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3-(4-fluorophenyl)-4-[1-(2-methoxyacetyl)piperidine-4-carbonyl]piperazin-2-one
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-1-[2-(dimethylamino)ethyl]-5-oxopyrrolidine-3-carboxamide
5-methyl-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
(cyclopropylmethyl)({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)propylamine
N-(2-methylpropyl)-2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}acetamide
7-(2-methyl-1H-1,3-benzodiazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
(3S,4R)-1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
methyl (2S,4S)-1-[(2-chloro-6-fluorophenyl)methyl]-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzamido]pyrrolidine-2-carboxylate
N-[(3-hydroxy-4-methoxyphenyl)methyl]-N-methyl-5-[(methylsulfanyl)methyl]furan-2-carboxamide
N-(pyridin-2-ylmethyl)-5-(pyridine-3-sulfonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-tert-butyl-4-hydroxy-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)pyrimidine-5-carboxamide
1-(cyclobutylmethyl)-3-hydroxy-3-({methyl[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}methyl)piperidin-2-one
methyl({[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}){[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}amine
N-cyclobutyl-4-{[(3R)-piperidin-3-yl]sulfamoyl}benzamide
4-(1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)morpholine
1-(1,3-benzothiazole-6-carbonyl)-N,N-dimethylazepan-4-amine
[1-(1H-imidazol-2-ylmethyl)-3-(2-methylpropyl)piperidin-3-yl]methanol
3-(oxolan-2-ylmethyl)-5-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
1-(difluoromethyl)-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-1H-pyrazole-5-carboxamide
1-(2-hydroxyethyl)-5-(3-methoxy-5-methylthiophene-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
5-ethyl-N-{[5-(3-methoxyphenyl)-1,2-oxazol-3-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)[(5-ethylpyridin-2-yl)methyl]methylamine
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-3-(1H-pyrazol-1-yl)benzamide
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]({[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
3-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-N,N-dimethylpropane-1-sulfonamide
1-(2-phenylethyl)-N-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H-1,2,3-triazole-4-carboxamide
4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidine
9-(2,4-difluorobenzoyl)-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-ol
1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}-3-(pyridin-2-yl)propan-1-one
3-methyl-4-(1-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-1,2,5-oxadiazole
4-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidine-4-carbonyl}-1,4-oxazepan-6-ol
1-{[4-(2,2-dimethylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}-4-(pyridin-3-yl)piperidin-4-ol
{4-[(4-chlorophenyl)methyl]-1-(oxan-4-yl)piperidin-4-yl}methanol
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-5,6-dimethylthieno[2,3-d]pyrimidin-4-amine
N-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
ethyl 4-[2-(dimethylamino)-2-(3-fluorophenyl)acetamido]piperidine-1-carboxylate
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-methyl-1,2-oxazole-3-carboxamide
5-[(4-fluorophenyl)methyl]-3-(2-methoxyethyl)-5-{1-[4-(1H-pyrazol-1-yl)butan-2-yl]piperidin-4-yl}imidazolidine-2,4-dione
3-(azocan-1-yl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}propanamide
2-(4-ethoxyphenoxymethyl)-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidine
(5S,9aS,9bS)-2-cyclopentyl-5-(3,5-dimethoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
5-[(3-hydroxypiperidin-1-yl)methyl]-N-[2-methyl-1-(pyrrolidin-1-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
1-[1'-(4-fluoro-3-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
1-[2-(2,3-difluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-3-methylpiperidine
1-(3-{2-ethyl-3H-imidazo[4,5-b]pyridin-6-yl}benzoyl)-4-methylpiperidine
(3S)-3-ethyl-4-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)morpholine
3-[(1-carbamoylpentyl)sulfamoyl]-N-cyclobutylbenzamide