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N-[2-(2-methoxyphenyl)ethyl]-2-[2-(trifluoromethyl)morpholin-4-yl]acetamide
(2S,4R)-4-amino-1-(2,3-dimethyl-1H-indole-5-carbonyl)-N-methylpyrrolidine-2-carboxamide
6-(2,5-dimethoxyphenyl)-N-[(2-fluorophenyl)methyl]-2-(4-methylpiperazin-1-yl)pyridine-3-carboxamide
6-[(6-chloro-4-oxo-4H-chromen-3-yl)methyl]-N-[2-(1H-indol-3-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
2-[2-methoxy-6-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]propanoic acid
3-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}-N-(3-methoxyphenyl)propanamide
2-(2,3-dichlorophenyl)-1,3-thiazole-4-carboxamide
2-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{4-[1-(furan-2-carbonyl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine
N-(2,4-dimethylphenyl)-N'-[(4-methoxyphenyl)methyl]-N'-(prop-2-yn-1-yl)propanediamide
1-{2-methoxy-4-[(4-methoxypiperidin-1-yl)methyl]phenoxy}-3-(morpholin-4-yl)propan-2-ol
2-(3-phenylpropyl)-4-[(trimethylpyrazin-2-yl)methyl]morpholine
2-{4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
(2E)-N-({3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-3-(thiophen-2-yl)prop-2-enamide
N-(1-benzothiophen-2-ylmethyl)-1-[2-(1,1-dioxo-1λ6-thiolan-3-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-methylpiperidine-3-carboxamide
2-(2-methoxy-4-methylphenoxymethyl)-N-[(6-methylpyridin-2-yl)methyl]-1,3-oxazole-4-carboxamide
N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-2-(pyridin-4-yl)ethane-1-sulfonamide
N-methyl-N-[2-(pyridin-2-yl)ethyl]-3-{1-[3-(pyridin-4-yl)propanoyl]piperidin-3-yl}propanamide
methyl 1-[(3R,5S)-1-(2-ethylbutyl)-5-{[3-(methylsulfanyl)phenyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-2-methylpropan-1-one
2-ethyl-5-[(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)methyl]pyrimidine
N-ethyl-2-{4-[1-(pyridin-2-yl)piperidine-3-carbonyl]piperazin-1-yl}acetamide
N-{5H,6H,7H-cyclopenta[b]pyridin-3-ylmethyl}-6-methyl-2-(pyridin-3-yl)pyrimidin-4-amine
4-[5-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carbonyl)furan-2-yl]-2-methylbut-3-yn-2-ol
N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-4-(pyridin-2-yl)pyrimidin-2-amine
1-(4-methylquinazolin-2-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)pyrrolidine-2-carboxamide
N-cyclopropyl-1-[(2-methylphenyl)methyl]-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(oxan-4-yl)piperazine
N-{2-[7-(2,3-dihydro-1-benzofuran-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}furan-3-carboxamide
2-(2-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethyl)pyridine
4-(3-fluorobenzoyl)-7-(pyridin-3-yl)-9-[2-(thiophen-2-yl)ethoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-({3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-2-(pyridin-2-yl)pyrimidine
1-(3-ethynylbenzoyl)-3-(4-methoxy-2-methylbenzoyl)piperidine
6-[4-(1-ethoxyethyl)phenyl]-N4,N4-dimethylpyrimidine-2,4-diamine
methyl 5-{[(3,4-dimethylphenyl)methyl]amino}-1-ethyl-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(2-{7-[(2,4-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
1-methyl-2-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}[(2-methylphenyl)methyl](prop-2-en-1-yl)amine
2-(4-{3-[1-(dimethylamino)ethyl]phenyl}-1H-pyrazol-1-yl)-N-methylacetamide
8-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
3-{1-[(2,6-dimethoxyphenyl)methyl]piperidin-4-yl}-N-[2-(dimethylamino)ethyl]propanamide
N-(2-phenylphenyl)-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carboxamide
N-(pyridin-3-ylmethyl)-3-[1-(thian-4-yl)piperidin-4-yl]propanamide
(2S,4S)-4-amino-1-[2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetyl]-N-methylpyrrolidine-2-carboxamide
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[3-(methylsulfanyl)propyl]-1H-pyrazole-3-carboxamide
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-6-(methoxymethyl)pyrimidin-4-amine
2-cyclopropyl-N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-N-[(4-phenyloxan-4-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{2-[(3,5-dimethyladamantan-1-yl)oxy]ethyl}acetamide