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5-{1-[2-(cyclohex-1-en-1-yl)ethyl]-1H-1,2,3-triazol-4-yl}pyrimidine
1-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
1-(1H-imidazol-2-ylmethyl)-4-phenylazepane
N-[(3R,4S)-4-cyclopropyl-1-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]pyrrolidin-3-yl]-2-ethoxyacetamide
(4aS,7aR)-1-[(6-chloro-2-fluoro-3-methylphenyl)methyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-{[3-(2-chlorophenyl)-1,2-oxazol-5-yl]methyl}-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
(9aR)-2-methyl-8-[(4-methylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(4aS,8aR)-1-(2-aminoethyl)-6-(quinoline-8-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-cyclopropyl-N-[(4-ethoxyphenyl)methyl]-2-[methyl(pyridin-3-ylmethyl)amino]acetamide
N-(1,1-dioxo-1λ6-thian-4-yl)-N-methyl-2-(naphthalen-2-yloxy)propanamide
1-(2,5-dimethylfuran-3-carbonyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
1-(2-methylphenyl)-4-(pyridine-3-carbonyl)-1,4-diazepane
N-cyclopropyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-propyl-1,3-oxazole-4-carboxamide
2-[(1-methylpiperidin-4-yl)(2-phenylethyl)amino]-1-(morpholin-4-yl)ethan-1-one
8-methoxy-3-{2-[1-(propan-2-yl)piperidin-2-yl]ethyl}-3,4-dihydroquinazolin-4-one
1-(4-acetyl-4-phenylpiperidin-1-yl)-4,4,4-trifluorobutan-1-one
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-{[butyl(methyl)amino]methyl}-7-methyl-1-(pyridin-2-ylmethyl)-1,2-dihydroquinolin-2-one
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-{[(3-ethoxy-4-methoxyphenyl)methyl]amino}-N-[2-(2-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
5-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-yl]-3-(2-phenylethyl)-1H-1,2,4-triazole
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-cyclopropyl-1-[(2,5-dimethylphenyl)methyl]pyrrolidine-2-carboxamide
3-(1H-1,3-benzodiazol-2-yl)-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}propan-1-one
4-(4-methoxyphenoxy)-1-[2-(2-methyl-1,3-thiazol-4-yl)ethyl]piperidine
N-(1H-indol-4-ylmethyl)-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propanamide
3-{2-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]ethyl}-1λ6-thiolane-1,1-dione
N-[(3-chlorophenyl)methyl]-3-[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]propanamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)benzamide
1-methyl-N-[(3-methylquinoxalin-2-yl)methyl]-N-(pyridin-4-ylmethyl)piperidin-4-amine
5-[2-chloro-5-(1H-pyrazol-1-yl)phenyl]-3-cyclopropyl-1H-1,2,4-triazole
1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(2-methyl-1H-imidazol-1-yl)propan-1-one
1-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]-4-(1H-pyrazol-1-yl)butan-1-one
1-[(4-fluorophenyl)methyl]-4-[2-(pyrrolidin-1-yl)benzoyl]-1,4-diazepane
2-{4-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperazin-1-yl}phenol
6-fluoro-2-oxo-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
4-(1-methyl-1H-imidazol-2-yl)-1-[(4-phenyl-1,3-thiazol-5-yl)methyl]-1H-1,2,3-triazole
3-[8-(3-fluoro-4-methoxybenzoyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl]propanoic acid
(2S)-4-methyl-2-(propan-2-yl)-1-[3-(pyridin-4-yl)propyl]piperazine
4-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N,N-dimethylbenzamide
2-benzyl-5-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1,3-benzoxazole
N-[2-(dimethylamino)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(2E)-N-ethyl-3-(furan-2-yl)-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)prop-2-enamide
9-(3-ethoxypropanoyl)-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
(1S,5R)-6-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
8-[(2-ethylphenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
pyridin-3-yl({1-[6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-4-yl})methanol
3-[(dimethylamino)methyl]-1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]pyrrolidin-3-ol
1-(3-phenyl-1,2,4-oxadiazol-5-yl)-4-(thiophen-2-ylmethyl)-1,4-diazepane
N3-tert-butyl-N5-[(1R)-1-(4-methoxyphenyl)ethyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[2-(2-methylpropanesulfonyl)ethyl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide