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1-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(3-methoxypropyl)piperidine
1-(2,3-dihydro-1H-inden-2-yl)-N-methyl-N-[(1-propyl-1H-imidazol-2-yl)methyl]piperidin-3-amine
N-methyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-ethyl-N-(pyridin-4-ylmethyl)acetamide
1-[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(thiophen-3-yl)ethan-1-one
2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-methyl-N-(pyridin-2-ylmethyl)-1,3-oxazole-4-carboxamide
1-ethyl-3-methyl-8-[(3-methylthiophen-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
5-fluoro-2-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridine
5-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-(2,4-difluorophenyl)-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepine
3-(3-methoxyphenoxy)-N-(3-methyl-1,2,4-thiadiazol-5-yl)azetidine-1-carboxamide
(3S,4S)-1-(1-cyclopentylpiperidine-4-carbonyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
N-cyclobutyl-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
3-(4-methoxyphenyl)-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-3-phenylpropanamide
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
1-{2-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
(2S)-1-{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxamide
1-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-2-methyl-3-(1H-pyrazol-1-yl)propan-1-one
2-(3-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]-1H-pyrazol-3-yl}phenyl)-N,N-dimethylbenzamide
N-{[7-(2,3-difluorobenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-3-sulfonamide
1-cyclohexyl-3-(cyclopropylmethyl)-5-(4-ethylpiperazine-1-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-(1-{[(2,2-diphenylethyl)carbamoyl]methyl}-1H-pyrazol-4-yl)furan-2-carboxamide
N-[2-(4-methyl-1H-imidazol-2-yl)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
2-[2-(1H-imidazol-4-yl)ethyl]-9-[2-(2-methylphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[1-(6-methylpyridin-2-yl)propyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-fluoro-6-(2-methylquinolin-5-yl)benzamide
2-{5-[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
4-[(4-fluorophenyl)methyl]-1-(piperidine-1-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
(1R,5S,8S)-8-methoxy-3-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-3-azabicyclo[3.2.1]octane
[(3-methoxyphenyl)methyl](methyl)({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amine
1-[(3aR,6aR)-2-cyclopropanecarbonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]-4-(propan-2-yl)-1,4-diazepane
2-hydroxy-N-[(3R,4R)-3-hydroxypiperidin-4-yl]-4-methoxybenzamide
1-[(4aR,8aR)-6-(thiophen-2-ylmethyl)-decahydro-1,6-naphthyridin-1-yl]-2-(2-methylphenyl)ethan-1-one
7-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
(1R,5R)-3-{5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
2-[4-methoxy-2-methyl-5-(propan-2-yl)phenyl]-1H-imidazole
(4aR,8aS)-6-{[3-(2-methylphenyl)phenyl]methyl}-1-(pyridin-3-ylmethyl)-decahydro-1,6-naphthyridin-2-one
1-[4-(4-{[(2,5-dimethoxyphenyl)methyl]amino}piperidin-1-yl)benzoyl]piperidin-3-ol
2-cyclopropyl-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1,3-benzoxazole-6-carboxamide
(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)(methyl)({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
N-[(3-chloro-1-benzothiophen-2-yl)methyl]-N-methyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](ethyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
4-ethyl-1-methyl-3-(1-{[4-(pyrrolidin-1-yl)phenyl]methyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-methyl-8-[(1-methyl-1H-imidazol-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxylic acid
1-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(4-fluoro-3-methylphenyl)ethan-1-one
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
4-methyl-3-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridine
5-(1H-1,3-benzodiazol-2-ylmethyl)-N-(2-methoxyethyl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-N-[2-(1H-imidazol-4-yl)ethyl]pyridine-2-carboxamide