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N-(1-{7-[(3-ethoxy-4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxane-4-carboxamide
1-[1-ethyl-3-(4-phenylpiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(2H-indazol-2-yl)ethan-1-one
[5-({[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amino}methyl)-2-(propan-2-yloxy)phenyl]methanol
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
2-[4-(2-chlorophenoxy)piperidin-1-yl]-5-(1H-imidazol-1-ylmethyl)pyridine
N-[5-({[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)amino}methyl)pyrimidin-2-yl]benzenesulfonamide
1-[benzyl(methyl)amino]-3-[4-({[(4-chlorophenyl)methyl]amino}methyl)phenoxy]propan-2-ol
N-[2-fluoro-5-({[2-(2-methylphenoxy)ethyl]carbamoyl}amino)phenyl]-2-methylpropanamide
3-(1,3-dimethyl-4-phenyl-1H-pyrazol-5-yl)-1-(2-methoxyethyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]urea
3-[(4-methoxyphenyl)methyl]-1-methyl-8-[3-(5-methylfuran-2-yl)butyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-(furan-3-carbonyl)piperidine
(1S,5R)-3-(2,6-difluoro-3-methoxybenzoyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]amino}pyridine-3-carbonitrile
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-4-(2-oxopiperidin-1-yl)butanamide
1-[(2E)-but-2-en-1-yl]-4-(4-carbamoyl-1,3-thiazol-2-yl)-1,4-diazepane-6-carboxylic acid
N-[1-(furan-2-ylmethyl)piperidin-4-yl]-3-methyl-1,2-oxazole-5-carboxamide
N,8-dimethyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
ethyl 4-[(2-chlorophenyl)methyl]-1-(5-methoxyfuran-2-carbonyl)piperidine-4-carboxylate
3-(propoxymethyl)-1-{1H-pyrrolo[2,3-b]pyridin-6-yl}pyrrolidine
(4aR,7aS)-1-(2-methoxyethyl)-4-[(1-methyl-1H-imidazol-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(4,6-dimethylpyrimidin-2-yl)amino]-3-(3-methoxyphenoxy)propan-2-ol
2-methoxy-1-{4-[6-(propan-2-yl)-1H-indole-2-carbonyl]-1,4-diazepan-1-yl}ethan-1-one
[3-benzyl-1-(thiophene-2-sulfonyl)piperidin-3-yl]methanol
7-chloro-2-(2-cyclopropylpyrimidin-5-yl)-N-(propan-2-yl)quinoline-4-carboxamide
1-{3-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
(2R,3R)-3-[4-(4-hydroxyphenyl)piperazin-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
[(1S,3S,3aS,6aR)-3-[4-methoxy-3-(methoxymethyl)phenyl]-5-methyl-1-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
5,6-dimethyl-2-{[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,3-dihydropyridazin-3-one
4-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}thiomorpholine
{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
2-{[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1-propyl-1H-imidazole
(1S,5R)-6-(1-benzofuran-5-carbonyl)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-(2,5-dioxoimidazolidin-4-yl)-N-{[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]methyl}acetamide
5-[1-(2-methoxy-2-methylpropyl)-1H-imidazol-2-yl]-2-(methoxymethyl)pyrimidine
methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}){[2-(propan-2-yl)pyrimidin-4-yl]methyl}amine
methyl 2-[3-(2-methoxybenzoyl)piperidine-1-carbonyl]benzoate
8-(furan-3-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
N,N-dimethyl-2-(pyridin-2-yl)-7-(1H-pyrrole-2-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(4aR,7aS)-1-acetyl-4-(quinoline-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-2-(ethylamino)-N-methylpyrimidine-5-carboxamide
3-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane-4-carbonyl}-4-phenylpyrrolidin-2-one
2-amino-4-(3-ethyl-1H-pyrazol-5-yl)-6-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
4-{2-[4-(2-methyl-1-benzofuran-7-carbonyl)piperazin-1-yl]ethyl}morpholine
2-({2-[1-(5-methoxyfuran-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
6-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
6-methyl-4-[3-(pyrrolidine-1-carbonyl)piperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
1-cyclopentyl-N-{[5-(methylcarbamoyl)furan-2-yl]methyl}-5-oxopyrrolidine-3-carboxamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[(3-methoxyphenyl)methyl]piperidin-4-yl}oxy)benzamide
5-cyclopropyl-N-[(2,4-dimethoxyphenyl)methyl]-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
3-fluoro-N-(1-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide