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1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}piperidine-3-carboxamide
propan-2-yl 4-chloro-3-(3-ethoxypropanamido)benzoate
2-[({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)amino]-4,6-dimethylpyridine-3-carbonitrile
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-{[3-(propan-2-yl)-4,5-dihydro-1,2-oxazol-5-yl]methyl}acetamide
1-(2,3-dihydro-1H-inden-2-yl)-3-[5-(2-phenylethyl)-1,3,4-thiadiazol-2-yl]urea
3-[2-(N-methylmethanesulfonamido)ethyl]-1-[2-(oxolan-2-ylmethoxy)phenyl]urea
2-(4-hydroxy-4-phenylpiperidin-1-yl)-2-[2-(propan-2-yloxy)phenyl]acetic acid
6-[(2,2-dimethylpropyl)amino]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
(2S,4S)-4-[4-({[(cyclohexylmethyl)carbamoyl](methyl)amino}methyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
ethyl 4-{[1-(4-benzenesulfonamidophenyl)piperidin-4-yl]amino}piperidine-1-carboxylate
1-(6,8-dimethoxy-4-methylquinolin-2-yl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2-methyl-3-(1H-pyrazol-1-yl)propanamide
2-propyl-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-1,3-thiazole-4-carboxamide
(3S,7S)-5-[2-(1H-imidazol-1-yl)acetyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-benzyl-N-methyl-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
N-(1-{7-[(4-methoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclopropanecarboxamide
2-{[(4aS,7aR)-4-(carboxymethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}-1,3-oxazole-4-carboxylic acid
1-[2-(azepan-1-yl)-2-oxo-1-phenylethyl]-4-butylpiperazine-2,3-dione
2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-1-[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]ethan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(2-phenylethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
N-(4-methylphenyl)-3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
7-(1-aminocyclobutanecarbonyl)-N,N-dimethyl-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-{[5-(2-methylprop-1-en-1-yl)-4-phenyl-1H-imidazol-1-yl]methyl}morpholine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(2-hydroxybutyl)-2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,3-oxazole-4-carboxamide
(3S,7S,8aS)-7-[({3-[(diethylamino)methyl]-4-methoxyphenyl}methyl)amino]-3-[(1R)-1-hydroxyethyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
(1S,5R)-1,3,3-trimethyl-N-[2-methyl-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-6-azabicyclo[3.2.1]octane-6-carboxamide
4-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-4H-1,2,4-triazole
4-(5-tert-butyl-1H-pyrazol-3-yl)-7-(2-oxoimidazolidin-1-yl)-1,2,3,4-tetrahydroquinolin-2-one
2-{8-[2-(1H-imidazol-4-yl)ethyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}acetic acid
N-cyclopentyl-1-(2-methylpropyl)-5-[3-(pyridin-2-yl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
6-(2-chlorophenyl)-N-(2,5-dihydroxy-2-methylpentyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
5-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)-1-{[3-(trifluoromethoxy)phenyl]methyl}pyrrolidin-2-one
1-ethyl-3-{2-[4-(2-hydroxyphenyl)piperazin-1-yl]-2-oxoethyl}-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
2-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-2,3-dihydro-1,2-benzothiazol-3-one
1-(8-fluoroquinoline-2-carbonyl)azetidine-2-carboxylic acid
3-[2-(azepan-1-yl)-2-oxoethyl]-4-[(2-methylphenyl)methyl]piperazin-2-one
(3S,4R)-1-[(8-chloroquinolin-2-yl)methyl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
N-(1H-1,2,3-benzotriazol-5-yl)azocane-1-carboxamide
2-(2-methoxyethyl)-N-[(3,4,5-trimethoxyphenyl)methyl]-1,3-benzoxazole-6-carboxamide
3-{[1-(2-phenylethyl)piperidin-4-yl]methyl}-1-(pyridin-3-yl)urea
5-(4-methanesulfonylphenyl)-1H-indazole
3-{5-[(2H-1,3-benzodioxol-5-yl)carbamoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-2-methylthieno[3,2-d]pyrimidin-4-amine
1-{[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-4-(hydroxymethyl)azepan-4-ol
2-[2-methyl-4-(4-methylphenyl)piperazin-1-yl]pyridine-4-carboxamide
6-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-3-(3,5-dimethyl-1H-pyrazol-4-yl)propan-1-one
5-(hydroxymethyl)-4-[(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)methyl]-2-methylpyridin-3-ol