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3-(1-methyl-1H-pyrazol-4-yl)-1-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propan-1-one
1-[9-methoxy-7-(6-methoxypyridazin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-phenylethan-1-one
7-cyclohexyl-2-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
3-(4-fluorophenyl)-3-{[1-(propan-2-yl)piperidin-4-yl]formamido}propanoic acid
2-methyl-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-1,3-thiazole-4-carboxamide
1-[1-(6-methylpyridazin-3-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
9-(pyrimidin-2-yl)-3,9-diazaspiro[5.5]undecane-2,4-dione
N,4-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,3-oxazole-5-carboxamide
6-(2-fluoro-4-methoxyphenyl)-7-methyl-8-oxo-N-(2-oxopiperidin-3-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3,4-dimethoxy-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)benzene-1-sulfonamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl]methanol
(2S,4S)-4-amino-N,N-diethyl-1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidine-2-carboxamide
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]methanesulfonamide
N-[(5-methyl-2-{3-[3-(pyridin-3-yl)propanamido]phenyl}-1,3-oxazol-4-yl)methyl]-5-propyl-1,2-oxazole-3-carboxamide
N-{2-[4-({[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl](methyl)amino}methyl)-5-methyl-1,3-oxazol-2-yl]phenyl}methanesulfonamide
(2,1,3-benzothiadiazol-5-ylmethyl)({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-1-(pyridin-2-yl)piperidine-3-carboxamide
N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-1-(propan-2-yl)piperidine-3-carboxamide
N-[(1S,2R)-2-(cycloheptylamino)cyclobutyl]-5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carboxamide
{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}(methyl)(2-phenoxyethyl)amine
methyl (2S,4S)-4-(2-fluorobenzamido)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]pyrrolidine-2-carboxylate
N4-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(methylsulfanyl)pyrimidine-4,6-diamine
N-cyclopentyl-6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-(3-chloro-1H-1,2,4-triazol-5-yl)-N-methyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}propanamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]-2-methoxypyridine-3-carbonitrile
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
1-(cyclopent-1-ene-1-carbonyl)-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-N,N-bis(prop-2-en-1-yl)-1,2-oxazole-3-carboxamide
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-[2-(propylsulfanyl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(2-chlorophenyl)ethyl]-3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzamide
8-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
methyl 3-[(3,3-dimethylbutanamido)methyl]-5-[2-(thiophen-3-yl)acetamido]benzoate
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-(thiolan-3-yl)pyridin-2-amine
methyl 1-(2-methoxyethoxy)-8-[3-(methylsulfanyl)propyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
2-(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridine-3-carboxamide
3-{[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-N-methyl-1,2,4-oxadiazole-5-carboxamide
(2R,6R)-4-({7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-triene-6-carboxylic acid
N3-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]piperidine-1,3-dicarboxamide
1-{[2-(5-methylfuran-2-yl)phenyl]methyl}-4-(thian-4-yl)piperazine
(4aS,7aR)-1-[(2,3-dimethoxyphenyl)methyl]-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-[(6-methylpyridin-2-yl)methyl]piperidine-3-carboxamide
(3aS,7aR)-2-[4-(4-methoxyphenyl)-4-oxobutanoyl]-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
2-(azepan-1-ylmethyl)-4-(7-chloroquinolin-4-yl)phenol
[2-({4-[(4-ethynylphenyl)methyl]piperazin-1-yl}methyl)phenyl]methanol
4-(2,3-dichlorophenyl)-1-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,3-triazole
2-[4-(1-benzothiophen-3-yl)-2-(morpholin-4-ylmethyl)phenoxy]-N-(cyclopropylmethyl)-N-propylacetamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2-(5-fluoro-2-methyl-1H-indol-3-yl)acetamide
2-[3-(1H-pyrazol-5-yl)phenyl]-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]acetic acid
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-(1,2-oxazole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one