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1-[(3S,4R)-4-amino-3-methoxypiperidin-1-yl]-2-(2-ethyl-1H-imidazol-1-yl)ethan-1-one
1-benzyl-N-({5-methyl-2-[3-(2-methylfuran-3-amido)phenyl]-1,3-oxazol-4-yl}methyl)-1H-pyrazole-4-carboxamide
2-(cyclopropylmethyl)-7-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
6-fluoro-N-methyl-N-[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
2-ethyl-5-(3-{[4-(pyridin-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)pyrimidine
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-2-(dimethylamino)-2-(4-fluorophenyl)acetamide
3-cyclopropaneamido-4-methyl-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}benzamide
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]pyrimidin-4-amine
3-[(4-methoxyphenyl)methyl]-3,4-dihydropteridin-4-one
3-[(1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-1H-1,2,3-triazol-4-yl)methyl]-2,3-dihydro-1,3-benzoxazol-2-one
N-[(3S)-2-oxoazepan-3-yl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-{1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-fluorobenzamide
1-benzyl-4-[2-(phenylsulfanyl)acetyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-7-fluoro-3-methyl-1H-indole-2-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(cyclopentylmethyl)piperidin-3-ol
1-ethyl-N,5-dimethyl-N-[1-(pyridin-3-yl)pentyl]-1H-pyrazole-4-carboxamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}propan-1-one
1-{[5-(hydroxymethyl)furan-2-yl]methyl}-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
({5-[1-(1-benzofuran-5-ylmethyl)piperidin-4-yl]-4-cyclopropyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
1-[5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]-4,4-dimethylpiperidine
2-[(3,5-difluorophenyl)methyl]-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N-methyl-2-(1H-pyrazol-1-yl)benzamide
N,N,3,6-tetramethyl-2-(2-phenylpyrimidin-5-yl)quinoline-4-carboxamide
3-(4-chloro-2-methylbenzoyl)-1-[4-(methylsulfanyl)benzoyl]piperidine
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2-(2-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
(1S,9R)-11-{6-[(thiophen-2-ylmethyl)amino]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
8-[(2-methoxyphenyl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[4-(3,5-dichloro-4-methylbenzoyl)-1-methylpiperazin-2-yl]ethan-1-ol
6-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3-({[(5-chlorothiophen-2-yl)methyl]amino}methyl)-N,N-diethylpyridin-2-amine
N-(1-cycloheptylpiperidin-3-yl)-1-ethyl-5-methyl-1H-pyrazole-4-sulfonamide
N-[1-(1-cyclopropanecarbonylpiperidin-4-yl)-1H-pyrazol-5-yl]-2-methoxybenzamide
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-2-{7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}ethan-1-one
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]acetamide
2-hydroxy-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)pyridine-3-carboxamide
N-methyl-4-sulfamoyl-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]benzamide
(2E)-N-{3-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}-3-(thiophen-2-yl)prop-2-enamide
N,N-dimethyl-1-[2-(phenylamino)pyrimidine-5-carbonyl]azepan-4-amine
N-(3-cyclopentaneamidophenyl)-3-methoxypiperidine-1-carboxamide
2-[4-(1H-indol-3-ylmethyl)-1-(3-methylbut-2-en-1-yl)piperazin-2-yl]ethan-1-ol
3-methoxy-1-(2-{2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydropyridin-2-one
N-[(3S,4S)-1-ethyl-4-methoxypyrrolidin-3-yl]-2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carboxamide
1-methyl-2-(5-{1-[1-(pyrimidin-4-yl)ethyl]-1H-imidazol-2-yl}furan-2-yl)-1H-1,3-benzodiazole
2-methyl-5-{[3-(2-phenylethyl)piperidin-1-yl]methyl}-[1,2,4]triazolo[1,5-a]pyrimidin-7-ol
4-(2-{1-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]piperidin-2-yl}ethyl)morpholine
1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-3-[2-(methylsulfanyl)benzoyl]piperidine
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-{[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}hexanamide
methyl (2S,4S,5R)-5-(2,3-difluorophenyl)-1-methyl-4-[(pyridin-3-ylmethyl)carbamoyl]pyrrolidine-2-carboxylate