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[3-(furan-3-ylmethyl)-9-(1H-imidazol-2-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
N-[(3S,4R)-1-(2H-1,3-benzodioxole-5-carbonyl)-4-propylpyrrolidin-3-yl]acetamide
2-methyl-4-phenyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyridine-3-carboxamide
(7S,9aR)-7-methyl-6,9-dioxo-N-phenyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
6-fluoro-N-methyl-2-oxo-N-(quinoxalin-6-ylmethyl)-1,2,3,4-tetrahydroquinoline-4-carboxamide
5-[2-(dimethylamino)-2-(3-methylphenyl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
N-(6-methoxy-2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)-2-(4-methyl-1,4-diazepan-1-yl)acetamide
4,6-dimethyl-5-{2-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidin-2-ol
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(2,4-diethoxy-3-methylphenyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-(2-methyl-1H-imidazol-1-yl)-1-[3-(thiophen-3-yl)propanoyl]piperidine-4-carboxylic acid
5-[2-(3-fluoro-4-methylphenyl)acetyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-ethyl-1-[4-(pyrrolidin-1-ylmethyl)benzoyl]piperidine-3-carboxylic acid
4,6-dimethyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}pyridine-3-carboxamide
1-[(3-fluorophenyl)methyl]-4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperazin-2-one
4-methyl-N-[4-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]-1,2,3,6-tetrahydropyridine-1-carboxamide
5-{4-[1-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}-2,1,3-benzoxadiazole
1-ethyl-3-methyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-1H-pyrazole-5-carboxamide
N-(4-acetylphenyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
{[1-butyl-2-(cyclohexanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(1-methylpiperidin-2-yl)methyl]amine
8-methyl-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 3-{[1-(cyclopropylmethyl)-5-(quinoxalin-5-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
N-methyl-1-{[(2,3,5-trifluorophenyl)carbamoyl]amino}cyclohexane-1-carboxamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
(3aS,6aR)-5-(1,3-dihydroxypropan-2-yl)-3-[(3,4-dimethoxyphenyl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
methyl 5-{[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]sulfonyl}-1-methyl-1H-pyrrole-2-carboxylate
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
N-(3,4-dimethylphenyl)-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
2-(2-chlorophenyl)-2-{[5-(propan-2-yl)-1,2-oxazol-3-yl]formamido}acetic acid
4-(4-phenyl-1H-1,2,3-triazol-1-yl)-1-(thian-4-yl)piperidine
2-(2-chloro-6-methoxyphenyl)-2-(4-cyclopentyl-3-oxopiperazin-1-yl)acetic acid
4-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-1,4-oxazepan-6-ol
4-[2-(3-cyclobutyl-1,2,4-oxadiazol-5-yl)ethyl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
3-(piperidine-1-carbonyl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}pyrazine-2-carboxamide
1-[(4-chlorophenyl)methyl]-4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]piperidine
methyl 5-({4-[(ethylcarbamoyl)methyl]piperazin-1-yl}methyl)-2-hydroxybenzoate
3-(benzyloxy)-1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidine
2-[4-(2-fluorophenyl)piperazine-1-carbonyl]-3,4-dihydroquinazolin-4-one
N-(3-chloro-4-fluorophenyl)-N'-ethyl-N'-(pyridin-4-ylmethyl)butanediamide
5-(3-fluoro-4-methoxyphenyl)-N-(oxan-2-ylmethyl)-1,2,4-triazin-3-amine
(3aR,6aR)-2-(cyclobutylmethyl)-5-[(2-fluoro-4-methoxyphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[4-ethyl-5-oxo-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N,N-dimethylpropane-1-sulfonamide
methyl (2S,4R)-1-[(2,6-difluorophenyl)methyl]-4-(2,3-dimethyl-1H-indole-7-amido)pyrrolidine-2-carboxylate
(2E)-1-{3-[(2,4-difluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}-3-(4-methoxyphenyl)prop-2-en-1-one
3-(4-{2-[(4-methylpiperidin-1-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-1H-1,2,3-triazol-1-yl)propan-1-amine
2-(dimethylamino)-2-(3-fluorophenyl)-N-[2-(quinolin-8-yloxy)ethyl]acetamide
2-ethyl-4-phenyl-9-(1,3-thiazol-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(6-methoxypyridazin-3-yl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
(1S,5R)-3-{3-fluoro-8-methylimidazo[1,2-a]pyridine-2-carbonyl}-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2,6-dimethyl-N-{3-[(pyridin-3-yl)amino]propyl}quinoline-4-carboxamide