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2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-[1-(pyridin-4-yl)propyl]benzamide
2,2,2-trifluoro-1-[4-(pyrimidin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
(2S,4R)-4-amino-N-ethyl-1-[2-(1,1,2,2-tetrafluoroethoxy)benzoyl]pyrrolidine-2-carboxamide
1-cyclopentanecarbonyl-N-[2-(pyridin-3-yl)ethyl]piperidine-4-carboxamide
3-{1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]pyrrolidin-2-yl}pyridine
1-ethyl-5-oxo-N-[(4-phenylphenyl)methyl]pyrrolidine-3-carboxamide
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(4-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)acetic acid
(2E)-3-(3-fluorophenyl)-1-{4-[4-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]piperidin-1-yl}prop-2-en-1-one
2-(4-{[2-(4-methoxyphenyl)imidazo[1,2-a]pyridin-3-yl]methyl}morpholin-3-yl)acetamide
(3S,4R)-1-[(5-ethylpyridin-2-yl)methyl]-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
2-(morpholin-4-ylmethyl)-N-(2,3,5-trifluorophenyl)-1,4-oxazepane-4-carboxamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]acetamide
1-methyl-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-4-ylmethyl)piperidin-4-amine
(3R,5R)-N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
2-[(5-methylpyrazin-2-yl)methyl]-9-[5-(propan-2-yl)pyrimidin-4-yl]-2,9-diazaspiro[5.5]undecan-3-one
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-4-(1H-pyrazol-4-yl)butanamide
6-(isoquinolin-5-yl)pyridine-2-carboxamide
2-ethyl-N-[1-(3,4,5-trimethoxyphenyl)ethyl]pyrimidine-5-carboxamide
3-({cyclohexyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)pyrrolidin-3-ol
5-(azepane-1-carbonyl)-1-(butan-2-yl)-N-[2-(2-methoxyphenyl)ethyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
3-(3-chloro-4-methylphenyl)-5-[(R)-methoxy(phenyl)methyl]-1,2,4-oxadiazole
3-{[({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)carbamoyl]methyl}-1,2,3-oxadiazol-3-ium-5-olate
2,2-dimethyl-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]oxane-4-carboxamide
2-methyl-5-[2-(pyridin-4-yl)-1H-imidazol-1-yl]phenol
3-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenol
5-{2-azaspiro[4.4]nonane-2-carbonyl}-1-(2-ethoxyethyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]acetamide
1-[3-(4-fluorophenyl)-1-methyl-1H-1,2,4-triazol-5-yl]piperidine
N-[3-(3-chlorophenyl)phenyl]-2-(2-methoxyethyl)morpholine-4-carboxamide
3-{[(4-fluorophenyl)methyl]sulfanyl}-N-[2-(methylsulfamoyl)ethyl]propanamide
2,5-dimethyl-3-{4-[3-(2-phenylpropyl)-1,2-oxazole-5-carbonyl]piperazin-1-yl}pyrazine
({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)(methyl)(pyridin-2-ylmethyl)amine
8-[5-(methoxymethyl)thiophene-2-carbonyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[(3S,4R)-4-amino-1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}pyrrolidin-3-yl]ethan-1-ol
4-(1-ethyl-5-oxopyrrolidine-3-carbonyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
3-{[(2H-1,3-benzodioxol-5-ylmethyl)(methyl)amino]methyl}-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
ethyl 4-(3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)piperazine-1-carboxylate
N-({4-[(3,5-dimethoxyphenyl)methoxy]phenyl}methyl)-5-methyl-N-[(3S)-2-oxoazepan-3-yl]thiophene-2-carboxamide
9-[2-(4-methylphenyl)acetyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
[1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidin-3-yl]methanol
2-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-6-(5-methylthiophen-2-yl)pyridine-3-carboxylic acid
6-(2-hydroxyethyl)-N-(2-methylpropyl)-N-[(3-methylthiophen-2-yl)methyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
(3R,4S)-1-(azepane-1-sulfonyl)-N,N-dimethyl-4-(5-methylfuran-2-yl)pyrrolidin-3-amine
N-(2-methoxyethyl)-N-methyl-3-{4-[2-(3-methylphenyl)acetamido]-1H-pyrazol-1-yl}benzamide
4-(1H-imidazol-1-ylmethyl)-5-methyl-2-(naphthalen-2-yl)-1,3-oxazole
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-6-methylpyridazin-3-amine
N-ethyl-1-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]-N-(pyridin-4-ylmethyl)piperidin-3-amine
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1-methyl-1H-imidazole-4-sulfonamide