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(2S)-1-[2-(pyridin-3-yloxy)acetyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
2-methyl-3-oxo-N-[4-(trifluoromethyl)phenyl]-2,9-diazaspiro[5.5]undecane-9-carboxamide
4-chloro-2-{[9-methoxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenol
methyl 2-(1-{[6-chloro-4-(morpholin-4-yl)quinazolin-2-yl]methyl}-3-oxopiperazin-2-yl)acetate
1-(5-chloro-3-methyl-1H-indole-2-carbonyl)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)piperidin-3-amine
3-[methyl({[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl})amino]propanamide
1-tert-butyl-3-(oxan-4-yl)-5-[(2-phenyl-1H-imidazol-1-yl)methyl]-1H-1,2,4-triazole
2-(pyridin-2-yl)-1-[3-(pyridine-2-carbonyl)piperidin-1-yl]ethan-1-one
N-cyclohexyl-1-{2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methylpiperidine-3-carboxamide
5-(2-fluorophenoxymethyl)-N-[2-(oxan-2-yl)ethyl]-1H-pyrazole-3-carboxamide
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-(2-methoxyethyl)benzamide
1-[2,3-dimethyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-[2-(ethylsulfanyl)ethyl]urea
methyl 6-{[3-(2-hydroxyethoxy)phenyl]methyl}-2-[(3-methylbutyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N,N-dimethylbenzamide
(5S,9aS,9bS)-2-(2-methoxyphenyl)-5-(quinolin-5-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
5-oxo-1-(pyridin-2-ylmethyl)-N-[2-(1H-pyrrol-1-yl)ethyl]pyrrolidine-3-carboxamide
9-(2-methoxy-3-methylbenzoyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
(1R,6S)-9-methyl-3-[6-(4H-1,2,4-triazol-4-yl)pyridine-2-carbonyl]-3,9-diazabicyclo[4.2.1]nonane
3-{4-[1-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}benzonitrile
2-[4-(2-ethoxyphenyl)phenyl]acetamide
4-[4-(azepane-1-carbonyl)piperidin-1-yl]-2-[(4-methoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
2-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-N-methylpyridine-3-carboxamide
8-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
N-(3-methyl-1,2,4-thiadiazol-5-yl)-4-(pyridin-2-yl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carboxamide
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-[(3-methylthiophen-2-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-(1,3-thiazol-5-yl)ethan-1-one
4-(3-methoxypropyl)-1-{[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl}piperidine
(4aS,8aR)-6-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-decahydro-1,6-naphthyridine-4a-carboxylic acid
3-(4-methylphenyl)-N-[2-(thiophene-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]propanamide
N-(2-methylquinolin-5-yl)-4-(pyridin-3-ylmethoxy)piperidine-1-carboxamide
4-(4-methoxyphenyl)-3-(1H-pyrazol-1-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(3-chloro-1,2-oxazol-5-yl)-1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]propan-1-one
1-(2-methoxybenzoyl)-4-[1-(2-methoxyethyl)pyrrolidine-3-carbonyl]piperazine
2-[(4-benzylpiperazin-1-yl)methyl]-N-methyl-N-(pyridin-3-ylmethyl)-1,3-oxazole-4-carboxamide
3-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-N-(4-methylphenyl)-3-oxopropanamide
4-ethyl-3-{1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(4aR,7aS)-1-acetyl-4-(3-phenylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-[(2-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
methyl 1-(6-methyl-2-oxo-1,2-dihydroquinoline-4-carbonyl)pyrrolidine-2-carboxylate
N-(3,5-dimethoxyphenyl)-3-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)propanamide
4-[4-(1H-imidazol-1-ylmethyl)phenyl]-1H-pyrazole
N-[2-(3-fluorophenyl)ethyl]-3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
4-[4-(2-chlorophenyl)-1H-1,2,3-triazol-1-yl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
2-[4-(5,6-dimethylpyridine-3-carbonyl)piperazin-1-yl]-4-phenylpyrimidine
N-(2-methoxyphenyl)-4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide
(3S,9aR)-8-(3-methylbenzoyl)-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
6-fluoro-2-oxo-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-(5-phenyl-1,3,4-thiadiazol-2-yl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]piperidin-4-amine
4-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-6-methylpyrimidin-2-amine