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(3R,4R)-1-[(5-ethylfuran-2-yl)methyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
2-{[(2-methylphenyl)methyl]sulfanyl}-N4-[2-(pyrazin-2-yl)ethyl]pyrimidine-4,6-diamine
2-(propan-2-yl)-N-[2-(pyrazin-2-yl)ethyl]-1,3-benzoxazole-5-carboxamide
2-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-[methyl(2-phenylethyl)amino]-2,3-dihydropyridazin-3-one
4-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidine-1-carbonyl]-1-ethyl-1,2-dihydropyridin-2-one
5-(methoxymethyl)-N-[(7-{[4-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]furan-2-carboxamide
1-{2-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-4-methylpyrimidin-5-yl}ethan-1-one
5-[(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]-N,N-dimethylpyridin-2-amine
N-[(2R,3R)-2-methoxy-1'-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-3-carboxamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-[(5-phenylthiophen-2-yl)methyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
(3S,7S)-5-[3-(dimethylamino)-1,2,4-thiadiazol-5-yl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}(methyl){[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
7-(2-propoxypropanoyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-[3-methyl-1-(propan-2-yl)-1H-pyrazol-5-yl]urea
3-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}benzonitrile
3-{4-[(2E)-3-(5-chloro-2-hydroxyphenyl)-2-methylprop-2-en-1-yl]piperazin-1-yl}pyrazine-2-carbonitrile
N-[2-(1H-pyrazol-1-yl)ethyl]quinoline-2-carboxamide
{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(isoquinolin-5-ylmethyl)methylamine
methyl 1-{9-methoxy-3-[(4-methylphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}piperidine-2-carboxylate
N-(3-chloro-4-methoxyphenyl)-3-[1-(3-methylfuran-2-carbonyl)piperidin-3-yl]propanamide
2-(2-{[5-(2-methylphenyl)-1,2,4-triazin-3-yl]amino}ethyl)-6-phenyl-2,3-dihydropyridazin-3-one
2-{1-[1-(4-fluorophenyl)cyclopropanecarbonyl]pyrrolidin-2-yl}pyridine
1-(2-methoxybenzoyl)-4-(oxolane-3-carbonyl)piperazine
3-(4-{[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenyl)prop-2-yn-1-ol
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-2-(1H-imidazol-2-yl)benzamide
5-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-2-methyl-3,4-dihydropyrimidin-4-one
1-tert-butyl-N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-5-oxopyrrolidine-3-carboxamide
(3S,4S)-1-(4,6-dimethylquinolin-2-yl)-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
(3S,7S,8aS)-7-[(1-benzothiophen-2-ylmethyl)amino]-3-(1H-indol-3-ylmethyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-({4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)pyridine
3-[(diethylamino)methyl]-1-(2,2-dimethylpropyl)-3-hydroxypiperidin-2-one
1-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
2-methoxy-N-[3-(4-{[1-(2-methyl-1,3-thiazol-4-yl)ethyl]amino}piperidin-1-yl)phenyl]benzamide
(4aR,7aS)-1-ethyl-4-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[2-(pyrrolidin-1-yl)benzoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-[(1S,3S)-3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}cyclopentyl]pyridine-3-carboxamide
{[2-(piperidin-1-yl)-2,3-dihydro-1H-inden-2-yl]methyl}({[4-(pyrimidin-2-yloxy)phenyl]methyl})amine
3-({1-[(2-chloro-6-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}methyl)morpholine
2-{[3-cyclopropyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,3-benzoxazole
2-[3-(3-methyl-3-phenylpiperidin-1-yl)-3-oxopropyl]-2,3-dihydro-1H-isoindol-1-one
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
{1-[4-(hydroxymethyl)cyclohexanecarbonyl]-3-(3-methylbut-2-en-1-yl)piperidin-3-yl}methanol
5-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-5-(2-phenylethyl)imidazolidine-2,4-dione
4-[(3S,5R)-5-[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine-1-carbonyl]piperidine-3-carbonyl]morpholine
ethyl 4-[(2S,4R)-4-amino-2-(methylcarbamoyl)pyrrolidin-1-yl]piperidine-1-carboxylate
5-[(E)-2-phenylethenyl]-2,3-dihydro-1H-indol-2-one
methyl 6-butanoyl-2-{[(3-fluorophenyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-[(4-fluorophenyl)methyl]-5-(3-methylfuran-2-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole
3-methyl-7-{[4-(2-methylpropyl)phenyl]methyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one