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2-[2-chloro-4-({[2-(1-hydroxycyclopentyl)ethyl](methyl)amino}methyl)phenoxy]acetamide
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
5-(5-acetylthiophen-2-yl)-N-butylfuran-2-carboxamide
(1R,5R)-6-[(2-butyl-1H-imidazol-4-yl)methyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-methyl-3-(2-methyl-1H-indol-1-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]propanamide
N-[(3S,4R)-1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
ethyl 2-[1-(6-methoxy-1-methyl-1H-indole-2-carbonyl)piperidin-2-yl]acetate
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
1-(3-{2-[(2-methoxyethyl)sulfanyl]-5-(3-methoxyphenyl)pyrimidin-4-yl}piperidin-1-yl)-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-methoxy-N-methyl-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-(6-carbamoylpyrazin-2-yl)-4-phenoxypiperidine-4-carboxylic acid
(1R,5S,6S)-6-({4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-3-azabicyclo[3.1.0]hexane
4-methoxy-3,5-dimethyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}benzamide
(3aR,6aS)-N-{4-[ethyl(phenyl)carbamoyl]phenyl}-octahydropyrrolo[3,4-c]pyrrole-2-carboxamide
1-{4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}-2-(pyridin-2-yl)ethan-1-one
3-(azepane-1-carbonyl)-1-ethyl-N-[(3,4,5-trifluorophenyl)methyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
2-{3-[2-(4-fluorophenyl)morpholine-4-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}ethan-1-ol
[(3R,4S)-4-[(4-methylpiperazin-1-yl)methyl]-1-{[3-(morpholin-4-yl)phenyl]methyl}pyrrolidin-3-yl]methanol
4-(5-{3-[(2-fluorophenyl)methoxy]azetidine-1-carbonyl}-1H-pyrazol-3-yl)phenol
1'-(2-ethylpyridine-4-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
7-[(2,3-dimethoxyphenyl)methyl]-2-(pyridin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-{4-[(2-ethoxyphenyl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
3-{2-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-[2-(1H-pyrazol-1-yl)ethyl]-1,4-diazepan-5-one
(3S,4S)-1-(6-oxo-1,6-dihydropyridazine-3-carbonyl)-4-propylpyrrolidine-3-carboxylic acid
2-amino-4-[1-(propan-2-yl)piperidin-4-yl]-6-(3,4,5-trifluorophenyl)pyridine-3-carbonitrile
4-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carbonyl)piperazine-1-carbaldehyde
3-(1,4-diazepane-1-sulfonyl)-N-(pyridin-3-ylmethyl)benzamide
5-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-[(3-methoxyphenyl)methyl]-4-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]morpholine
(1S,5R)-6-[(5-ethylpyridin-2-yl)methyl]-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-[3-(2,4-dimethyl-1,4-diazepane-1-carbonyl)phenyl]propanamide
4-(piperidin-1-ylmethyl)-N-[2-(pyridin-4-yl)ethyl]benzamide
5-(morpholine-4-sulfonyl)-2-[(2R)-oxolane-2-carbonyl]-1,2,3,4-tetrahydroisoquinoline
1,3-dimethyl-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-methylpyrimidine-5-carboxamide
1-(1-{[4-(difluoromethoxy)phenyl]methyl}piperidin-4-yl)piperidine-4-carboxylic acid
2-{[3-(oxolan-3-yl)propyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
(3R,4S)-4-[(2,1,3-benzoxadiazol-4-ylmethyl)(methyl)amino]oxolan-3-ol
N-[4-(3-methylphenyl)phenyl]-1-propanoylpiperidine-4-carboxamide
1-(5-ethyl-1,2-oxazole-4-carbonyl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
methyl[(2-methyl-1H-imidazol-4-yl)methyl][1-(pyrazin-2-yl)propan-2-yl]amine
2-[(E)-2-(4-methoxyphenyl)ethenyl]-1H-1,3-benzodiazole-5-carbonitrile
2-(4-methylphenyl)-2-[4-(piperidin-1-yl)butanamido]acetic acid
3-(1-methyl-1H-1,2,3-triazol-4-yl)-1-(pyridin-3-ylmethyl)-1-(1,2,3,4-tetrahydronaphthalen-1-yl)urea
2-{4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(3-methylbut-2-en-1-yl)piperazin-2-yl}ethan-1-ol
(1R,3S)-3-{2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}cyclopentan-1-amine
ethyl 2-({[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)amino)acetate
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide