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3-{1-[(2-methylphenyl)methyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
4-{1,1-dimethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-2-(3-fluorophenoxymethyl)-1,3-oxazole
N-[(2-{3-[2-(4-methoxyphenyl)acetamido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-2-methylfuran-3-carboxamide
8-[2-(2-fluorophenyl)acetyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1,5,6-trimethyl-3-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
N-[2-(azepan-1-yl)-2-phenylethyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
2-{2-[1-(1H-indazole-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-3-sulfamoylthiophene-2-carboxamide
1-[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidine-3-carbonitrile
1-{5-[(2E)-but-2-en-1-yl]-1,3,4-oxadiazole-2-carbonyl}-4-[(3-methylpyridin-2-yl)methyl]piperazine
[9-(4-cyclopentylpyrimidin-2-yl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
1-(4-fluorophenyl)-4-[3-(1H-pyrazol-4-yl)propyl]piperazine
methyl 8-[(3-methoxyphenyl)methyl]-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
N-{1-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-2-methyl-1-oxopropan-2-yl}thiophene-2-carboxamide
2-(3-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-ylmethyl}-2-methyl-1H-indol-1-yl)acetamide
N-(4-methoxy-2-methylphenyl)-3-[1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidin-3-yl]propanamide
(3S,9aR)-3-benzyl-8-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-[(3,4-dimethoxypyridin-2-yl)methyl]-5-methyl-1-(4-methylphenyl)piperazin-2-one
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
2-benzyl-9-(dimethyl-1,3-oxazole-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(3-chloro-1,2-oxazol-5-yl)-N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}propanamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-{4-[2-(3-methylphenyl)acetamido]-1H-pyrazol-1-yl}benzamide
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-amine
1-(2-chlorophenyl)-3-[2-(4-ethylmorpholin-2-yl)ethyl]urea
N-[3-(cyclohexylsulfanyl)propyl]-1-(4-hydroxyphenyl)-5-oxopyrrolidine-3-carboxamide
(3S,4R)-1-[2-(azepan-1-yl)acetyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
2-{[1-(pyridin-3-yl)propan-2-yl]amino}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
4-(5-{[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
(3S,4R)-4-(4-fluorophenyl)-1-(oxan-4-yl)pyrrolidine-3-carboxylic acid
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N,5,6-trimethylpyrimidin-4-amine
6-(2-chlorophenyl)-7-(cyclopropylmethyl)-N-[(2S)-1-methoxypropan-2-yl]-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
5-{1-[(2-hydroxypyridin-4-yl)methyl]pyrrolidin-2-yl}-N-[2-(1H-pyrazol-1-yl)ethyl]thiophene-2-carboxamide
{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)[2-(piperidin-1-yl)ethyl]amine
1-{3-[4-(3-methoxybenzoyl)piperazin-1-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
2-{2-[5-(4-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1,3-benzoxazole
4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)-1-[(2,3-dimethoxyphenyl)methyl]piperidine
2-fluoro-5-{2-[2-(pyridin-2-yl)ethyl]piperidine-1-carbonyl}phenol
N-[(3R,4S)-1-[benzyl(methyl)sulfamoyl]-4-cyclopropylpyrrolidin-3-yl]acetamide
2-({4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-6-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)thieno[2,3-d]pyrimidin-4-amine
4-[3-(4-methoxyphenyl)propanoyl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
4-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-1-cyclohexyl-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
N4-(cyclohex-1-en-1-ylmethyl)-7-(piperidin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-[1-(cyclohexylmethyl)piperidin-3-yl]-1-ethyl-1H-pyrazole-4-sulfonamide
1-(2-methoxyphenyl)-4-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperazin-2-one
1-{2-[({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]morpholin-4-yl}ethan-1-one
S-[2-(2-cyclopropylacetyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-3-hydroxybutane-1-sulfonamido
4-(2-methylquinolin-6-yl)-1-[(2S)-piperidine-2-carbonyl]piperidin-4-ol
7-(propan-2-yl)-2-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
4-[3-(furan-2-yl)-3-phenylpropyl]-4H-1,2,4-triazole