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(2S,4S)-1-[(2-chlorophenyl)methyl]-4-{[(2,4-difluorophenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
[(2S)-1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-yl]methanol
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperidin-3-ol
1-methyl-3-(pyrrolidine-1-carbonyl)-N-[2-(thiophen-2-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3R,4S)-1-[5-(morpholine-4-carbonyl)pyridin-2-yl]-4-(propan-2-yl)pyrrolidin-3-amine
N-benzyl-2-[(isoquinolin-5-yloxy)methyl]-N-methyl-1,3-oxazole-4-carboxamide
5-methyl-N-(2-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)thiophene-2-carboxamide
(2R,6S)-2,6-dimethyl-4-{1-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-4-yl}morpholine
{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}[(trimethylpyrazin-2-yl)methyl]amine
N-[2-(7-{[4-(propan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]furan-2-carboxamide
(2S,4S)-4-(4-{2-[(dimethylamino)methyl]phenoxymethyl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
3-[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]phenol
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[1-(thiophen-2-yl)ethyl]benzamide
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-2H-1,3-benzodioxole-5-carboxamide
N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-4,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[(2,5-dichlorophenyl)methyl]-4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
(1R,5S,8S)-3-[(5-chloro-2,4-dimethoxyphenyl)methyl]-N,N-dimethyl-3-azabicyclo[3.2.1]octan-8-amine
3-{2-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]propanamide
2-methyl-2-[5-(6-methyl-2H-1,3-benzodioxol-5-yl)-4-phenyl-1H-imidazol-1-yl]propane-1,3-diol
N-(cyclobutylmethyl)-1-methyl-N-(oxolan-2-ylmethyl)-5-phenyl-1H-pyrrole-2-carboxamide
N-methyl-5-{[(1S,5R)-7-oxo-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}furan-2-carboxamide
N-{[4-(1H-imidazol-1-yl)phenyl]methyl}-1-methyl-N-(pyridin-4-ylmethyl)piperidin-4-amine
1-(1H-indole-2-carbonyl)-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
N-[1-(3,5-difluorophenyl)ethyl]-4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzamide
(3S,5R)-N3-cyclopentyl-N5-(2,3-dihydro-1H-inden-5-yl)piperidine-3,5-dicarboxamide
N-(2-fluoroethyl)-3-{[3-(1H-1,2,4-triazol-1-yl)propyl]sulfamoyl}benzamide
2-(benzylsulfanyl)-5-{[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl}pyrimidine
5-{1-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,3-triazol-4-yl}pyrimidine
1-[3-(5-methylfuran-2-yl)butyl]-4-(1H-pyrazol-3-yl)piperidine
3-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-N-(propan-2-yl)propanamide
N-[2-(3-chlorophenyl)ethyl]-2-({1-oxaspiro[4.4]nonan-3-yl}amino)acetamide
1-[(4-fluorophenyl)methyl]-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-2-carboxamide
1-(2-{[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}pyrimidin-4-yl)piperidin-3-ol
4-(2-ethylphenyl)-5-(furan-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
4-[(2-{1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]piperidin-3-yl}-1H-imidazol-1-yl)methyl]pyridine
2-methoxy-1-[3-(2-phenylethyl)piperidin-1-yl]ethan-1-one
N-[(1-ethylpiperidin-3-yl)methyl]-3-methanesulfonylbenzamide
4-methyl-1-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pentane-1,2-dione
3-[4-(5-methylpyrimidin-2-yl)phenyl]aniline
2-{1-cyclopentyl-4-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]piperazin-2-yl}ethan-1-ol
1-methyl-N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1H-pyrazole-3-carboxamide
N-{2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-4-(1H-1,2,4-triazol-1-yl)butanamide
N-[2-(pyridin-2-yl)ethyl]-2-[4-(pyrimidin-2-yl)-2-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)phenoxy]acetamide
1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-8-(1-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-amino-1-(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
(3R,4R)-4-cyclobutyl-1-(4-fluoro-2-methylbenzoyl)-3-methylpiperidin-4-ol
2-[4-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-1-yl]-N-methylacetamide
2-methyl-4-(naphthalen-1-yl)-1H-imidazole
4-[4-(5-chloro-2-methylphenyl)piperazin-1-yl]-6-(methoxymethyl)pyrimidine