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3-({1-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]piperidin-4-yl}methyl)benzoic acid
3-(2-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-oxoethyl)-4-methylpiperazin-2-one
2-[3-(4-fluorophenoxymethyl)-5-(1-methanesulfonamidoethyl)-1H-1,2,4-triazol-1-yl]acetic acid
N-methyl-2-[2-(1-{[(1-methyl-1H-indazol-3-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)phenoxy]acetamide
3-{1-methyl-5-[5-(oxolan-2-yl)thiophen-2-yl]-1H,4H-pyrazolo[3,4-d]imidazol-3-yl}pyridine
N-(2-methoxyethyl)-3-(2-methyl-1H-indol-1-yl)-N-(1-methylpiperidin-4-yl)propanamide
4-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetyl}-1-(4-methylphenyl)piperazin-2-one
5-[1-(cyclohex-1-ene-1-carbonyl)piperidin-4-yl]-3-(oxolan-2-ylmethyl)-5-(pyridin-3-yl)imidazolidine-2,4-dione
N-{[7-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(phenylsulfanyl)acetamide
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-N-{[2-(trifluoromethyl)phenyl]methyl}propanamide
4-cyclobutyl-N-[(5-ethylpyridin-2-yl)methyl]-6-methylpyrimidin-2-amine
2-{2-[3-(benzyloxy)phenyl]-1H-imidazol-1-yl}ethan-1-ol
(3R,4R)-4-cyclobutyl-1-({2-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-3-methylpiperidin-4-ol
2-methyl-8-{[5-(1,3-oxazol-5-yl)thiophen-2-yl]sulfonyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-(4-ethyl-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-(thiophen-3-ylmethyl)acetamide
(5-{1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1H-imidazol-2-yl}furan-2-yl)methanol
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
N-cyclopropyl-1-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-1-methyl-N-(pyridin-4-ylmethyl)azepane-2-carboxamide
2-{[2-(2,3-dihydro-1H-indol-1-yl)ethyl]amino}propan-1-ol
(3S)-1-{1-methyl-5-[3-(pyridin-2-yl)azetidine-1-carbonyl]-1H-1,3-benzodiazol-2-yl}pyrrolidin-3-ol
1'-(2-propoxyethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-phenyl-5-{[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}-1,3-thiazole
N-[(2R)-1-(benzyloxy)-3-hydroxypropan-2-yl]-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
3-[5-(2-fluorobenzenesulfonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
1-(carbamoylmethyl)-N-{[1-(2-fluorophenyl)pyrrolidin-3-yl]methyl}piperidine-4-carboxamide
ethyl 2-{1-[(5-methoxy-1H-indazol-3-yl)methyl]piperidin-2-yl}acetate
(2S)-4-methyl-2-[2-(2,3,6-trimethylphenoxy)acetamido]pentanamide
2-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-N,1-bis(propan-2-yl)-1H-1,3-benzodiazole-5-sulfonamide
1-[3-(piperidin-4-ylmethyl)benzoyl]-4-(trifluoromethyl)piperidine
1-(3-hydroxy-4-methoxyphenyl)-5-oxopyrrolidine-3-carboxylic acid
5-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)imidazolidine-2,4-dione
6-(2-methylpropyl)-4-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydropyrimidin-2-one
[1-({1-[(4-chloro-1-methyl-1H-pyrazol-3-yl)methyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
5-butyl-4-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-1-(3-methylphenyl)piperazin-2-one
2-(1-benzyl-3-oxopiperazin-2-yl)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}acetamide
N-[2-(1-hydroxycyclopentyl)ethyl]-4-methylpyrimidine-5-carboxamide
1-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}-4-(pyrrolidine-1-sulfonyl)piperazine
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-phenoxyacetamide
4-chloro-N-[(3R,4S)-4-cyclopropyl-1-(4-methylpent-3-en-1-yl)pyrrolidin-3-yl]-1-methyl-1H-pyrazole-5-carboxamide
9-(3,5-dimethyl-1-benzofuran-2-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
4-(5-{4-[(2-fluorophenyl)methyl]piperidine-1-carbonyl}pyrimidin-2-yl)morpholine
2-(2-chlorophenyl)-N-[(4-hydroxyphenyl)methyl]-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-[(4aR,8aS)-1-(furan-2-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-4-phenylbutan-1-one
N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(oxolan-2-ylmethyl)-2-(thiophen-2-yl)acetamide
1-ethyl-N-methyl-3-(2-methylpropyl)-N-[(1-phenylpyrrolidin-3-yl)methyl]-1H-pyrazole-5-carboxamide
(1S,5R)-6-propyl-3-[4-(1H-pyrazol-3-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(dimethylamino)ethyl]-2-(2-fluorophenyl)-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)acetamide
3-[(4-fluorophenyl)formamido]-N-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]propanamide
{5-[3-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]pyridin-2-yl}methanamine