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1-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-methyl-3-(1H-1,2,4-triazol-1-yl)propan-1-one
4-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]butanoic acid
1-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
(1S,5R)-3-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-amino-N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-4-methylpyrimidine-5-carboxamide
(3S,4R)-1-{[2-(4-fluorophenyl)imidazo[1,2-a]pyridin-3-yl]methyl}-4-(hydroxymethyl)piperidin-3-ol
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-methyl-N-(2-methylprop-2-en-1-yl)acetamide
4-[2-(2,2-diphenylethyl)morpholine-4-carbonyl]pyridin-1-ium-1-olate
2-butyl-1-[5-(methoxymethyl)thiophene-2-carbonyl]-2,5-dihydro-1H-pyrrole
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-5-methoxyfuran-2-carboxamide
N-[(4-ethylphenyl)methyl]-N-methyl-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
1-[2-(1-methylpiperidin-2-yl)ethyl]-1,2-dihydroquinoxalin-2-one
1-methyl-3-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(3-methoxyphenyl)-3-[1-(thian-4-yl)piperidin-4-yl]propanamide
N-(2-hydroxyethyl)-3-[5-(oxan-4-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
methyl 8-[2-(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl)acetyl]-1-(2-methoxyethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
1-(4-{[4-(6-methylpyridine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-one
1-(2-methoxyethyl)-1-(1-methylpiperidin-4-yl)-3-[2-(propan-2-ylsulfanyl)phenyl]urea
(3S,4S)-4-propyl-1-{thieno[2,3-d]pyrimidin-4-yl}pyrrolidine-3-carboxylic acid
5-(azepane-1-carbonyl)-1-(butan-2-yl)-N-[3-(methylsulfanyl)propyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
2-(1-methylpyrrolidin-3-yl)-9-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-2,9-diazaspiro[5.5]undecan-3-one
1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
({3-[(3-fluorophenyl)methoxy]-4-methoxyphenyl}methyl)(methyl)(pyrazin-2-ylmethyl)amine
4-(pyridin-2-yl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}pyrimidin-2-amine
ethyl 5-(furan-2-ylmethyl)-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(3R,7S,8aS)-7-{[(4-methylphenyl)methyl]amino}-3-(2-methylpropyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
7-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}pyrazolo[1,5-a]pyridine
3-(but-2-yn-1-yl)-5-{1-[(2,5-dimethoxyphenyl)methyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
(2R,3R,6R)-3-(2-methoxyphenyl)-5-(pyridin-4-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(2,4-dimethoxyphenyl)methyl]-3-(1-methylpiperidin-3-yl)propanamide
1-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane
2-methyl-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-(3-chloro-1,2-oxazol-5-yl)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]propanamide
3-(5-{[2-(cyclopentyloxy)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl)pyridine
N4-cyclohexyl-N2-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]morpholine-2,4-dicarboxamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-6-(methoxymethyl)-N-methylpyrimidin-4-amine
[(4-{1-ethyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}-1,3-thiazol-2-yl)methyl]dimethylamine
N-methyl-2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carboxamide
4-{[5-(1-cyclohexyl-1H-1,2,3-triazol-4-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-propylpiperidine
2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-{spiro[indene-1,4'-piperidine]-1'-yl}ethan-1-one
[1-(5-chlorothiophene-2-carbonyl)-3-(3-methoxypropyl)piperidin-3-yl]methanol
N-(3-chloro-4-fluorophenyl)-3-[1-(2-oxo-2-phenylacetyl)piperidin-4-yl]propanamide
N-(1-benzothiophen-2-ylmethyl)-N-methyl-3-(pyrazin-2-yl)propanamide
1-[cyclohexyl(methyl)amino]-3-(2-methoxy-4-{[methyl(oxan-4-yl)amino]methyl}phenoxy)propan-2-ol
2-{4-[(4aS,8aR)-decahydroisoquinoline-2-carbonyl]piperidin-1-yl}-7-methanesulfonyl-4-methylquinazoline
[(3R,4R)-1-(4,6-dimethylpyrimidin-2-yl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
methyl 8-[(2,4-dimethoxy-3-methylphenyl)methyl]-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
3-cyclopropyl-N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-1H-pyrazole-5-carboxamide
1-[2-(3-methoxyphenyl)-1,3-benzoxazole-6-carbonyl]piperidin-3-ol
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}pyrrolidin-3-amine