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9-[(2-fluoro-5-methoxyphenyl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(4-chlorophenyl)methyl]-N-{2-[2-(trifluoromethyl)phenyl]ethyl}-1H-1,2,3-triazole-4-carboxamide
4-[4-(furan-2-ylmethyl)piperazin-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
1-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-5-oxopyrrolidine-3-carboxylic acid
2-{[(3R,4S)-1-(1-acetylpiperidin-4-yl)-4-propylpyrrolidin-3-yl]amino}pyridine-3-carbonitrile
5-tert-butyl-4-{[(1,1-dioxo-1λ6-thiolan-3-yl)(ethyl)amino]methyl}furan-2-carboxamide
9-methoxy-7-(2-methoxyphenyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(3R)-1-{[2-(4-chlorophenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}pyrrolidin-3-ol
3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]-5-{1-[(4-methoxyphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
5-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
(3S,4S)-1-(1H-1,3-benzodiazole-2-carbonyl)-4-(3-methoxyphenyl)piperidin-3-ol
1-benzyl-5-{[(1-hydroxycyclohexyl)methyl]amino}-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-phenylpiperidine-4-carbonitrile
methyl (1R,3S,3aR,6aS)-3-(3-fluoro-2-hydroxyphenyl)-1-(1H-imidazol-4-ylmethyl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
1-({[5-(oxolan-2-yl)-1,3,4-thiadiazol-2-yl]carbamoyl}methyl)piperidine-4-carboxamide
N-cyclohexyl-3,5-dimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-indole-2-carboxamide
N-{4-[4-(4-methoxybutyl)piperazine-1-carbonyl]phenyl}pentanamide
1-(2-oxo-2-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}ethyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N,6-dimethyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-N-[1-(1,3-thiazol-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
5-(4-chlorophenyl)-3-[4-(3-chlorophenyl)piperazin-1-yl]-1,2,4-triazine
5-(1-benzofuran-2-yl)-3-{2-[2-(pyridin-2-yl)ethyl]piperidin-1-yl}-1,2,4-triazine
1-ethyl-3-(4-methylpiperazine-1-carbonyl)-N-{[4-(trifluoromethyl)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[4-(morpholine-4-carbonyl)phenyl]-N-{2-[4-(trifluoromethyl)phenyl]ethyl}piperidin-4-amine
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-1H-pyrrole-2-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine
N-[4-(3-methylphenyl)phenyl]-1-(pyrazine-2-carbonyl)piperidine-4-carboxamide
1-[3-methoxy-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]urea
1-benzyl-4-(furan-3-ylmethyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
6-oxo-7-(propan-2-yl)-N-[2-(thiophen-2-yl)ethyl]-2,7-diazaspiro[4.5]decane-2-carboxamide
1-ethyl-8-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-cyclopropyl-6-ethyl-N-[(2-methoxyphenyl)methyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
3-(morpholine-4-carbonyl)-N-(3-phenylpropyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{2-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]-2-oxoethyl}piperidin-2-one
{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl){[5-(pyrimidin-2-ylsulfanyl)furan-2-yl]methyl}amine
N-({1-[(4-fluoro-3-methylphenyl)methyl]piperidin-3-yl}methyl)oxane-4-carboxamide
(1R,5S)-6-[2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carbonyl]-6-azabicyclo[3.2.1]octane
2-(3-cyclopropyl-5-{[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]methyl}-1H-1,2,4-triazol-1-yl)-3-methylpyridine
(3R,5S)-5-(morpholine-4-carbonyl)-N-(quinolin-2-ylmethyl)piperidine-3-carboxamide
3-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-[2-(oxolan-2-ylmethoxy)phenyl]urea
2-(3-acetyl-1H-pyrazol-1-yl)-N-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)acetamide
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-2-(morpholin-4-yl)butanamide
3-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-5-(piperidin-4-yl)-5-propylimidazolidine-2,4-dione
ethyl 1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-4-(2-phenylethyl)piperidine-4-carboxylate
N-{[2-(4-benzylmorpholin-2-yl)-6-oxo-1,6-dihydropyrimidin-4-yl]methyl}acetamide
8-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-(cyclopropylmethyl)-9-[(4-methyl-1H-imidazol-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-butyl-4-[2-(1,4-oxazepan-4-yl)-2-oxo-1-phenylethyl]piperazine-2,3-dione
2-acetamido-N-{[5-methyl-7-(2-methylquinolin-6-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide