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6-(benzyloxy)-1-[3-(2-oxopyrrolidin-1-yl)propyl]-4-(quinolin-4-ylmethyl)-1,4-diazepan-2-one
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-[2-(1-methyl-1H-imidazol-2-yl)ethyl]benzamide
1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-3-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-5-yl}urea
N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-2-(1H-1,2,4-triazol-1-yl)benzamide
{[2-(4-methoxyphenyl)-7-methylquinolin-3-yl]methyl}(methyl)(pyrimidin-4-ylmethyl)amine
N,6-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-oxo-4-(2-phenylethyl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-({2-[4-(morpholin-4-yl)butoxy]phenyl}methyl)piperidine-4-carbonitrile
(3R,9aR)-3-benzyl-8-(3-methylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-1-(2-methylpropyl)-4-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,4-diazepan-2-one
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(4-methylpiperidine-4-carbonyl)piperidine
N,1-dimethyl-N-{2-phenyl-1-[1-(3-phenyl-1,2-oxazole-5-carbonyl)piperidin-4-yl]ethyl}-1H-pyrazole-3-carboxamide
3-{4-[4-(1,2-oxazolidine-2-carbonyl)phenoxy]piperidine-1-carbonyl}pyridine
1-[2-(4-methoxyphenyl)ethyl]-6-oxo-N-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-3-carboxamide
N-[(3R,5S)-1-cyclopropanecarbonyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-6-methylpyridine-3-carboxamide
(3R,5S)-5-(3-fluorophenoxymethyl)-1-[(4-hydroxyphenyl)methyl]-N-[2-(2-oxoimidazolidin-1-yl)ethyl]piperidine-3-carboxamide
2-(ethylsulfanyl)-5-{[2-(2-methoxyethyl)piperidin-1-yl]methyl}pyrimidine
3-{2-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]ethyl}-1λ6-thiolane-1,1-dione
2-(3-methoxypropyl)-9-(1-methyl-1H-imidazole-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
7-hydroxy-6-methoxy-4-(2-propylpyrimidin-5-yl)-1,2,3,4-tetrahydroquinolin-2-one
(4aR,8aS)-6-[(2,5-dimethylphenyl)methyl]-1-(2-methoxyethyl)-decahydro-1,6-naphthyridin-2-one
1-[4-(aminomethyl)phenyl]-3-[(1,4-dimethylpiperazin-2-yl)methyl]urea
1-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-4-propyl-1,4-diazepan-6-ol
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1-(pyridine-3-carbonyl)piperidin-4-amine
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]acetamide
5-[(3-cyclohexylpyrrolidin-1-yl)methyl]-3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazole
N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-4-methylpiperidine-4-carboxamide
N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
2-[1-(2,2-dimethylpropyl)-4-[(3-methyl-1H-indol-2-yl)methyl]piperazin-2-yl]ethan-1-ol
2-{1-[(1S)-1-carbamoyl-2-methylpropyl]-1H-imidazol-2-yl}benzoic acid
3-(4-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-6-yl)pyridine
2-(4-methanesulfonylphenyl)-1-{2-oxa-7-azaspiro[4.5]decan-7-yl}ethan-1-one
(1,4-dioxan-2-ylmethyl)[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]methylamine
N-{1-[(4-methylphenyl)methyl]cyclopropyl}-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide
N4,6-dimethyl-N4-[(4-methyl-1,3-thiazol-2-yl)methyl]-5-(prop-2-en-1-yl)pyrimidine-2,4-diamine
1-[3-(3-methylphenoxymethyl)piperidin-1-yl]-4-(morpholin-4-yl)butan-1-one
3-[(3R,4S)-1-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
1-[4-({[1-(2-methoxyethyl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl)amino)piperidin-1-yl]ethan-1-one
2-(4-fluorophenoxymethyl)-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1,3-oxazole-4-carboxamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxybenzene-1-sulfonamide
1-{2-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]-5-propyl-1,3,4-oxadiazol-2-amine
2-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-[4-(4-phenyl-1H-imidazol-5-yl)thiophen-2-yl]ethan-1-one
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
3-[(1H-indol-4-ylmethyl)amino]-1-(1,2,3,4-tetrahydroquinolin-1-yl)propan-1-one
2-[(4aS,8aR)-6-[(4-chlorophenyl)methyl]-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-1-yl]acetamide
4-({3-methoxy-2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)piperazin-2-one
3,5-dimethyl-1-[1-(thiophen-3-ylmethyl)azetidin-3-yl]-1H-pyrazole
2-(1-benzyl-4-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}piperazin-2-yl)ethan-1-ol
1-{[1-(1-ethylpiperidin-3-yl)piperidin-3-yl]methyl}pyrrolidin-2-one