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2-({4-[5-(3-fluorophenyl)-2-(trifluoromethyl)pyrimidin-4-yl]piperidin-1-yl}methyl)-1H-1,3-benzodiazole
{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(ethyl)(pyridin-4-ylmethyl)amine
(2-methylpropyl)({[5-(1H-pyrazol-5-yl)furan-2-yl]methyl})(pyridin-2-ylmethyl)amine
ethyl 1-[(4,5-dimethylfuran-2-yl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylate
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[3-(pyridin-3-yl)propyl]acetamide
2-{1-[(8-methoxy-2H-chromen-3-yl)methyl]piperidin-3-yl}-1,2,3,4-tetrahydroisoquinoline
2-methanesulfonamido-N-[(3R,4S)-1-(2-methoxyethyl)-4-propylpyrrolidin-3-yl]acetamide
(3aS,6aS)-2-(ethanesulfonyl)-5-(3-methoxypyrazin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-cyclopentyl-9-(3-phenoxypropanoyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{3-[3-(pyridin-2-yl)azetidine-1-carbonyl]phenyl}imidazolidin-2-one
2-methyl-5-[3-(oxolan-2-ylmethyl)-1,2,4-oxadiazol-5-yl]-1H-1,3-benzodiazole
2-(pyridin-2-yl)-1-{spiro[azepane-4,2'-chromene]-1-yl}ethan-1-one
4-(1-methyl-1H-imidazol-2-yl)-1-[1-(1-methylpiperidin-4-yl)piperidine-4-carbonyl]piperidine
3-[ethyl({[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl})amino]-1λ6-thiolane-1,1-dione
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-2-methoxy-2-phenylacetamide
5-[3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)phenyl]-1,3-oxazole
1-[6-amino-2-(dimethylamino)pyrimidin-4-yl]-3-(cyclopropylmethyl)piperidine-3-carboxylic acid
1-benzyl-N-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}pyrrolidin-3-amine
[2-(1H-indol-1-yl)ethyl](methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
N-methyl-3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
4-methyl-7-{[(pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}-2H-chromen-2-one
N-{[7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
4-({4-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]furan-2-yl}methyl)morpholine
1-{4-[4-(1-hydroxycyclopentyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-3,3-dimethylbutan-1-one
4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}pyrimidine-5-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-1-[1-(3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propan-1-one
4-(3,3-dimethylpyrrolidine-1-carbonyl)-2-(1-ethyl-1H-pyrazol-4-yl)-7,8-dimethylquinoline
4-chloro-3-fluoro-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]benzamide
9-[2-(2,4-difluorophenyl)acetyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-{[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)amino}-2-phenylacetic acid
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-1-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
2-{2-[1-(4-oxo-4-phenylbutanoyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
N,N-dimethyl-2-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}aniline
3-{1-[(5-chloro-2-hydroxyphenyl)methyl]piperidin-4-yl}-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
2-amino-8-[2-(dimethylamino)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
5-ethyl-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}pyrazolo[1,5-a]pyrimidin-7-amine
{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)(oxan-2-ylmethyl)amine
2-[4-({[(1-methanesulfonylpiperidin-3-yl)methyl]carbamoyl}amino)phenyl]-N-methylacetamide
(2R,3R)-3-amino-1'-(4-methoxypyrimidin-2-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-[3-({1-[(1-ethyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}oxy)benzoyl]morpholine
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-4-amine
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)acetamide
ethyl 2-{[7-(pyridine-4-amido)-1,2,3,4-tetrahydroisoquinoline-2-carbonyl]amino}acetate
4-[3-(2-methylphenyl)piperidine-1-carbonyl]quinoline
5-chloro-4-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-2-methoxyphenol
2-[(4aS,8aR)-2-oxo-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-6-yl]-6-methylpyridine-3-carbonitrile
8-(1-methoxypropan-2-yl)-3-(2-methylpropyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{[(3-cyano-4,6-dimethylpyridin-2-yl)amino]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
6-{[4-(propan-2-yl)phenyl]methyl}-4-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine