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1-({1-[6-(cyclopropylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-3-yl}methyl)pyrrolidin-2-one
4-[(3-fluorophenyl)methyl]-11-(morpholin-4-yl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
methyl 5-[(6-acetamidoquinolin-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-5-(morpholin-4-ylmethyl)furan-3-carboxamide
1-(1-{[5-(1-methyl-1H-1,3-benzodiazol-2-yl)furan-2-yl]methyl}piperidin-4-yl)pyrrolidin-2-one
1-[3-(2-ethylphenoxy)azetidin-1-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
N-[(2S)-1-[4-(3-cyanophenyl)-3-oxopiperazin-1-yl]-3-(1H-imidazol-4-yl)-1-oxopropan-2-yl]acetamide
(1S,5R)-N-(4-methylphenyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-[(2,4-difluorophenyl)methyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
1-[2-(2-fluorophenoxy)phenyl]-3-[3-(oxolan-3-yl)propyl]urea
N-(4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}phenyl)acetamide
3-{4-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1H-1,2,3-triazol-1-yl}propan-1-amine
4-{4-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-2-oxopiperazin-1-yl}benzonitrile
1-(cyclopropylmethyl)-5-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(2-methoxyphenyl)methyl]-N3-(3-methylbutyl)-4-oxo-N5-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
5-ethyl-5-{1-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
N-{1-azabicyclo[2.2.2]octan-3-yl}-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
5-(4-acetylphenoxymethyl)-N-(2-phenylpropyl)-1,2-oxazole-3-carboxamide
N-ethyl-N-[2-(2-methylphenoxy)ethyl]-1-benzofuran-2-carboxamide
4-{5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carbonyl}-1,4-diazepane-1-carbaldehyde
5-cyclopropyl-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-1H-pyrazole-3-carboxamide
N-(2-chlorophenyl)-3-{1-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}propanamide
1-(1-cyclopentylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
3-[2-(4-fluorophenyl)ethyl]-1-(1,3-thiazol-4-ylmethyl)piperidine
1-{3-[(1-cyclopentylpiperidin-4-yl)oxy]benzoyl}piperidine-4-carboxamide
4-(2-methylpyrrolidine-1-carbonyl)-N-[2-(1H-pyrrol-1-yl)ethyl]benzene-1-sulfonamide
ethyl 4-[(3-methoxyphenyl)methyl]-1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidine-4-carboxylate
N-(1-{7-[(4-fluoro-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylpropanamide
2-amino-4-(1H-imidazol-4-yl)-6-(1-propyl-1H-1,2,3-benzotriazol-5-yl)pyridine-3-carbonitrile
{3-[(4-fluorophenyl)methyl]-1-(quinoxalin-2-yl)piperidin-3-yl}methanol
N-[(2S)-1-methoxypropan-2-yl]-5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-amine
(4aR,7aS)-1-acetyl-4-[(2-methylpyrimidin-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-chloro-3-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
5-(3-methylpiperazine-1-carbonyl)-N-(propan-2-yl)pyrimidin-2-amine
N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
3-[2-(4-methoxyphenyl)phenyl]-1-[(1-methylpiperidin-2-yl)methyl]urea
{2-[4-(2-amino-1,3-thiazol-4-yl)phenyl]phenyl}methanol
3-phenyl-N-(1-{1-[3-(pyridin-3-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
N-[(3-methoxyphenyl)methyl]-6-methyl-2-(morpholin-4-yl)pyrimidin-4-amine
N-[(1S,2R)-2-[(oxan-4-yl)amino]cyclobutyl]-2-(phenylamino)pyrimidine-5-carboxamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetamide
2-{4-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
2-(2-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-oxoethyl)-2,3-dihydro-1H-indazol-3-one
1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-4-(pyridin-2-ylmethyl)-1,4-diazepane
4-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]morpholine-2-carboxylic acid
methyl (2S)-1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidine-2-carboxylate
(1S,5R)-3-(2-phenoxyethyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-3-(pyridin-3-yl)propanamide
1-{1-[(1-hexylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}propan-2-ol
4-{2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1-benzofuran-5-yl}-1-[(2,4-dimethylphenyl)methyl]piperidin-4-ol