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(1S,6R)-9-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3,9-diazabicyclo[4.2.1]nonan-4-one
4-{3-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]pyridin-2-yl}morpholine
methyl 3-(3-carbamoylpropyl)-1-cyclohexyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylate
2-{4-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-1H-pyrazol-1-yl}-N-(1-methyl-1H-1,2,3-triazol-4-yl)acetamide
3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}propanamide
(3aR,6aR)-2-(2-hydroxyethyl)-5-(1-phenylcyclohexanecarbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-ethyl-2,3-dimethyl-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-[(3,4-dimethoxyphenyl)methyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1,3-benzoxazole-6-carboxamide
1-[2-methoxy-4-({[(2-methoxyphenyl)methyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
ethyl 4-(2-phenoxyethyl)-1-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carbonyl]piperidine-4-carboxylate
(1S,5R)-6-methyl-3-{4-[(pyridin-2-ylsulfanyl)methyl]benzoyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
2-methyl-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-2-(thiophen-2-ylformamido)propanamide
2-(2H-1,3-benzodioxol-5-yl)-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
N-[(5-ethylpyridin-2-yl)methyl]-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
2-chloro-N-propyl-4-({[2-(1,3-thiazol-4-yl)ethyl]carbamoyl}amino)benzamide
N-({8-[(4-methoxy-3-methylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)furan-2-carboxamide
(1R,5S)-6-[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-6-azabicyclo[3.2.1]octane
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-(4-methoxy-3-methylbenzoyl)piperidin-3-ol
1-cycloheptyl-N-[2-(naphthalen-2-yl)ethyl]-6-oxopiperidine-3-carboxamide
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N,1,3-trimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1-benzothiophene-2-carboxamide
(1S,3R)-N1-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-1,2,N2,N3,3-pentamethylcyclopentane-1,3-dicarboxamide
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-(1-methyl-1H-pyrazole-4-carbonyl)piperidin-4-ol
2-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-5-methoxy-4H-pyran-4-one
N-[(2-fluorophenyl)methyl]-1-methyl-5-[(pyridin-4-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]propanamide
4-hydroxy-2-methyl-N-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]pyrimidine-5-carboxamide
2-methoxy-4-[4-(pyrrolidine-1-carbonyl)phenyl]phenol
1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-3,3-diphenylpiperidine
1-(2,2-dimethylpropyl)-3-hydroxy-3-({[(3-methyl-1H-pyrazol-5-yl)methyl]amino}methyl)piperidin-2-one
2-({3-[(6,7-dimethoxy-4-methylquinolin-2-yl)amino]propyl}(2-hydroxyethyl)amino)ethan-1-ol
N-[(2-fluorophenyl)methyl]-2-{methyl[1-(pyridin-3-yl)propyl]amino}acetamide
(3S,5R)-5-[(4-fluorophenyl)carbamoyl]-1-(2-methylpropyl)piperidine-3-carboxylic acid
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl){[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}amine
1-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
(3R)-1-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)pyrrolidin-3-ol
(2S,4R)-4-amino-N-methyl-1-(9-methyl-9H-carbazole-3-carbonyl)pyrrolidine-2-carboxamide
1-(3-methylfuran-2-carbonyl)-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine
1-(2,8-dimethylquinoline-4-carbonyl)-4-phenylpiperidine-4-carbonitrile
6-(2-{[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)pyrimidin-4-ol
2-phenyl-1-(1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperidin-4-yl)ethan-1-ol
N,4-dimethyl-N-(1,2-oxazol-5-ylmethyl)-3-(2-oxoimidazolidin-1-yl)benzamide
1-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
(2S)-2-[4-(3-cyanophenyl)-1H-1,2,3-triazol-1-yl]-4-(methylsulfanyl)butanoic acid
3-[2-(2-methoxyethyl)morpholin-4-yl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraene
[1-(3-chloro-4-methoxybenzoyl)-3-(cyclopropylmethyl)piperidin-3-yl]methanol
(1S,5R)-6-(4-chlorobenzenesulfonyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-2-(pyridin-2-ylsulfanyl)acetamide
ethyl 4-({4-[(1R,2R)-2-phenylcyclopropanecarbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazine-1-carboxylate