-2-methoxyphenoxy]propan-2-ol
1-methyl-4-{1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}-1,4-diazepane
(1R,5R)-6-benzyl-3-(1-methyl-1H-pyrazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-cyclopropyl-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-5-oxopyrrolidine-3-carboxamide
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-3-(5-methyl-1H-1,2,4-triazol-3-yl)propanamide
4-(2H-1,3-benzodioxol-5-yloxy)-1-(2-methylpyridin-4-yl)piperidine-4-carboxylic acid
1-[3-(2-phenylethyl)piperidin-1-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
8-(dimethyl-1,3-thiazole-5-carbonyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane
3-[(2R,3R,6R)-5-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
(1S,5R)-3-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
[4-({1-[3-(1H-imidazol-2-yl)benzoyl]pyrrolidin-3-yl}methyl)phenyl]methanol
4-chlorophenyl (7S,9aR)-7-benzyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-oxo-1,6-dihydropyridine-2-carboxamide
3-(1H-1,2,4-triazol-1-yl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]propanamide
3-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2-{1-[1-(pyridine-2-carbonyl)piperidin-4-yl]piperidin-4-yl}ethyl)pyrrolidin-2-one
4-{1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-3-propylmorpholine
1-[3-(difluoromethoxy)benzoyl]-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
N-{[3-(2H-1,3-benzodioxol-5-ylmethoxy)phenyl]methyl}-2,3-dimethyl-N-(pyridin-2-ylmethyl)-1H-indole-7-carboxamide
N-[(1-methylpiperidin-3-yl)methyl]-3-phenoxypropanamide
N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-phenyl-1,4-diazepane
1-(6-methyl-2-propylpyrimidin-4-yl)piperidine-4-carboxamide
N,N-dimethyl-5-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)cyclohexanecarboxamide
2-hydroxy-N-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}-2-methylpropanamide
N-benzyl-2-[4-(4-{[1-(thiophen-3-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]acetamide
1-(2-hydroxyethyl)-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
4-{[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
N-{[2-(4-acetylpiperazin-1-yl)-7-methylquinolin-3-yl]methyl}-N-cyclopropyl-2-methylpropanamide
(3S,4S)-1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)-4-(morpholin-4-yl)pyrrolidin-3-ol
5-[4-hydroxy-1-(2-methylpropyl)piperidin-4-yl]-N-methyl-N-(quinolin-5-ylmethyl)-1-benzofuran-2-carboxamide
[(3R,4R)-1-[1-(4-chlorophenyl)cyclopropanecarbonyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
3-[2-(methylcarbamoyl)-4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl]piperidine-1-carboxamide
1-(morpholin-4-yl)-2-[4-(5-propyl-1,3,4-oxadiazol-2-yl)piperazin-1-yl]ethan-1-one
[(3R,4R)-1-(4,6-dimethylpyrimidin-2-yl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
(3R,4R)-1-[3-(3-fluorophenyl)benzoyl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
3-(azetidine-1-carbonyl)-N-[3-(3-hydroxypiperidin-1-yl)propyl]benzene-1-sulfonamide
3-(cyclohexylamino)-N-cyclopentyl-5-(phenylsulfamoyl)benzamide
N-(1-cycloheptylpiperidin-3-yl)-2-(1-propylpiperidin-4-yl)acetamide
1-(azepan-1-yl)-3-[3-({methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
N-[4-(furan-2-yl)phenyl]-1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidine-3-carboxamide
2-{6-hydroxy-4-[3-(hydroxymethyl)-7-methylquinolin-2-yl]-1,4-diazepan-1-yl}acetamide