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(butan-2-yl)(1H-imidazol-2-ylmethyl)(pyridin-4-ylmethyl)amine
2-(4-chlorophenyl)-7-(methylsulfanyl)-3-(morpholin-4-ylmethyl)quinoline
N-{[6-(3-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-3-fluoro-N-(2-methoxyethyl)benzamide
1-(5-ethyl-1,2,4-oxadiazol-3-yl)-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
N3-(3-ethoxypropyl)-N5-[(4-methylphenyl)methyl]-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-[2-(methylsulfamoyl)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-[1-(1-benzofuran-2-ylmethyl)piperidin-3-yl]-4-(4-fluorophenyl)piperazine
methyl (2S,4S,5R)-2-ethyl-4-[(1-hydroxy-2-methylpropan-2-yl)carbamoyl]-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylate
2-{[(2-hydroxyethyl)({[4-(methylsulfanyl)phenyl]methyl})amino]methyl}quinolin-8-ol
1-(2-fluorophenyl)-4-{4-[3-(methylsulfanyl)propyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}piperidin-4-ol
3-[2-(4-phenylpiperidin-1-yl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
propyl[(4-{1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)methyl]amine
3-(5-ethyl-1,3,4-thiadiazol-2-yl)-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]urea
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-1-[3-(pyridin-4-yl)azetidin-1-yl]ethan-1-one
N-benzyl{[2,3-dimethyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]amino}sulfonamide
N-{[2-(2,5-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(furan-2-ylmethyl)propanamide
1-(1-{[1-ethyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}-3,5-dimethyl-1H-pyrazol-4-yl)ethan-1-one
1-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-2-[4-(dimethylamino)phenyl]ethan-1-one
2-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-1-phenylethan-1-ol
2-{5-methyl-4-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]-2-oxopiperazin-1-yl}benzonitrile
1-(2-methoxy-4-{[methyl(oxan-4-yl)amino]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
methyl 2-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidine-1-carbonyl)benzoate
6-methoxy-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}pyrimidin-4-amine
1-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
2-(5-{[4-(dimethylamino)phenyl]methyl}-3-methyl-1H-1,2,4-triazol-1-yl)ethan-1-ol
1-[4-(3-acetylphenyl)phenyl]-3-[2-(dimethylamino)ethyl]-3-methylurea
N-[(2-chlorophenyl)methyl]-1-methyl-N-(propan-2-yl)pyrrolidine-3-carboxamide
(1R,5R)-6-benzyl-3-(5-methoxyfuran-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N'1-[3-methoxy-4-(3-methylbutanamido)phenyl]cyclopropane-1,1-dicarboxamide
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(3-methyl-1H-pyrazol-5-yl)methyl]amine
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-{2-[4-(1H-imidazol-1-yl)butoxy]phenyl}-1-methyl-1H-1,3-benzodiazole
N-{1-[(2-hydroxy-6-methoxyquinolin-3-yl)methyl]piperidin-4-yl}methanesulfonamide
1-{2-[(1-phenyl-1H-pyrazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-7-yl}propan-1-one
5-(4-methoxyphenyl)-N-[1-(pyridin-3-yl)propan-2-yl]-1,2,4-triazin-3-amine
1-[(3S,4R)-3-cyclopropyl-4-[(pyrimidin-2-yl)amino]pyrrolidin-1-yl]-4-(morpholin-4-yl)butan-1-one
6-[3-(5-fluoro-2-methoxybenzoyl)piperidine-1-carbonyl]-2,2-dimethyl-3,4-dihydro-2H-pyran-4-one
N-[2-(2-fluorophenyl)ethyl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
5-(3,4-difluorophenoxymethyl)-N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
2-({4-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethan-1-ol
4-ethyl-3-({1-[2-methyl-3-(1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(5-chloro-2-methoxyphenyl)-3-{1-[2-(1H-pyrazol-1-yl)acetyl]piperidin-3-yl}propanamide
5-(quinoxalin-2-yl)-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
N-methyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[(1-methylpiperidin-2-yl)methyl]-1,2-oxazole-3-carboxamide
6-{3-[2-(3-methoxyphenyl)ethyl]piperidine-1-carbonyl}-2-methyl-2,3,4,5-tetrahydropyridazin-3-one
6-{[(3S)-2-oxoazepan-3-yl]amino}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
N,2-dimethyl-N-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1-benzofuran-5-carboxamide
N-[(2,3-dimethylphenyl)methyl]-4-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
(1R,7S)-6-(azetidine-1-carbonyl)-3-[2-(piperidin-1-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
5-ethyl-5-{1-[4-(morpholin-4-yl)benzoyl]piperidin-4-yl}-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione