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1-methyl-3-(propan-2-yl)-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-1H-pyrazole-5-carboxamide
1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}-3-(trimethyl-1H-pyrazol-1-yl)propan-1-one
3-chloro-6-methyl-N-{[1-(morpholin-4-ylmethyl)cyclopropyl]methyl}pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-[2-(7-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-4-methoxybenzamide
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-1-[4-(2-ethoxyphenyl)piperazin-1-yl]propan-1-one
{4-[(2,4,5-trimethylphenyl)methyl]morpholin-2-yl}methanamine
(3R,4R)-1-{[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-4-(hydroxymethyl)piperidin-3-ol
3-(2-methyl-2H-1,2,3-benzotriazol-4-yl)-1-[2-(3-phenylpiperidin-1-yl)ethyl]urea
3-[1-(1-cyclooctylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]pyridine
3-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyridin-2-ol
N-ethyl-2-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
(1S,5R)-6-(2-methoxyethyl)-3-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(dimethylamino)ethyl]-N-ethyl-2-(3-fluorobenzamido)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
2-methoxy-1-[2-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine-3-carbonyl)-4-methylpiperazin-1-yl]ethan-1-one
[(3-chlorophenyl)methyl](methyl)[(4-methyl-5-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)methyl]amine
5-[1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-pyrazol-3-yl]-N-[(3-methoxyphenyl)methyl]-4-methyl-1,3-thiazol-2-amine
N-[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]-2-ethylpyrimidine-5-carboxamide
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-2-methoxy-N-methylbenzamide
2-chloro-5-acetamido-N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]benzamide
4-[2-(2-fluorophenyl)ethyl]-3-[(trimethyl-1H-pyrazol-1-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-methyl-N-(thiophen-2-ylmethyl)benzamide
1-methyl-6-(pyridin-3-yl)-N-[1-(thiophen-2-yl)propan-2-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
7-(cyclohexylmethyl)-2-(1H-imidazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
6-methyl-2-({[(1s,4s)-4-aminocyclohexyl]amino}methyl)quinolin-4-ol
1-{4-[2-(naphthalen-1-ylmethyl)morpholin-4-yl]-4-oxobutyl}piperidin-2-one
3-[methyl(1,2-oxazol-3-ylmethyl)sulfamoyl]-N-(1,2-oxazol-3-ylmethyl)benzamide
N,N-dimethyl-7-(3-methylbenzoyl)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-({7-[2-(2-chlorophenoxy)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1H-1,3-benzodiazole-5-carboxamide
3-(4-chlorophenyl)-5-(oxolan-2-ylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
5-(3-fluorophenoxymethyl)-N-methyl-N-(oxan-2-ylmethyl)-1H-pyrazole-3-carboxamide
8-(2-methylpyridine-3-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
[1-(1-{[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methanol
3-[(2R,3R,6R)-5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-[(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]-1H-pyrazole-4-carboxamide
2-{4-[3-(pyridin-2-yl)azetidin-1-yl]piperidin-1-yl}-5-(trifluoromethyl)pyridine
N-[1-(1H-imidazol-1-yl)butan-2-yl]-6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-ethyl-3-({ethyl[2-hydroxy-2-(3-hydroxyphenyl)ethyl]carbamoyl}amino)-4-methylbenzamide
2-{4-[(4-ethoxypiperidin-1-yl)methyl]phenoxy}acetic acid
3-({[5-(1H-1,3-benzodiazol-1-ylmethyl)-1H-pyrazol-3-yl]formamido}methyl)-1,2,4-oxadiazole-5-carboxamide
N-methyl-N-[(1-methylpiperidin-3-yl)methyl]-2-phenylbenzamide
{1-[6-(2-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]azepan-2-yl}methanol
(2S,4R)-1-(adamantan-2-yl)-4-[(4-methoxyphenyl)sulfanyl]-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
2-{1-[(1-cyclopentyl-1H-imidazol-5-yl)methyl]pyrrolidin-2-yl}-6-methyl-1H-1,3-benzodiazole
N-methyl-N-(prop-2-en-1-yl)-3-{[1-(pyrrolidin-1-yl)propan-2-yl]sulfamoyl}benzamide
1-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]-N-(1,2-oxazol-3-ylmethyl)piperidin-4-amine
3-(1H-imidazol-2-yl)-1-[1-(4-phenoxyphenyl)-1H-1,2,3,4-tetrazol-5-yl]piperidine
2-{2-[4-(1-cyclohexyl-1H-1,2,4-triazol-5-yl)-1H-1,2,3-triazol-1-yl]ethyl}piperidine
1-(cyclohex-3-en-1-ylmethyl)-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
2-cyclopropyl-8-{[2-(2-hydroxyethoxy)phenyl]methyl}-2,8-diazaspiro[5.5]undecan-3-one