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N3-[2-(4-fluorophenyl)ethyl]-N5-methyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-[4-(1H-indol-2-ylmethyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
ethyl 2-[4-(2-methoxyphenoxy)piperidin-1-yl]-1,3-oxazole-4-carboxylate
N,2,6-trimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]pyrimidine-4-carboxamide
2-benzyl-8-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
3-{2-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
1-[5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-2-methyl-1,4-diazepan-5-one
1-[3-(thiomorpholine-4-carbonyl)benzenesulfonyl]-1,4-diazepane
2,2-dimethyl-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-4-oxo-3,4-dihydro-2H-pyran-6-carboxamide
1-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
4-{[2-(2-carboxyethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]methyl}benzoic acid
({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
4-(piperidin-1-yl)-1-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)piperidine-4-carboxamide
2-ethyl-4-methyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,3-oxazole-5-carboxamide
8-(6-methylpyridine-3-carbonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)benzamide
(4S)-1-[(2,6-dimethoxyphenyl)methyl]-3,3,4-trimethylpiperidin-4-ol
(1R,5R)-6-benzyl-3-[4-(difluoromethoxy)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-3,3,3-trifluoropropanamide
3-[1-(morpholin-4-ylmethyl)cyclopentyl]-1-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
1-{2-oxo-2-[4-(oxolane-2-carbonyl)-1,4-diazepan-1-yl]ethyl}-1,2-dihydroquinolin-2-one
3-{3-[methyl(2-methylpropyl)amino]propyl}-8-(6-oxo-1,6-dihydropyridine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]naphthalene-2-carboxamide
1-(4,7-dimethylquinazolin-2-yl)-N-(oxan-4-ylmethyl)azepan-4-amine
N-({1-[(6-chloropyridin-3-yl)methyl]pyrrolidin-3-yl}methyl)-6-methylpyridine-3-carboxamide
1-ethyl-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-[(4-methoxypyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-5-methyl-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
2-(benzyloxy)-1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]ethan-1-one
4-{2-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}-1-(propan-2-yl)-1H-pyrazole
2-methyl-5-[4-(2-phenoxyethyl)phenyl]-1,3,4-oxadiazole
1-(4-ethylpiperazin-1-yl)-3-[2-methoxy-4-({methyl[2-(oxan-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
methyl 3-{4-[2-amino-3-cyano-6-(6-methoxypyridin-3-yl)pyridin-4-yl]-1H-pyrazol-1-yl}propanoate
N-(2-hydroxyethyl)-3,5,7-trimethyl-N-[(3-methylthiophen-2-yl)methyl]-1H-indole-2-carboxamide
3-({[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
5-({[(3-{2-[4-(4-methoxybenzenesulfonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
1-[2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-3-ethylpiperidin-3-ol
4-(4-methanesulfonyl-1,4-diazepane-1-carbonyl)-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
6-(1-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-3-yl)-3,4-dihydropyrimidin-4-one
methyl 2-(2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamido)acetate
2-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-1,3-thiazole-4-carboxamide
2-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-6-(methoxymethyl)pyridine
2-{[1-(4-phenylphenyl)ethyl]amino}propane-1,3-diol
N-[2-(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)-2-oxoethyl]acetamide
N-[2-(dimethylamino)ethyl]-2-(3-fluorophenyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)acetamide
methyl 1-[(3S,5S)-5-{[3-(methylsulfanyl)phenyl]carbamoyl}-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-[(1R)-1-(3-methoxyphenyl)ethyl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
4-amino-N-(butan-2-yl)-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
1-ethyl-5-{methyl[(2-methylpyridin-4-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-[2-(4-phenylpyrimidin-2-yl)ethyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide