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N-benzyl-4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-methylbenzamide
3-(3-methoxyphenyl)-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazole-4-carboxamide
1-{[4-(propan-2-yl)phenyl]methyl}-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
4-(benzylamino)-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]butanamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-1-cyclohexyl-1H-1,2,3-triazole-4-carboxamide
2-(2,5-dimethylphenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
5,6-dimethyl-3-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl}-1,2-dihydropyridin-2-one
4-(1H-pyrazol-1-yl)-1-(thiophene-2-sulfonyl)piperidine-4-carboxylic acid
methyl (2S,4S,5R)-1,2-dimethyl-5-(2-methylphenyl)-4-{[2-(methylsulfanyl)ethyl]carbamoyl}pyrrolidine-2-carboxylate
N-cyclopropyl-N-({2-[methyl(thiophen-3-ylmethyl)amino]-7-(methylsulfanyl)quinolin-3-yl}methyl)-2H-1,3-benzodioxole-5-carboxamide
(3R,4S)-4-(4-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-1-yl)oxolan-3-ol
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(3-methylfuran-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(2-{1-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
2-[(3-methoxyphenyl)methyl]-4-(piperidine-1-sulfonyl)morpholine
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-cyclopropanecarbonyl-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-[2-(1H-indol-3-yl)ethyl]acetamide
3-{1-[3-(2-hydroxyphenyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}benzoic acid
N-(4-chlorophenyl)-3-[1-(quinoline-6-carbonyl)piperidin-3-yl]propanamide
2-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
(3S,5R,9R)-5-hydroxy-11-(2-methoxybenzoyl)-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
(2S,4S)-N-ethyl-4-{2-[4-(hydroxymethyl)phenyl]acetamido}-1-(3-methylbut-2-en-1-yl)pyrrolidine-2-carboxamide
4-benzyl-3-{2-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-2-oxoethyl}piperazin-2-one
9-[(2Z)-5-methyl-2-phenylhex-2-en-1-yl]-1,4,9-triazaspiro[5.5]undecan-5-one
4-(hydroxymethyl)-1-[(1-methyl-1H-indol-2-yl)methyl]azepan-4-ol
1-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-4-(2-methylphenyl)-1,4-diazepane
N-(2-methylphenyl)-3-[(3S,4R)-1-(pyridin-3-ylmethyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanamide
4-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-2-methoxypyridine-3-carbonitrile
1-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)phenyl]imidazolidine-2,4-dione
4-(5-{[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]methyl}pyrimidin-2-yl)morpholine
(2S,4S,5R)-5-(2,3-difluorophenyl)-1-methyl-4-(morpholine-4-carbonyl)pyrrolidine-2-carboxylic acid
1-[6-methyl-3-({methyl[2-(pyrrolidin-1-yl)ethyl]amino}methyl)quinolin-2-yl]piperidin-3-ol
2-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]pyrido[2,3-d]pyrimidin-4-amine
3-{3-[cyclohexyl(methyl)amino]propyl}-8-[(2R)-pyrrolidine-2-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-(1,3-benzothiazol-2-yl)-4-(3-fluorobenzenesulfonyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(3-methoxyphenyl)methyl]-3-(1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)propanamide
2-methyl-6-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1,3-benzoxazole
2-(1-butyl-1H-pyrazol-4-yl)-N-methyl-N-(propan-2-yl)quinoline-4-carboxamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(1H-imidazol-2-ylmethyl)pyrrolidine-3-carboxylic acid
4-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-amine
N-(3-cyano-4-methylphenyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carboxamide
1-acetyl-N-{[1-(cyclohex-2-en-1-yl)-1,2,3,6-tetrahydropyridin-4-yl]methyl}piperidine-4-carboxamide
3-{2-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-[(2-fluorophenyl)methyl]piperazin-2-one
(3S,9aR)-3-ethyl-8-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-{4-[2-(3-chlorophenoxy)propanoyl]piperazin-1-yl}-1,2-dihydropyrazin-2-one
2-(2-aminoethyl)-N-[2-(diethylamino)-2-(furan-2-yl)ethyl]quinazolin-4-amine
N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-4-(pyrimidin-2-yl)-1,4-diazepane-1-carboxamide
2-[(3S,4R)-3-acetamido-4-(propan-2-yl)pyrrolidin-1-yl]-6-phenylpyridine-3-carboxylic acid
5-cyclopropyl-N-{[2-(diethylamino)pyridin-3-yl]methyl}-1,3-oxazole-4-carboxamide
N-[4-({[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]carbamoyl}methoxy)phenyl]propanamide
6-(3-chloro-4-methylbenzoyl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine