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N-[3-(morpholin-4-yl)propyl]-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(2-chloropyridin-3-yl)methyl]-2-[(5-hydroxy-6-methyl-1,2,4-triazin-3-yl)sulfanyl]-N-methylacetamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(methylsulfanyl)propanamide
2-propyl-N-(pyridin-4-ylmethyl)-1,3-thiazole-4-carboxamide
2-({4-[3-(1H-pyrazol-3-yl)phenyl]phenyl}sulfanyl)acetamide
(1-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methanol
2-(1H-indazol-3-yl)-N-[3-(1H-pyrazol-1-yl)phenyl]acetamide
6-{[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]sulfonyl}-3-methyl-2,3-dihydro-1,3-benzoxazol-2-one
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1-phenylcyclopropyl)acetamide
methyl 4-(5-oxo-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepane-1-carbonyl)benzoate
1-methyl-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
2-butyl-N-[3-(pyridin-3-yl)propyl]-1,3-benzoxazole-5-carboxamide
2-[4-(2-{[(4-fluorophenyl)methyl]carbamoyl}ethyl)piperidin-1-yl]acetic acid
4-[1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl]thiomorpholine
1-{3-[2-(4-methoxypiperidin-1-yl)-2-oxoethyl]morpholin-4-yl}-2-(thiophen-2-yl)ethan-1-one
N-[(3-methyl-1H-pyrazol-5-yl)methyl]-4-[(2-methylprop-2-en-1-yl)oxy]benzamide
3-{2-[4-(6-ethylpyrimidin-4-yl)piperazin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-tert-butyl-2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-[2-(dimethylamino)-4-(4-hydroxypiperidin-1-yl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]-2-hydroxybutan-1-one
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-(thiophen-3-yl)acetamide
ethyl 4-(cyclopropylmethyl)-1-[(5-ethylthiophen-2-yl)sulfonyl]piperidine-4-carboxylate
3-(1H-pyrazol-1-yl)-1-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
4-{[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]amino}pyrimidine-5-carboxylic acid
4-[2-(propan-2-yloxy)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
4-{1-[3-(pyrrolidin-1-ylmethyl)phenyl]-1H-imidazol-2-yl}pyridine
5-[2-(pyridin-3-yl)-1H-imidazol-1-yl]pyridin-3-amine
1-methyl-3-(naphthalen-2-ylmethyl)-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(pyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)sulfonyl]-N-methylthiophene-2-carboxamide
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-(5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)piperazine
4-(3,3-difluoropiperidin-1-yl)-N,N,2-trimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
(1H-imidazol-4-ylmethyl)(methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
5-[2-oxo-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decane-8-carbonyl]pyridine-2-carbonitrile
N-({1-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
N-{1-[1-(2-hydroxypropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenoxypropanamide
N-[(1-ethyl-1H-indazol-3-yl)methyl]-4-(pyridin-2-yl)pyrimidin-2-amine
1-phenyl-4-[2-(pyrrolidin-1-yl)-6-(thiophen-3-yl)pyridine-3-carbonyl]piperazine
6-[(3-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-(1,3-thiazole-4-carbonyl)-1,4-diazepan-2-one
4-[2-oxo-4-(2-propoxybenzoyl)piperazin-1-yl]benzonitrile
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-{[(pyridin-4-ylmethyl)amino]methyl}piperidin-2-one
3-ethyl-N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N-methylpentanamide
N'-[2-(4-fluorophenyl)ethyl]-N'-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N,N-dimethylbutanediamide
2-(3-chloro-4-fluorophenyl)-2-[(1-methyl-3-propyl-1H-pyrazol-5-yl)formamido]acetic acid
N-benzyl-N-[(3-methylpyridin-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-N-[3-(1H-1,2,3-triazol-1-yl)propyl]piperidin-4-amine
3-cyclohexyl-N-methyl-N-{2-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}propanamide
N-(1,2-diphenylethyl)-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
2-(pyridin-4-yl)-N-(5,6,7,8-tetrahydronaphthalen-2-ylmethyl)pyrimidine-5-carboxamide
methyl 5-(6-ethylpyrimidin-4-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate