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6-methyl-5-{5-[2-(methylsulfanyl)phenyl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-[(4-chlorophenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
4-[4-(1H-indazole-3-carbonyl)piperazin-1-yl]quinazoline
1-({[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)propan-2-ol
(1R,5R)-6-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N5-(3-methoxypropyl)-N6-[3-(methylsulfanyl)propyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-(2-fluorophenyl)-N-[2-(furan-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]acetamide
8-[2-(methylamino)pyridine-4-carbonyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1-(propan-2-yl)piperidine-4-carboxamide
2-{7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}acetamide
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-2-(2-oxopyrrolidin-1-yl)propanamide
3,3-diphenyl-1-(piperidine-1-sulfonyl)piperidine
2-[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]acetic acid
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzamide
1-{[3-({1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}-4-(pyridin-3-ylmethyl)piperazine
4-(5-methoxy-1H-indazole-3-carbonyl)-1,4-oxazepan-6-ol
1-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}-3-(3,5-dimethyl-1H-pyrazol-1-yl)propan-1-one
{[5-(methoxymethyl)furan-2-yl]methyl}({[2-(piperidin-1-yl)-2,3-dihydro-1H-inden-2-yl]methyl})amine
ethyl 1-(5,8-dimethoxy-3-{[(2-methylpropyl)amino]methyl}quinolin-2-yl)piperidine-4-carboxylate
2-(cyclohex-1-en-1-yl)-1-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
3-{[(dicyclopropylmethyl)(methyl)amino]methyl}-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
1-(2-{methyl[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]amino}ethyl)piperidin-2-one
N-(adamantan-1-ylmethyl)-N-methyl-3-(pyrazin-2-yl)propanamide
N-cyclopropyl-N-{[2-(4-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}cyclobutanecarboxamide
2-(2,4-dimethylphenyl)-2-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]acetic acid
2,3-dimethyl-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)-1H-indole-7-carboxamide
4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-2-(morpholin-4-ylmethyl)-1,4-oxazepane
N,1-dimethyl-N-(1,2-oxazol-5-ylmethyl)-1H-1,2,3-benzotriazole-5-carboxamide
1-cyclopentyl-4-{[3-hydroxy-2-oxo-1-(2-phenylethyl)piperidin-3-yl]methyl}piperazin-2-one
4,4,4-trifluoro-1-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]butan-1-one
1-{5H,6H-benzo[h]quinazolin-2-yl}-N-(cyclopropylmethyl)-5-methyl-N-propyl-1H-pyrazole-4-carboxamide
5-(methoxymethyl)-N-[3-methyl-1-(7-{[4-(propan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)butyl]furan-2-carboxamide
N-(1-{2-[4-(2-methoxybenzoyl)piperazin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2-phenoxyacetamide
6-{4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]piperazin-1-yl}pyridine-3-carboxamide
3-{1-[2-(2-hydroxyethoxy)ethyl]piperidin-3-yl}benzoic acid
(1-benzothiophen-2-ylmethyl)[(4-{[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]methylamine
4-{1-[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
2-ethyl-4-methyl-N-{2-[3-(trifluoromethyl)phenyl]ethyl}-1,3-oxazole-5-carboxamide
4-phenyl-3-(piperidin-4-yl)-1-[2-(1H-pyrrol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(azepan-1-yl)-2-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
2-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]-3,5,7-trimethyl-1H-indole
N-[2-(cyclohex-1-en-1-yl)ethyl]-N-{[2-(4-hydroxypiperidin-1-yl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-1,3-thiazole-5-carboxamide
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-methyl-2-(1H-pyrazol-1-yl)butanamide
2-[5-(2-amino-4-methyl-1,3-thiazol-5-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]acetic acid
methyl (1R,3S,3aR,6aS)-3-(3,5-dichloro-4-methylphenyl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
3-methyl-1-{1-[6-(4-methylpiperazin-1-yl)pyridine-3-carbonyl]piperidin-3-yl}butan-1-one
5,7-dimethyl-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
{[4-(butan-2-yloxy)-3-chlorophenyl]methyl}[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
N-butyl-N-methyl-3-({methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide