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4-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-4-yl}pyridine
2-[(1S,5R)-6-[(2,4-dichlorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
5-({2-[2-(thiophen-2-yl)ethyl]piperidin-1-yl}sulfonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
(2R)-2-amino-3-(4-chlorophenyl)-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
5-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}-1-(3-phenylpropyl)piperidin-2-one
2-chloro-4-({6-[(dimethylamino)methyl]-1,4-oxazepan-4-yl}methyl)phenol
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[3-(thiophen-3-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]-3-(pyridin-2-yl)propan-1-one
ethyl 1-[(4-methoxyphenyl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
4-[(2-fluoro-3-methylphenyl)methyl]-9-(2-methoxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-1,3-thiazole-4-carboxamide
N-[4-(3-methoxyphenyl)phenyl]-1-(1,3-thiazol-2-ylmethyl)piperidine-3-carboxamide
5-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1-propyl-1H-pyrazole-4-carboxamide
3-methyl-4-({3-[4-(piperidin-1-yl)butoxy]phenyl}methyl)piperazin-2-one
4,6-dimethyl-1-{2-[(1-phenoxypropan-2-yl)amino]ethyl}-1,2-dihydropyrimidin-2-one
N-[3-(4-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]ethane-1-sulfonamide
[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amine
2-methanesulfonyl-N-(oxolan-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
5-{4-[(8-chloro-4-hydroxyquinolin-2-yl)methyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
N-methyl-2-(2-methylpropanoyl)-N-(1,3-thiazol-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
3-(2H-1,3-benzodioxol-5-yl)-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
2-{4-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]-1H-pyrazol-1-yl}-N-(1-ethyl-1H-1,2,3-triazol-4-yl)acetamide
[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl](methyl){[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N,N-diethyl-2-{[4-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-2-oxo-1-(2-phenylethyl)-1,4-diazepan-6-yl]oxy}acetamide
4-(4-chlorophenyl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]butanamide
5-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-N,N-dimethylazepan-4-amine
N,N-dimethyl-5-{[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]methyl}pyridin-2-amine
3-[4-(2,5-difluorophenyl)-1H-pyrazol-5-yl]-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidine
5-oxo-1-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidine-3-carboxylic acid
2-(dimethylamino)-N-(2-ethyl-1,3-dihydroxypropan-2-yl)-2-(4-methylphenyl)acetamide
5-(2-chlorophenyl)-N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]furan-2-carboxamide
(2S,4S)-4-[4-(cyclohexylmethyl)-1H-1,2,3-triazol-1-yl]-N-ethylpyrrolidine-2-carboxamide
2-[(2,6-dimethoxypyridin-3-yl)formamido]-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetic acid
4-ethyl-3-{1-[2-(pyridin-2-yl)pyrimidine-5-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
[(2S)-1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]pyrrolidin-2-yl]methanol
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-N-methyl-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
2-[2-(3-carboxypiperidin-1-yl)pyrimidin-4-yl]pyridine-4-carboxylic acid
10-methoxy-5-{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
N-{2-[4-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}furan-2-carboxamide
N,1-diethyl-N-[1-(4-methoxyphenyl)propyl]-3-methyl-1H-pyrazole-4-carboxamide
6-[({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)amino]pyrazine-2-carboxamide
1-(carbamoylmethyl)-N-[(1-ethyl-1H-indazol-3-yl)methyl]piperidine-3-carboxamide
1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-4-methyl-1,2,3,6-tetrahydropyridine
5-(4-fluoro-2-methylphenyl)-1-(1H-imidazol-2-ylmethyl)-4-phenyl-1H-imidazole
N-(1-benzothiophen-5-ylmethyl)-3-(1-methyl-1H-pyrazol-4-yl)propanamide
7-acetamido-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
5-{[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]methyl}-2-(pyrrolidin-1-yl)pyrimidine