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4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-6-[(3-methoxyphenyl)methoxy]-1-(pyridin-2-ylmethyl)-1,4-diazepan-2-one
3-(4-chlorophenyl)-4-{[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}-1H-pyrazole
1-[4-({[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}amino)piperidin-1-yl]ethan-1-one
4-(4-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}phenyl)but-3-yn-1-ol
1-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-5-{2-[(pyridin-3-ylmethyl)amino]ethyl}pyrrolidin-2-one
3-(3,3-diethylpyrrolidine-1-carbonyl)-5-(2-fluorophenoxymethyl)-1H-pyrazole
6-{[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}-N-[1-(naphthalen-1-yl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[1-(3-methylphenyl)-1H-pyrazol-4-yl]pyrimidin-2-amine
6-cyclopentyl-2-methoxy-3-{[(pentan-3-yl)amino]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}urea
4-(4-methoxyphenyl)-3-(4-methyl-1H-imidazol-5-yl)-4H-1,2,4-triazole
(3R,4R)-N-tert-butyl-3-hydroxy-3,4-dimethylpyrrolidine-1-carboxamide
1-[4-methyl-3-(propan-2-yl)phenyl]-3-[1-(pyridin-3-ylmethyl)piperidin-3-yl]urea
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-(3-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-N-methylpropanamide
2,2-dimethyl-5-[4-(3-methylphenyl)piperazine-1-carbonyl]thiomorpholin-3-one
3-[(4-{[4-(methylsulfanyl)phenyl]methyl}piperazin-1-yl)methyl]piperidin-3-ol
2-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1-(furan-3-ylmethyl)-1H-imidazole
2-butyl-8-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-(1-butyl-1H-pyrazol-4-yl)-7,8-dimethyl-4-(pyrrolidine-1-carbonyl)quinoline
2-[1-(furan-3-ylmethyl)-4-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazin-2-yl]ethan-1-ol
N-methyl-3-(4-methyl-1,3-thiazol-5-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
(3S,5R)-1-[(3-hydroxyphenyl)methyl]-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine
4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
(3R,5S)-5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-1-(2-phenylethyl)piperidine-3-carboxamide
N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
5-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]-5-[(3-fluorophenyl)methyl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
4-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-2-oxoethyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
4-{[2-(5-fluoro-2-methoxyphenyl)-1H-imidazol-1-yl]methyl}-3,5-dimethyl-1-(propan-2-yl)-1H-pyrazole
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-2,3-dihydro-1,4-benzodioxine-6-carboxamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(thiophen-3-ylmethyl)piperidin-3-amine
1-(4-methoxyphenyl)-3-methyl-4-(morpholine-4-carbonyl)piperazin-2-one
N-methyl-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[1-(pyridin-3-yl)propyl]acetamide
6-cyclopropyl-4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-3-methyl-[1,2]oxazolo[5,4-b]pyridine
2-butyl-N-(2-hydroxy-3-methoxypropyl)-1,3-benzoxazole-5-carboxamide
2-(difluoromethoxy)-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
N-(1-methyl-1H-pyrazol-3-yl)-2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}acetamide
methyl 1-(6,7-dimethoxy-2-{[methyl(oxolan-3-yl)amino]methyl}quinazolin-4-yl)piperidine-4-carboxylate
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methyl-4-(piperidin-3-ylmethyl)benzamide
N'-(2H-1,3-benzodioxol-5-ylmethyl)-N'-(pentan-3-yl)-N-(1,3,4-thiadiazol-2-yl)ethanediamide
2-amino-1-{3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethan-1-one
methyl 2-(1-{[4-methyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}-3-oxopiperazin-2-yl)acetate
6-[(diethylamino)methyl]-N-[(2R)-oxolan-2-ylmethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-[2-(piperidin-1-ylmethyl)phenyl]-3-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}urea
1-({4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}methyl)piperidine
(2S,4S)-4-amino-N,N-diethyl-1-[2-(4-hydroxypiperidin-1-yl)acetyl]pyrrolidine-2-carboxamide
5-methyl-1'-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2,5-dimethylpyrimidine