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1-{2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}-2-(1H-1,3-benzodiazol-1-yl)propan-1-one
1-(2,6-difluoro-4-methoxybenzoyl)-3-propylpiperidine-3-carboxylic acid
3-(7-chloro-2-ethyl-3-methyl-1-benzofuran-5-yl)-1-methyl-1-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]urea
2-[4-(2,3-dihydro-1,4-benzodioxine-6-sulfonyl)morpholin-3-yl]-N-propylacetamide
N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
N-(2-hydroxyethyl)-N-methyl-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
5-({[6-(dimethylamino)pyrimidin-4-yl]amino}methyl)pyrrolidin-2-one
N-(1,2,3,4-tetrahydronaphthalen-2-yl)-3-(4H-1,2,4-triazol-4-yl)benzamide
3-fluoro-5-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]benzonitrile
(4aR,7aS)-1-acetyl-4-(2,3-dichlorobenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(propan-2-yl)-2-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl]-1,3-thiazole
methyl 1-[(3R,5S)-1-cyclopentyl-5-[4-(4-fluorophenyl)piperazine-1-carbonyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-(3-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidine-1-carbonyl}phenyl)pyrrolidin-2-one
2-{[2-(1H-pyrrol-1-yl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
4-methyl-1-({3-[4-(piperidin-1-yl)butoxy]phenyl}methyl)-1,4-diazepan-5-one
4-ethyl-3-{1-[1-(methoxymethyl)cyclobutanecarbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(2-chloro-6-fluorophenyl)ethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-(5-chloro-6-methyl-1-benzofuran-3-yl)-1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]ethan-1-one
8-[2-(2-chloro-6-fluorophenyl)acetyl]-1-methoxy-1,8-diazaspiro[4.5]decan-2-one
4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-(3-phenylprop-2-yn-1-yl)-N-propylbenzamide
2-(4-{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)ethan-1-ol
N-{3-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-3-oxopropyl}-N-methylmethanesulfonamide
3-[(3S,4R)-1-benzyl-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]-N-(3-methylphenyl)propanamide
(2S,4S)-1-{[4-(diethylamino)phenyl]methyl}-4-{[(2,5-difluorophenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
2-(3-{[benzyl(methyl)amino]methyl}phenyl)-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
3-{4-[2-(3-methylphenyl)acetamido]-1H-pyrazol-1-yl}-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}benzamide
1-(diethylamino)-3-(2-methoxy-4-{[(propan-2-yl)amino]methyl}phenoxy)propan-2-ol
2-(methylsulfanyl)-5-{[3-(pyrrolidin-1-yl)piperidin-1-yl]methyl}pyrimidine
2-[1-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
2-(2-methylpropyl)-6-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
5-benzyl-5-[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]-3-[2-(pyrrolidin-1-yl)ethyl]imidazolidine-2,4-dione
(2S,4S)-4-amino-1-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetyl}pyrrolidine-2-carboxylic acid
N-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-N-[(2E)-3-phenylprop-2-en-1-yl]cyclopropanamine
4-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1-cyclopropylpyrrolidin-2-one
(2S)-2-({1-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]piperidin-4-yl}amino)-3-phenylpropan-1-ol
9-(6-methylpyrimidin-4-yl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
(4aR,8aR)-7-(6-cyanopyridine-3-carbonyl)-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
4-benzyl-3-ethyl-1-[4-(methylamino)benzoyl]-1,4-diazepan-5-one
1-(2-benzylmorpholin-4-yl)-2-(pyridin-2-ylsulfanyl)ethan-1-one
2-(4-fluoro-3-methylphenyl)-1-[3-(3-methoxypropyl)piperidin-1-yl]ethan-1-one
N-[4-(difluoromethoxy)phenyl]-4-(pyridin-3-ylmethoxy)piperidine-1-carboxamide
6-chloro-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]imidazo[1,2-a]pyridine-2-carboxamide
(3aR,6aR)-2-(2-hydroxyethyl)-5-(5-phenyl-1,2-oxazole-3-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-3-methyl-1-[4-(thiophen-2-ylmethoxy)phenyl]urea
(3aR,6aR)-2-(3-aminopropanoyl)-5-cyclopropanecarbonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-1-[4-(thiophen-2-ylmethoxy)phenyl]urea
1-(furan-3-carbonyl)-4-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}-1,4-diazepane
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-2-phenylacetamide
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(4-methyl-1H-pyrazol-1-yl)propanamide
3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-5-propyl-1,2,4-oxadiazole