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N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-2-oxo-4-phenylbutanamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-amine
4-{[(dimethylsulfamoyl)amino]methyl}-1-(2-phenoxyethyl)azepan-4-ol
(2R)-N1-{3-chloro-4-[(propan-2-yl)carbamoyl]phenyl}pyrrolidine-1,2-dicarboxamide
N-(3,4-dimethylphenyl)-1-(oxan-4-yl)piperidin-3-amine
(2S)-2-amino-3-(1H-imidazol-4-yl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
3-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-6-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
N-benzyl-1-(4,7-dimethylquinazolin-2-yl)azepan-4-amine
3-{[1-butyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}-1λ6-thiolane-1,1-dione
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]ethan-1-one
1-(2-{[(4-hydroxy-5,8-dimethylquinolin-2-yl)methyl]amino}ethyl)imidazolidin-2-one
methyl 3-[1-(4-chlorophenyl)cyclopropaneamido]-5-{[3-(dimethylcarbamoyl)propanamido]methyl}benzoate
2-({[1-(thiophen-3-ylmethyl)piperidin-3-yl]oxy}methyl)pyridine
N-(cyclopent-3-en-1-yl)-2-(4-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}morpholin-3-yl)acetamide
N-ethyl-1-(furan-2-ylmethyl)-N-(pyridin-4-ylmethyl)piperidin-3-amine
4-[7-(3-methylbut-2-enoyl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
2-(4-{[2-(furan-2-yl)phenyl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
methyl 5-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
(3aS,6aS)-2-[(2-chloro-4-fluorophenyl)methyl]-5-(dimethylcarbamoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}azetidin-3-yl)-3,5-dimethyl-1H-pyrazole
3-ethyl-5-{[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-pyrazole
3-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-1-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]urea
6-(3-chlorophenyl)-N-ethyl-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-amino-2-methyl-1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]propan-1-one
4-(cyclopropylmethyl)-1-[2-(methylsulfanyl)pyrimidine-5-carbonyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-[(4-fluorophenyl)methyl]-3-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)propanamide
2-(3-fluoro-5-methylphenyl)-6-(piperidine-1-carbonyl)pyrazine
2-{4-[(4-ethoxyphenyl)methyl]-1-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
1-[5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]azonane
2-(1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)-1,3-benzoxazole
2-(5-{2-[(dimethylamino)methyl]phenyl}-1-(3-fluorophenyl)-1H-1,2,4-triazol-3-yl)acetamide
N-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-chlorobenzamide
2,6-difluoro-N-({7-[(4-phenyl-1,3-thiazol-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
7-[(2-fluorophenyl)methyl]-2-[(2E)-2-methylbut-2-en-1-yl]-2,7-diazaspiro[4.5]decan-6-one
(3S,4S)-4-(morpholin-4-yl)-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}pyrrolidin-3-ol
methyl({[4-(2-methylphenyl)phenyl]methyl})({5-[(oxolan-2-ylmethyl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)amine
methyl[(3-methyl-1,2-oxazol-5-yl)methyl][3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propyl]amine
N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methyl-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamide
1-(2-methoxyphenyl)-3-(2-methylpropyl)-5-(1H-1,2,4-triazol-5-yl)-1H-1,2,4-triazole
methyl 6-(azepan-1-ylmethyl)-3-(thiophene-3-amido)thieno[2,3-b]pyridine-2-carboxylate
2-methyl-8-{[2-(2-phenylethoxy)phenyl]methyl}-2,8-diazaspiro[4.5]decan-3-one
4-(4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-5-methyl-2-oxopiperazin-1-yl)benzonitrile
ethyl 2-(4-{[3-(methanesulfonylmethyl)piperidine-1-carbonyl]amino}phenyl)acetate
3-({ethyl[2-(pyrrolidin-1-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
1-(3-{[3-(2-methylphenoxy)azetidin-1-yl]methyl}phenyl)ethan-1-one
methyl 8-(2,2-diphenylacetyl)-1-methoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
4-(4-methylphenyl)-3-[(propan-2-yloxy)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-1-ethyl-N-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
4-ethyl-1-[(4-methoxypyridin-2-yl)methyl]-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one