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diethyl({2-[5-(1-ethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl})amine
1-{2-[1-(5-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-5-methyl-1,3-oxazole-4-carboxamide
N-(4-{[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenyl)acetamide
9-methoxy-7-(6-methoxypyridazin-3-yl)-4-(naphthalene-1-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-ethyl-N-[1-(pyrimidin-2-yl)piperidin-3-yl]-1H-indole-2-carboxamide
{1-[(2,5-dimethyl-1H-indol-3-yl)methyl]-4-[(4-methoxyphenyl)methyl]piperidin-4-yl}methanol
2-{[1-(4-methoxyphenyl)cyclopentyl]formamido}-N,N-dimethylpropanamide
N-{[2-(4-acetylpiperazin-1-yl)-6-methylquinolin-3-yl]methyl}-N-[2-(cyclohex-1-en-1-yl)ethyl]-2,3-dimethoxybenzamide
8-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(4-{[4-(difluoromethoxy)phenyl]methyl}-1-[(4-fluorophenyl)methyl]piperazin-2-yl)ethan-1-ol
2-(2-{[2-(2-chlorophenyl)-2-hydroxyethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
(3R,4R)-1-(4-amino-5-methylpyrimidin-2-yl)-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]piperidin-3-amine
methyl (2S)-2-cyclopropyl-2-[({[4-(N-methylacetamido)phenyl]carbamoyl}methyl)amino]acetate
N-(3,3-dimethyl-2-oxobutyl)-2-(methylamino)pyrimidine-5-carboxamide
6-(dimethylamino)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
6-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]pyridine-2-carbonitrile
3-{[1-ethyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1-methyl-1H-indole
1-(4-ethylpiperazin-1-yl)-3-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)propan-1-one
2-[(3S,4R)-3-acetamido-4-(propan-2-yl)pyrrolidin-1-yl]-N-[(2-methylphenyl)methyl]acetamide
1-benzyl-N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-1H-pyrazole-4-carboxamide
2-(5-acetylthiophen-3-yl)-1-[4-(pyridin-3-ylmethyl)piperazin-1-yl]ethan-1-one
2-ethyl-8-(9H-purin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
5-{[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]methyl}-2-methoxybenzoic acid
(2S,4R)-4-{[(4-chlorophenyl)methyl]amino}-N-(2-methoxyethyl)-1-(propan-2-yl)pyrrolidine-2-carboxamide
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-hydroxy-4-methylbenzamide
3-[3-(furan-2-yl)benzoyl]-9-methoxy-10-(thiomorpholine-4-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
7-methyl-2-({2-oxo-3-oxatricyclo[7.3.1.05,13]trideca-1(12),5(13),6,8,10-pentaen-8-yl}methyl)-2,7-diazaspiro[4.5]decan-6-one
[(8-methoxyquinolin-2-yl)methyl](methyl)[1-(pyrimidin-4-yl)ethyl]amine
{[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl}[1-(pyrazin-2-yl)propan-2-yl]amine
8-(butan-2-yl)-3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(2-methylpropyl)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1,2-oxazole-5-carboxamide
3-(2-amino-1,3-thiazol-4-yl)-1-[4-(pyridin-4-yl)piperazin-1-yl]propan-1-one
({5-[1-(5-chloropyridine-3-carbonyl)piperidin-4-yl]-4-ethyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
(4aS,7aR)-1-[2-(6-methylpyridin-2-yl)ethyl]-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-methyl-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-5-[1-(thiophen-3-ylmethyl)-1H-pyrazol-3-yl]-1,3-thiazol-2-amine
1-(furan-2-ylmethyl)-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}piperidine-4-carboxamide
3-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-[2-methyl-3-(pyrrolidine-1-carbonyl)phenyl]urea
1-[(4-methyloxan-4-yl)methyl]-4-(pyridin-3-ylmethyl)piperazine
1-(4-{[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one
6-oxo-N-{[4-(piperidine-1-carbonyl)phenyl]methyl}piperazine-2-carboxamide
5-(4-chloro-2-methoxyphenoxymethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-2-(2-methoxyphenoxy)acetamide
N,2,5-trimethyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
5-[3-(morpholine-4-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-1,3-benzodiazole
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
5-{[1-benzyl-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}quinoxaline
N-[2-(4-{[methyl(naphthalen-1-ylmethyl)amino]methyl}phenoxy)ethyl]-1,3-thiazole-5-carboxamide
4-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-1-[(4-methylphenyl)methyl]piperazin-2-one