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6-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]pyrimidine-2,4-diamine
4-(4-chloro-2-hydroxybenzoyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
(4S)-3-[(3,4-difluorophenyl)methyl]-4-(propan-2-yl)-1,3-oxazolidin-2-one
N-[3-({[1-(2-methoxyphenyl)propan-2-yl]amino}methyl)-5-(pyrrolidine-1-carbonyl)phenyl]acetamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
5-(2-chloro-4-fluorophenoxymethyl)-N-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}-1,2-oxazole-3-carboxamide
(1S,5R)-N-(3-carbamoyl-4-methoxyphenyl)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carboxamide
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-(2-hydroxy-3-methoxypropyl)propanamide
2-(2-fluoro-3-methoxyphenyl)-5-(methanesulfonylmethyl)pyridine
1-cyclopentyl-N-(2,3-dihydro-1H-inden-2-yl)-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
(2R,4S)-1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-hydroxypiperidine-2-carboxylic acid
1-{2-[(2-chlorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-(2-hydroxyethyl)piperidine-3-carboxamide
2,7,8-trimethyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)quinoline-4-carboxamide
N,N-dimethyl-1-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}pyrrolidin-3-amine
1-(2H-1,3-benzodioxol-5-yl)-5-[1-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1H-1,2,4-triazole
1-[(2-cyclohexylpyrimidin-5-yl)methyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
3-(furan-2-yl)-5-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-[(4-fluorophenyl)methyl]-3-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]propanamide
2-(3-methoxyphenyl)-3-[(4-methoxypiperidin-1-yl)methyl]-7-(methylsulfanyl)quinoline
3-methyl-N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
2-fluoro-5-[4-(2-hydroxyethyl)-1H-pyrazol-1-yl]benzoic acid
ethyl 4-[(2-chlorophenyl)methyl]piperidine-4-carboxylate
1-(furan-2-ylmethyl)-N-methyl-N-[2-(pyridin-4-yl)ethyl]piperidine-3-carboxamide
3-(2-{cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
2-[1-benzyl-4-(9H-purin-6-yl)piperazin-2-yl]ethan-1-ol
5-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1,3-benzothiazole
4-(6-cyclopropylpyrimidin-4-yl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{4-[6-(dimethylamino)pyrimidin-4-yl]-6-hydroxy-1,4-diazepan-1-yl}propanoic acid
3-{2-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]-2-oxoethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
2-(2-{[methyl(oxan-2-ylmethyl)amino]methyl}phenoxy)-1-(piperidin-1-yl)ethan-1-one
2-[2-(dimethylamino)ethyl]-9-(5-propylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
3,5-dichloro-N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N,4-dimethylbenzamide
5-methoxy-3-methyl-2-({4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}methyl)-1H-indole
[(2-methoxypyrimidin-5-yl)methyl]({[4-(methylsulfanyl)phenyl]methyl})propylamine
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-3-(2-methylphenyl)-3-phenylpropanamide
N-[3-(4-{[(5-chlorothiophen-2-yl)methyl]amino}piperidin-1-yl)phenyl]-2-methoxybenzamide
5-[(2S)-oxolan-2-yl]-3-(thiophen-3-yl)-1,2,4-oxadiazole
1-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(morpholin-4-yl)ethan-1-one
5-[2-(6-methoxynaphthalen-2-yl)morpholine-4-carbonyl]-2-methylphenol
3-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-(3,4,5-trimethoxyphenyl)urea
2-[(isoquinolin-5-yloxy)methyl]-N-[(5-methylfuran-2-yl)methyl]-1,3-oxazole-4-carboxamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(oxolan-3-ylmethyl)piperidine-4-carboxamide
2-(2-{1-[3-(1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
N-[3-(1H-indol-1-yl)propyl]-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
5-{2-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-2-oxo-1,3-oxazolidine-4-carboxamide
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1-[4-methyl-6-(propan-2-yl)quinazolin-2-yl]piperidine-4-carboxamide
1-methyl-3-{2-oxo-2-[4-(thiomorpholin-4-yl)piperidin-1-yl]ethyl}-3-(4-phenylphenyl)pyrrolidine-2,5-dione
1-[5-(4-chlorophenyl)-1,2,4-triazin-3-yl]azocane
4-(2-methyl-1H-imidazol-1-yl)-1-[3-(2-phenylacetyl)piperidin-1-yl]butan-1-one