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4-(4-acetamido-1H-pyrazol-1-yl)-N-{[4-(trifluoromethoxy)phenyl]methyl}benzamide
N-{[1-(2-methoxypyridine-3-carbonyl)piperidin-3-yl]methyl}-1H-indole-2-carboxamide
9-(4-chloro-2-fluorobenzoyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane
4-(cyclopropylmethyl)-1-[(4-methoxy-3-methylphenyl)methyl]-1,4-diazepan-5-one
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
2-{4-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidine-1-carbonyl]piperidin-1-yl}acetamide
3-(pyridin-3-yl)-7-thia-2,4,5-triazatricyclo[6.4.0.02,6]dodeca-1(12),3,5,8,10-pentaene
3-[1-(6,7-diethoxy-3-methyl-1-benzofuran-2-carbonyl)piperidin-3-yl]propanamide
methyl 1-[(3S,5S)-1-(3-methylbut-2-en-1-yl)-5-[(quinolin-2-ylmethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
4-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]-N-[2-(methylsulfanyl)phenyl]-4-oxobutanamide
2-cyclopentyl-9-(3-fluoropyridine-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[2-(benzenesulfonyl)ethyl]-5-methyl-1-(4-methylphenyl)piperazin-2-one
N,N-dimethyl-5-({methyl[(3-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)pyrimidin-2-amine
1-cyclopentyl-4-[({6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}(methyl)amino)methyl]pyrrolidin-2-one
1-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethan-1-one
3-[2-(dimethylamino)ethyl]-5-[1-(3-fluorobenzoyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
1-{5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1H-pyrazole-3-carbonyl}-3-ethylpiperazine
7-(1-benzothiophen-3-yl)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[3-(4-phenylbenzoyl)piperidine-1-carbonyl]pyridin-1-ium-1-olate
methyl (2S)-1-[2-(4-{4-[4-(morpholin-4-yl)piperidin-1-yl]piperidin-1-yl}phenyl)acetyl]pyrrolidine-2-carboxylate
1-{2-[1-(2,3-dihydro-1H-inden-5-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,2,3,4-tetrazole
3-(1H-1,2,3-benzotriazol-5-yl)-1-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}urea
{2-oxo-2-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethyl}urea
(3aR,6aR)-2-cyclopentyl-N-[2-(2-hydroxyethoxy)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
6-{3-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-3-oxopropyl}-2,3-dihydropyridazin-3-one
3-(4-methyl-1H-pyrazol-1-yl)-1-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
3-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-3,9-diazaspiro[5.5]undecane
2-[3-(2-methoxybenzoyl)piperidine-1-carbonyl]-N,N-dimethylaniline
1-{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}-3-(methoxymethyl)piperidine
4-(1-{5-[2-(piperidin-1-yl)-2,3-dihydro-1H-inden-2-yl]-1,2,4-oxadiazol-3-yl}ethyl)morpholine
1-[(2,3-difluorophenyl)methyl]-3-{[(1,3-dihydroxy-2-methylpropan-2-yl)amino]methyl}-3-hydroxypiperidin-2-one
(2R)-2-amino-3-phenyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)propanamide
N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazin-3-amine
N-{1-[(3-chlorophenyl)methyl]-1H-pyrazol-5-yl}-2-(2,5-dioxoimidazolidin-1-yl)acetamide
1-(2,3-dimethyl-1H-indole-7-carbonyl)-4-phenylpiperidine-4-carbonitrile
3-[2-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)ethyl]-2,3-dihydro-1,3-benzoxazol-2-one
(3R,5S)-N-{[3-(methylsulfanyl)phenyl]methyl}-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
1-[1-(1-methylcyclopropanecarbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
(1R,3S)-3-methoxy-7-(2-methoxypyridine-4-carbonyl)-7-azaspiro[3.5]nonan-1-ol
3-{2-[4-(1-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
(4aS,7aR)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-[2-amino-4-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-2,2-dimethyl-3,4-dihydro-2H-pyran-4-one
(1H-imidazol-4-ylmethyl)({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)methylamine
N-(5-hydroxyadamantan-2-yl)-3-(2-phenylethyl)-1,2-oxazole-5-carboxamide
1-methyl-3-{[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
3-{2-oxo-2-[4-(oxolane-2-carbonyl)-1,4-diazepan-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
[1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)piperidin-4-yl](thiophen-2-yl)methanol
2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]-1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}ethan-1-one
2-[2-({[3-(1H-pyrazol-1-yl)phenyl]methyl}amino)pyrimidin-4-yl]pyridine-4-carboxylic acid