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N-[(3S,4R)-1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
N-cyclopentyl-N-({4-[(2-fluorophenyl)methoxy]phenyl}methyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-3-propanamidobenzamide
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
2-(4-methylbenzoyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
1-{2,6-dimethylimidazo[1,2-a]pyridine-3-carbonyl}-4-(5-methylpyridin-2-yl)piperidin-4-ol
N3-cyclooctyl-N5-[(3-fluorophenyl)methyl]-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-{4-[3-(furan-2-yl)benzoyl]-2-oxopiperazin-1-yl}benzonitrile
2-methyl-N-(thiolan-3-yl)pyrido[2,3-d]pyrimidin-4-amine
N-methyl-5-(propan-2-yl)-N-[1-(pyrimidin-4-yl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
8-(5-chlorothiophene-2-carbonyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-(2,6-diaminopyrimidin-4-yl)-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylic acid
2-ethyl-5-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)pyrimidine
N-[2-(propan-2-yloxy)ethyl]-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
1-(4-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidine-1-carbonyl}phenyl)ethan-1-one
{5-[(4-{5-ethyl-6-methylthieno[2,3-d]pyrimidin-4-yl}piperazin-1-yl)methyl]furan-2-yl}methanol
1-(3-{[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-(thiophen-3-yl)ethan-1-one
4-(naphthalen-2-ylmethyl)-3-[2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]piperazin-2-one
2-[methyl(2,2,6,6-tetramethylpiperidin-4-yl)amino]-2-[4-(propan-2-yloxy)phenyl]acetic acid
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[(1r,4r)-4-hydroxycyclohexyl]benzamide
methyl 2-{methyl[1-(4-methylpyridin-2-yl)propan-2-yl]carbamoyl}benzoate
[(2R)-1-[5-(4-methoxyphenyl)furan-2-carbonyl]pyrrolidin-2-yl]methanol
4-[(4-methyl-1H-imidazol-2-yl)methyl]-8-thia-4,6-diazatricyclo[7.6.0.02,7]pentadeca-1(9),2(7),5-trien-3-one
4-benzyl-3-ethyl-1-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)-1,4-diazepan-5-one
2-[4-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)phenyl]-6-(oxolan-3-yl)-3,4-dihydropyrimidin-4-one
4-(2,5-dimethoxyphenyl)-3-(3,3,3-trifluoropropyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-{2-oxo-2-[4-(2-phenoxyethyl)piperazin-1-yl]ethyl}imidazolidine-2,4-dione
5-(1H-indol-1-ylmethyl)-N-(oxan-2-ylmethyl)-1H-pyrazole-3-carboxamide
N-ethyl-2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]-N-(pyridin-4-ylmethyl)acetamide
1-(2H-1,3-benzodioxol-5-yl)-4-[3-(4-chlorobenzoyl)piperidin-1-yl]piperidine
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(2-methylpropanoyl)piperidin-4-yl]oxy}benzamide
N-methyl-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-2-yl)ethyl]acetamide
1-ethyl-4-{[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methyl}-1H-indole
3-[2-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-oxoethyl]-4,5-dimethyl-2,3-dihydro-1,3-oxazol-2-one
3-({[3-(2-amino-1,3-thiazol-4-yl)propyl]carbamoyl}amino)-N,2-dimethylbenzamide
3,4-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propyl-5-sulfamoylbenzamide
2-[1-(2-phenylethyl)-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl]ethan-1-ol
3-(prop-2-en-1-yl)-1-[(1-propyl-1H-pyrazol-4-yl)sulfonyl]piperidine-3-carboxylic acid
2-(2H-1,3-benzodioxol-5-yloxy)-1-[3-(4-fluorophenyl)pyrrolidin-1-yl]ethan-1-one
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-[2-(5-chloro-2-methyl-1H-indol-3-yl)ethyl]acetamide
2-(cyclopropylmethyl)-N-[2-(pyridin-3-yloxy)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-2-(oxan-4-yl)acetamide
N-(pyridin-2-ylmethyl)-4-(1,2,3,4-tetrahydroisoquinolin-7-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-cyano-N-methyl-N-[2-(piperidin-1-yl)ethyl]benzamide
2-amino-N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-2-methylpropanamide
N-[2-(4-ethyl-1,3-thiazol-2-yl)ethyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-3-(1,3,6-trimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
N-(1,3-benzothiazol-6-yl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
8-(butan-2-yl)-1-(2-methoxyethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione