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N-[(2,6-difluoro-3-methoxyphenyl)methyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
1,3,5-trimethyl-7-[2-methyl-6-(piperidin-3-yl)pyrimidin-4-yl]-3,7-diazabicyclo[3.3.1]nonan-9-ol
2-(ethoxymethyl)-N-methyl-N-(thiophen-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
ethyl 1-(butylcarbamoyl)-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
(1S,5R)-6-(cyclobutylmethyl)-3-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3,6-diazabicyclo[3.2.2]nonane
6-[(diethylamino)methyl]-N-[2-(methylsulfamoyl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-(2-chloro-3,4-dimethoxyphenyl)-7-hydroxy-6-methyl-1,2,3,4-tetrahydroquinolin-2-one
{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[2-(trifluoromethyl)phenyl]methyl})amine
2-methoxy-5-[2-(oxolan-3-yl)-1H-imidazol-1-yl]pyridine
3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-(2-phenylethyl)propanamide
(3aS,7aR)-5-methyl-2-(2-methyl-1,3-benzothiazole-6-carbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
methyl 3-[(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)carbamoyl]propanoate
5-tert-butyl-4-{[7-(2-hydroxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]methyl}furan-2-carboxamide
N-(3-chlorophenyl)-4-[3-methyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]butanamide
N-[(2R,3R)-1'-[(3-ethoxy-2-hydroxyphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
2-methyl-N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-1,3-thiazole-4-carboxamide
1-[(2-ethyl-1,3-thiazol-4-yl)methyl]-3-propylpiperidine-3-carboxylic acid
3-(6-methoxynaphthalene-2-carbonyl)-N,N-dimethylpiperidine-1-sulfonamide
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl](methyl)[(1-phenylpyrrolidin-3-yl)methyl]amine
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-ethyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1H-pyrazole-3-carboxamide
3-methyl-N-[2-(7-methyl-1H-indol-3-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-methyl-1,2,3,6-tetrahydropyridine
1-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carbonyl]-4-methanesulfonyl-1,4-diazepane
5-[2-(4-fluorophenyl)piperidine-1-carbonyl]-2-methylphenol
N,1,3-trimethyl-N-(1-{1-[(3-methylphenyl)methyl]piperidin-4-yl}-2-phenylethyl)-1H-pyrazole-5-carboxamide
8-(2,6-dimethylhept-5-en-1-yl)-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-amino-1-{4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methylpropan-1-one
N-({2-[2-(2-cyclopentylacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
3-{2-[4-(3-chlorophenyl)piperazin-1-yl]-2-oxoethyl}-4-cyclopentylpiperazin-2-one
3-{[1-(4-chlorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}-3,4-dihydro-1,2,3-benzotriazin-4-one
N-(2-methoxyethyl)-4-methyl-3-{[methyl(2-methylprop-2-en-1-yl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
ethyl 1-(4-phenyl-1,3-thiazol-2-yl)-5-({[(1r,4r)-4-hydroxycyclohexyl]amino}methyl)-1H-pyrazole-4-carboxylate
3-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-8-methoxy-3,4-dihydroquinazolin-4-one
6-oxo-1-(3-phenylpropyl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-3-carboxamide
2-[({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]phenol
2-methyl-5-(2-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}-2-oxoethyl)-3,4-dihydropyrimidin-4-one
N-(5-aminopentyl)-3-(azocan-1-yl)propanamide
3-(4-tert-butylbenzoyl)-1-cyclobutylpiperidine
N-({1-[6-(azepan-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-3-yl}methyl)acetamide
3-{2-[4-(naphthalen-1-yl)piperazin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(1H-1,2,4-triazol-1-yl)propanamide
4-[(4-methyl-5-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]morpholine
{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)methylamine
4-amino-2-{4-[(8-hydroxyquinolin-2-yl)methyl]piperazin-1-yl}pyrimidine-5-carbonitrile
2-hydroxy-N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
2-(1H-pyrazol-1-yl)-N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)acetamide
1-[2-(dimethylamino)-2-(2-methylphenyl)acetamido]cyclopentane-1-carboxylic acid
2-methyl-4-phenyl-N-[1-(pyrazin-2-yl)propan-2-yl]-1,3-thiazole-5-carboxamide
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide