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3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-(propan-2-yl)propanamide
4-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}-1λ6-thiomorpholine-1,1-dione
N-[(1-benzylpiperidin-3-yl)methyl]quinoline-8-sulfonamide
2-{4-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-1-(3-methylbut-2-en-1-yl)piperazin-2-yl}ethan-1-ol
1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3-carbonitrile
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]acetamide
1-(propan-2-yl)-2-{[4-(thian-4-yl)piperazin-1-yl]methyl}-1H-1,3-benzodiazole
2-(azepan-1-yl)-N-[2-(dimethylsulfamoyl)ethyl]-2-oxoacetamide
4-hydroxy-4-(1H-imidazol-1-ylmethyl)-N-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)piperidine-1-carboxamide
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
(2S,4R)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]-N,N-dimethyl-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
N-[(3-methoxyphenyl)methyl]-1-(4,6,7-trimethylquinazolin-2-yl)piperidine-4-carboxamide
8-[2-(thiophen-3-yl)acetyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-methoxy-2-[(5-propyl-1,2-oxazol-3-yl)formamido]propanoic acid
7-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
methyl N-[2-oxo-4-(2,4,5-trimethoxyphenyl)-1,2,3,4-tetrahydroquinolin-7-yl]carbamate
3-ethoxy-N-methyl-N-(quinolin-5-ylmethyl)propanamide
3-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propan-1-ol
N-(1-{[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}piperidin-4-yl)methanesulfonamide
N-[(8-{[3-(benzyloxy)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]furan-2-carboxamide
4-(4-chlorophenyl)-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]butan-1-one
N-(1-{1-[(4-methoxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N,1,3-trimethyl-1H-pyrazole-5-carboxamide
2-[3-(benzyloxy)piperidin-1-yl]pyrimidine
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(5-fluoropyrimidin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidine
1-(cyclopropylmethyl)-4-[4-(pyridin-2-ylmethoxy)phenyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-{2-[2-(4-fluorophenyl)piperidin-1-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
(1S,5R)-3-cyclobutanecarbonyl-6-(1H-indole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-(4-{2-[(3S,4R)-4-amino-3-methoxypiperidin-1-yl]-2-oxoethyl}phenyl)imidazolidin-2-one
N-[2-(4-methoxyphenyl)ethyl]-1-methyl-N-[(1-methylpiperidin-4-yl)methyl]-1H-pyrrole-2-carboxamide
1-(propane-1-sulfonyl)-N-{thieno[2,3-d]pyrimidin-4-yl}azepan-3-amine
3,4-dimethoxy-N-{[7-methoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)benzamide
N-[2-(methylsulfanyl)phenyl]-3-(3-methylthiophene-2-carbonyl)piperidine-1-carboxamide
2-{2-[4-(furan-2-yl)phenyl]-1H-imidazol-1-yl}-N,N-dimethylethane-1-sulfonamide
2-[4-(pyridin-2-yl)-2-[(3,3,4-trimethylpiperazin-1-yl)methyl]phenoxy]acetic acid
8-(2-methoxy-6-methylbenzoyl)-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(2-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-oxoethyl)imidazolidine-2,4-dione
1-(6,7-dimethoxy-4-methylquinolin-2-yl)azetidin-3-ol
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N,2-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
N-(2-{7-[(2-fluoro-5-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxolane-2-carboxamide
N4-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)pyrimidine-2,4-diamine
4-(3-ethoxy-5-fluorophenyl)-N-methylbenzamide
(cyclopentylmethyl)({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
2-{3-[2-(3-methoxyphenyl)ethyl]piperidine-1-carbonyl}-5-methylphenol
1-{[1-propyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-5-(trifluoromethyl)-1,2-dihydropyridin-2-one
1-cyclopropyl-N-[2-(dimethylamino)ethyl]-N-[(2-methylphenyl)methyl]-5-oxopyrrolidine-3-carboxamide
1-[(2-fluorophenyl)methyl]-6-oxo-N-[2-(pyridin-3-yloxy)ethyl]piperidine-3-carboxamide
2-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-5-methylphenol
N-(oxolan-3-yl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide