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5-methyl-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1-methyl-1H-imidazole-5-carboxamide
5-(3-methoxyphenyl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1,2,4-triazin-3-amine
N-(4-fluoro-2-methylphenyl)-3-{1-[4-(2-oxopyrrolidin-1-yl)butanoyl]piperidin-3-yl}propanamide
2-(pyrimidin-2-ylsulfanyl)-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}acetamide
5-acetyl-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]thiophene-2-carboxamide
N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-2-(2,3,6-trimethylphenoxy)acetamide
1-cyclopentyl-N3,N3-diethyl-N5-methyl-4-oxo-N5-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-{3-[2-(oxolan-3-yl)-1H-imidazol-1-yl]phenyl}acetamide
N-{4-[2-(oxolan-3-yl)-1H-imidazol-1-yl]phenyl}methanesulfonamide
4-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}morpholine-2-carboxylic acid
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-propyl-1,3-thiazole-4-carboxamide
2-amino-4-(2-butoxy-3-methoxyphenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-[(3-chlorophenyl)methyl]-3-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]propanamide
1-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-3-methoxypiperidine
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
1-[(1-ethylpiperidin-3-yl)methyl]-4-phenylpiperidine-4-carbonitrile
8-[(2-cyclohexylpyrimidin-5-yl)methyl]-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(1-{1-[2-(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl)acetyl]piperidin-4-yl}-2-(4-fluorophenyl)ethyl)-2-methoxy-N-methylacetamide
N-(1-methyl-1H-indazol-3-yl)-2-[3-(3-methylpyrazin-2-yl)-1H-pyrazol-1-yl]acetamide
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-3-(2-methoxyphenyl)benzamide
3-({4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-2-(pyridin-4-yl)acetamide
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-5,6,7,8-tetrahydroquinazolin-2-amine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]piperidin-3-ol
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)isoquinoline-1-carboxamide
2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-3-methylquinoxaline
6-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]pyridine-2-carbonitrile
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-4-(2-methoxyethyl)piperazine-1-carboxamide
2-{4-[(propan-2-yl)amino]pyrimidin-2-yl}benzamide
8-(1H-indol-3-ylmethyl)-3-methyl-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-[ethyl(2-methylprop-2-en-1-yl)amino]-1-methyl-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-methyl-5-[4-(2-methyl-1-benzofuran-5-carbonyl)piperazin-1-yl]-2,3-dihydropyridazin-3-one
N-(furan-3-ylmethyl)-6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl](methyl){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
N-(cyclopropylmethyl)-N-(2-methoxyethyl)-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
5-[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]quinoline
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(3S,4S)-1-ethyl-4-(naphthalen-2-yl)piperidin-3-ol
3-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-methyl-1-(3-methylcinnolin-5-yl)urea
[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]({[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl})amine
(3S,4R)-1-[(3-fluoro-4-methoxyphenyl)methyl]-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-[(3-methylquinoxalin-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(morpholin-4-yl)-3-[3-({[2-(pyrazin-2-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
N-(3-hydroxy-3-methylbutyl)-N,2,7-trimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
(1S,5R)-3-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetyl}-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(4aS,7aR)-1-[(2,6-dimethoxyphenyl)methyl]-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{4-[4-(1-propylpiperidin-4-yl)piperazin-1-yl]phenyl}ethan-1-one
1-(4-cyclobutanecarbonyl-1,4-diazepan-1-yl)-2-(dimethylamino)-2-(2-fluorophenyl)ethan-1-one
(2S,4S)-4-(2-propyl-1,3-thiazole-4-amido)pyrrolidine-2-carboxylic acid